FR2368959A1 - COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT - Google Patents
COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCTInfo
- Publication number
- FR2368959A1 FR2368959A1 FR7732620A FR7732620A FR2368959A1 FR 2368959 A1 FR2368959 A1 FR 2368959A1 FR 7732620 A FR7732620 A FR 7732620A FR 7732620 A FR7732620 A FR 7732620A FR 2368959 A1 FR2368959 A1 FR 2368959A1
- Authority
- FR
- France
- Prior art keywords
- guanidinoalcanoic
- compositions containing
- acid derivatives
- medicinal product
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- 239000002253 acid Substances 0.000 title abstract 2
- 229940126601 medicinal product Drugs 0.000 title 1
- 230000004071 biological effect Effects 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000004110 gluconeogenesis Effects 0.000 abstract 1
- 230000002440 hepatic effect Effects 0.000 abstract 1
- 230000003345 hyperglycaemic effect Effects 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Emergency Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Cette invention concerne une composition ayant une activité biologique. Cette composition renferme un mélange d'un dérivé d'acide guanidino-alcanoïque et un inhibiteur de gluconéogenèse hépatique. Elle est utilisable pour le traitement d'affections hyperglycémiques comme le diabète sucré.This invention relates to a composition having biological activity. This composition contains a mixture of a derivative of guanidino-alkanoic acid and an inhibitor of hepatic gluconeogenesis. It can be used for the treatment of hyperglycemic conditions such as diabetes mellitus.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB45450/76A GB1552179A (en) | 1976-11-02 | 1976-11-02 | Pharmaceutical compositions for treating hyperglycaemia |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| FR2368959A1 true FR2368959A1 (en) | 1978-05-26 |
Family
ID=10437252
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7732620A Withdrawn FR2368959A1 (en) | 1976-11-02 | 1977-10-28 | COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS5362834A (en) |
| AU (1) | AU2998777A (en) |
| BE (1) | BE860307A (en) |
| DE (1) | DE2747764A1 (en) |
| DK (1) | DK485777A (en) |
| FI (1) | FI773213A7 (en) |
| FR (1) | FR2368959A1 (en) |
| GB (1) | GB1552179A (en) |
| IL (1) | IL53207A0 (en) |
| NL (1) | NL7711993A (en) |
| SE (1) | SE7712328L (en) |
| ZA (1) | ZA776432B (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0370994A3 (en) * | 1988-11-25 | 1990-12-27 | Gert Prof. Dr. Lubec | Treatment of glucose-intermediated cross-linking of collagen in patients with diabetes mellitus by arginin, spermidin, creatin or agmatin |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU7316591A (en) * | 1990-02-28 | 1991-09-18 | Upjohn Company, The | Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders |
| US5599841A (en) * | 1990-02-28 | 1997-02-04 | The Upjohn Company | Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders |
| WO1993003724A1 (en) * | 1991-08-26 | 1993-03-04 | The Upjohn Company | Pharmaceutical composition containing 3-guanidinopropionic acid and pioglitazone glibenclamide or glimepiride |
| US6008253A (en) * | 1991-08-26 | 1999-12-28 | The Upjohn Company | Use of 3-guanidinopropionic acid to increase endurance, stamina and exercise capacity in a mammal |
| CA2117282A1 (en) * | 1991-11-22 | 1993-05-27 | Ofer Lider | Non-peptidic surrogates of the arg-gly-asp sequence and pharmaceutical compositions comprosing them |
| WO1997013507A1 (en) * | 1995-10-11 | 1997-04-17 | Avicena Group, Inc. | Use of creatine analogues for the treatment of disorders of glucose metabolism |
| US6099859A (en) | 1998-03-20 | 2000-08-08 | Andrx Pharmaceuticals, Inc. | Controlled release oral tablet having a unitary core |
| EP1768951A4 (en) * | 2004-06-17 | 2011-06-15 | Musc Found For Res Dev | NON-NATURAL AMINO ACIDS |
| DE102007034102A1 (en) * | 2007-07-21 | 2009-01-22 | Alzchem Trostberg Gmbh | Abrasion-resistant and free-flowing glycocyamine-containing moldings and process for their preparation |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1195199A (en) * | 1966-11-25 | 1970-06-17 | Horlicks Pharmaceuticals Ltd | Improvements in Compositions comprising Insulin. |
-
1976
- 1976-11-02 GB GB45450/76A patent/GB1552179A/en not_active Expired
-
1977
- 1977-10-24 IL IL53207A patent/IL53207A0/en unknown
- 1977-10-24 AU AU29987/77A patent/AU2998777A/en active Pending
- 1977-10-25 DE DE19772747764 patent/DE2747764A1/en active Pending
- 1977-10-27 FI FI773213A patent/FI773213A7/en not_active Application Discontinuation
- 1977-10-28 BE BE182218A patent/BE860307A/en unknown
- 1977-10-28 FR FR7732620A patent/FR2368959A1/en not_active Withdrawn
- 1977-10-28 ZA ZA00776432A patent/ZA776432B/en unknown
- 1977-11-01 SE SE7712328A patent/SE7712328L/en not_active Application Discontinuation
- 1977-11-01 DK DK485777A patent/DK485777A/en unknown
- 1977-11-01 NL NL7711993A patent/NL7711993A/en not_active Application Discontinuation
- 1977-11-02 JP JP13209477A patent/JPS5362834A/en active Pending
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1195199A (en) * | 1966-11-25 | 1970-06-17 | Horlicks Pharmaceuticals Ltd | Improvements in Compositions comprising Insulin. |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0370994A3 (en) * | 1988-11-25 | 1990-12-27 | Gert Prof. Dr. Lubec | Treatment of glucose-intermediated cross-linking of collagen in patients with diabetes mellitus by arginin, spermidin, creatin or agmatin |
Also Published As
| Publication number | Publication date |
|---|---|
| DK485777A (en) | 1978-05-03 |
| AU2998777A (en) | 1979-05-03 |
| FI773213A7 (en) | 1978-05-03 |
| ZA776432B (en) | 1978-08-30 |
| IL53207A0 (en) | 1977-12-30 |
| GB1552179A (en) | 1979-09-12 |
| JPS5362834A (en) | 1978-06-05 |
| SE7712328L (en) | 1978-05-02 |
| NL7711993A (en) | 1978-05-05 |
| DE2747764A1 (en) | 1978-05-03 |
| BE860307A (en) | 1978-04-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |