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FR23C1050I2 - Compose d'alkynylbenzene 3,5-disubstitue et un sel de celui-ci - Google Patents

Compose d'alkynylbenzene 3,5-disubstitue et un sel de celui-ci

Info

Publication number
FR23C1050I2
FR23C1050I2 FR23C1050C FR23C1050C FR23C1050I2 FR 23C1050 I2 FR23C1050 I2 FR 23C1050I2 FR 23C1050 C FR23C1050 C FR 23C1050C FR 23C1050 C FR23C1050 C FR 23C1050C FR 23C1050 I2 FR23C1050 I2 FR 23C1050I2
Authority
FR
France
Prior art keywords
alkynylbenzene
disubstituted
salt
compound
disubstituted alkynylbenzene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR23C1050C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taiho Pharmaceutical Co Ltd
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of FR23C1050I1 publication Critical patent/FR23C1050I1/fr
Application granted granted Critical
Publication of FR23C1050I2 publication Critical patent/FR23C1050I2/fr
Active legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
FR23C1050C 2012-01-19 2023-12-19 Compose d'alkynylbenzene 3,5-disubstitue et un sel de celui-ci Active FR23C1050I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012009467 2012-01-19
PCT/JP2013/050740 WO2013108809A1 (fr) 2012-01-19 2013-01-17 Composé d'alkynylbenzène 3,5-disubstitué et un sel de celui-ci

Publications (2)

Publication Number Publication Date
FR23C1050I1 FR23C1050I1 (fr) 2024-01-26
FR23C1050I2 true FR23C1050I2 (fr) 2024-12-13

Family

ID=48799233

Family Applications (1)

Application Number Title Priority Date Filing Date
FR23C1050C Active FR23C1050I2 (fr) 2012-01-19 2023-12-19 Compose d'alkynylbenzene 3,5-disubstitue et un sel de celui-ci

Country Status (23)

Country Link
US (1) US9108973B2 (fr)
EP (1) EP2657233B1 (fr)
JP (1) JP5355825B1 (fr)
KR (1) KR101623286B1 (fr)
CN (1) CN103958512B (fr)
AU (1) AU2013210403B2 (fr)
BR (1) BR112014017749B1 (fr)
CA (1) CA2854093C (fr)
DK (1) DK2657233T3 (fr)
ES (1) ES2516392T3 (fr)
FI (1) FIC20230038I1 (fr)
FR (1) FR23C1050I2 (fr)
HU (1) HUS2300043I1 (fr)
MX (1) MX351513B (fr)
MY (1) MY171055A (fr)
NL (1) NL301254I2 (fr)
NO (1) NO2023046I1 (fr)
PL (1) PL2657233T3 (fr)
PT (1) PT2657233E (fr)
RU (1) RU2576384C1 (fr)
SG (1) SG2014009286A (fr)
TW (1) TWI508964B (fr)
WO (1) WO2013108809A1 (fr)

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RU2679130C2 (ru) 2012-07-11 2019-02-06 Блюпринт Медсинс Корпорейшн Ингибиторы рецептора фактора роста фибробластов
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CN107698593A (zh) * 2016-08-09 2018-02-16 南京天印健华医药科技有限公司 作为fgfr抑制剂的杂环化合物
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WO2021146424A1 (fr) 2020-01-15 2021-07-22 Incyte Corporation Hétérocycles bicycliques en tant qu'inhibiteurs de fgfr
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Also Published As

Publication number Publication date
JP5355825B1 (ja) 2013-11-27
RU2576384C1 (ru) 2016-03-10
AU2013210403B2 (en) 2016-01-14
KR101623286B1 (ko) 2016-05-20
PL2657233T3 (pl) 2015-01-30
HUS2300043I1 (hu) 2024-01-28
FIC20230038I1 (fi) 2023-12-18
WO2013108809A1 (fr) 2013-07-25
TWI508964B (zh) 2015-11-21
PT2657233E (pt) 2014-10-24
DK2657233T3 (da) 2014-09-22
FR23C1050I1 (fr) 2024-01-26
TW201335156A (zh) 2013-09-01
AU2013210403A1 (en) 2014-06-26
BR112014017749A8 (pt) 2017-07-11
EP2657233A1 (fr) 2013-10-30
HK1198164A1 (zh) 2015-03-13
NO2023046I1 (no) 2023-12-20
CA2854093C (fr) 2016-07-05
MY171055A (en) 2019-09-23
ES2516392T3 (es) 2014-10-30
KR20140080551A (ko) 2014-06-30
CN103958512A (zh) 2014-07-30
CN103958512B (zh) 2016-01-20
CA2854093A1 (fr) 2013-07-25
BR112014017749A2 (pt) 2017-06-20
BR112014017749B1 (pt) 2021-08-03
JPWO2013108809A1 (ja) 2015-05-11
EP2657233B1 (fr) 2014-08-27
SG2014009286A (en) 2014-04-28
MX351513B (es) 2017-10-17
EP2657233A4 (fr) 2013-12-04
MX2014008605A (es) 2014-08-27
US9108973B2 (en) 2015-08-18
NL301254I2 (nl) 2024-01-10
NL301254I1 (fr) 2023-12-20
US20140343035A1 (en) 2014-11-20

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