[go: up one dir, main page]

FR2368959A1 - COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT - Google Patents

COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT

Info

Publication number
FR2368959A1
FR2368959A1 FR7732620A FR7732620A FR2368959A1 FR 2368959 A1 FR2368959 A1 FR 2368959A1 FR 7732620 A FR7732620 A FR 7732620A FR 7732620 A FR7732620 A FR 7732620A FR 2368959 A1 FR2368959 A1 FR 2368959A1
Authority
FR
France
Prior art keywords
guanidinoalcanoic
compositions containing
acid derivatives
medicinal product
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7732620A
Other languages
French (fr)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of FR2368959A1 publication Critical patent/FR2368959A1/en
Withdrawn legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Cette invention concerne une composition ayant une activité biologique. Cette composition renferme un mélange d'un dérivé d'acide guanidino-alcanoïque et un inhibiteur de gluconéogenèse hépatique. Elle est utilisable pour le traitement d'affections hyperglycémiques comme le diabète sucré.This invention relates to a composition having biological activity. This composition contains a mixture of a derivative of guanidino-alkanoic acid and an inhibitor of hepatic gluconeogenesis. It can be used for the treatment of hyperglycemic conditions such as diabetes mellitus.

FR7732620A 1976-11-02 1977-10-28 COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT Withdrawn FR2368959A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB45450/76A GB1552179A (en) 1976-11-02 1976-11-02 Pharmaceutical compositions for treating hyperglycaemia

Publications (1)

Publication Number Publication Date
FR2368959A1 true FR2368959A1 (en) 1978-05-26

Family

ID=10437252

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7732620A Withdrawn FR2368959A1 (en) 1976-11-02 1977-10-28 COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT

Country Status (12)

Country Link
JP (1) JPS5362834A (en)
AU (1) AU2998777A (en)
BE (1) BE860307A (en)
DE (1) DE2747764A1 (en)
DK (1) DK485777A (en)
FI (1) FI773213A7 (en)
FR (1) FR2368959A1 (en)
GB (1) GB1552179A (en)
IL (1) IL53207A0 (en)
NL (1) NL7711993A (en)
SE (1) SE7712328L (en)
ZA (1) ZA776432B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0370994A3 (en) * 1988-11-25 1990-12-27 Gert Prof. Dr. Lubec Treatment of glucose-intermediated cross-linking of collagen in patients with diabetes mellitus by arginin, spermidin, creatin or agmatin

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU7316591A (en) * 1990-02-28 1991-09-18 Upjohn Company, The Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders
US5599841A (en) * 1990-02-28 1997-02-04 The Upjohn Company Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders
WO1993003724A1 (en) * 1991-08-26 1993-03-04 The Upjohn Company Pharmaceutical composition containing 3-guanidinopropionic acid and pioglitazone glibenclamide or glimepiride
US6008253A (en) * 1991-08-26 1999-12-28 The Upjohn Company Use of 3-guanidinopropionic acid to increase endurance, stamina and exercise capacity in a mammal
CA2117282A1 (en) * 1991-11-22 1993-05-27 Ofer Lider Non-peptidic surrogates of the arg-gly-asp sequence and pharmaceutical compositions comprosing them
WO1997013507A1 (en) * 1995-10-11 1997-04-17 Avicena Group, Inc. Use of creatine analogues for the treatment of disorders of glucose metabolism
US6099859A (en) 1998-03-20 2000-08-08 Andrx Pharmaceuticals, Inc. Controlled release oral tablet having a unitary core
EP1768951A4 (en) * 2004-06-17 2011-06-15 Musc Found For Res Dev NON-NATURAL AMINO ACIDS
DE102007034102A1 (en) * 2007-07-21 2009-01-22 Alzchem Trostberg Gmbh Abrasion-resistant and free-flowing glycocyamine-containing moldings and process for their preparation

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1195199A (en) * 1966-11-25 1970-06-17 Horlicks Pharmaceuticals Ltd Improvements in Compositions comprising Insulin.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1195199A (en) * 1966-11-25 1970-06-17 Horlicks Pharmaceuticals Ltd Improvements in Compositions comprising Insulin.

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0370994A3 (en) * 1988-11-25 1990-12-27 Gert Prof. Dr. Lubec Treatment of glucose-intermediated cross-linking of collagen in patients with diabetes mellitus by arginin, spermidin, creatin or agmatin

Also Published As

Publication number Publication date
DK485777A (en) 1978-05-03
AU2998777A (en) 1979-05-03
FI773213A7 (en) 1978-05-03
ZA776432B (en) 1978-08-30
IL53207A0 (en) 1977-12-30
GB1552179A (en) 1979-09-12
JPS5362834A (en) 1978-06-05
SE7712328L (en) 1978-05-02
NL7711993A (en) 1978-05-05
DE2747764A1 (en) 1978-05-03
BE860307A (en) 1978-04-28

Similar Documents

Publication Publication Date Title
FR2455028A1 (en) NOVEL ACYLCARNITIN AMIDES, ESPECIALLY USEFUL AS CENTRAL NERVOUS STIMULANTS, AND PROCESS FOR THEIR PREPARATION
FR2453148A1 (en) NOVEL ARYLSULFINYL DERIVATIVES OF ACETOHYDROXAMIC ACID, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC APPLICATION
FR2430410A1 (en) PHENETHANOLAMINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
FR2427329A1 (en) NEW DERIVATIVES OF PHENOXYALKYLCARBOXYLIC ACIDS AND THEIR APPLICATION IN THERAPEUTICS, IN PARTICULAR AS HYPOLIPIDEMATING AND HYPOCHOLESTEROLEMATING AGENTS
FR2392667A1 (en) SUSTAINED-RELEASE PHARMACEUTICAL COMPOSITION CONSISTING OF PROPRANOLOL
FR2416234A1 (en) METRONIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING
FR2415112A1 (en) NEW SPIROTHIENOHYDANTOINS DERIVATIVES AND PHARMACEUTICAL COMPOSITION CONTAINING THEM
ATE60579T1 (en) PYRROLIDINAMIDE DERIVATIVES WITH ANTIPROPYLENE ENDOPEPTIDASE ACTIVITY, COMPOSITIONS CONTAINING THEM, PROCESSES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM.
BE903183A (en) NOVEL BENZONORBORNENE DERIVATIVES, PREPARATION METHODS THEREOF, AND MEDICINAL AND COSMETIC COMPOSITION CONTAINING THEM
FR2397403A1 (en) NEW DERIVATIVES OF 1-ACYL 2-CYANO-AZIRIDINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS
FR2368959A1 (en) COMPOSITIONS CONTAINING GUANIDINOALCANOIC ACID DERIVATIVES, USED AS A MEDICINAL PRODUCT
FR2457689A1 (en) HYPOLIPEMIC CARNITINE-BASED MEDICINE
JPS5665869A (en) Novel 22hydroxyalkyll3*4*55trihydroxyypiperidine compound* its manufacture and drug
FR2393577A1 (en) B- (P-HALOGENOPHENYL) -G-AMINOBUTYRIC ACID BASED MEDICINAL PRODUCT FOR THE TREATMENT OF ANXIETY NEPROSIS
FR2358415A1 (en) PEPTIDIC DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2374288A1 (en) NEW INTERPHENYLENES-11,12-SECOPROSTAGLANDINS USEFUL AS MEDICINAL PRODUCTS
FR2405067A1 (en) PHARMACEUTICAL COMPOSITIONS CONTAINING MONOFUNCTIONAL DERIVATIVES OF PSORALENE FOR THE TREATMENT OF SKIN DISORDERS
FR2453152A1 (en) NEW PROSTAGLANDIN DERIVATIVES AND MEDICAMENTS CONTAINING THEM
FR2414042A1 (en) PROCESS FOR THE PRODUCTION OF N-METHYLMORANOLINE AND NEW PRODUCT THUS OBTAINED
FR2450837A1 (en) 6-B-SUBSTITUTED PENICILLANIC ACIDS B-LACTAMASE INHIBITORS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM
FR2447189A1 (en) NOVEL COSMETIC COMPOSITIONS FOR THE TREATMENT OF HAIR AND SKIN CONTAINING AS ACTIVE INGREDIENTS OF ALKYLENE-DITHIOETHERS
FR2440353A1 (en) NOVEL ARYLETHANOLS, PROCESSES FOR OBTAINING THEM AND THEIR USE AS A MEDICINAL PRODUCT
FR2378741A1 (en) GARYL GOXO ISOVALERIC ACIDS WITH ANTIPHLOGISTIC AND ANTALGIC PROPERTIES
KR950032191A (en) Cyclohexane Derivatives, Methods of Making the Same, and Use of Compounds to Treat Diseases
FR2369216A1 (en) WATER TREATMENT PRODUCTS CONTAINING ACYLIMINO DIACETIC ACIDS

Legal Events

Date Code Title Description
ST Notification of lapse