FI952797L - D-vitamiinianalogin uusi kiteinen muoto - Google Patents

D-vitamiinianalogin uusi kiteinen muoto Download PDF

Info

Publication number: FI952797L
Authority: FI; Finland
Prior art keywords: analogue; vitamin; crystalline form; new crystalline; new
Prior art date: 1993-01-15

Application number

FI952797A

Other languages

English (en)

Swedish (sv)

Other versions

FI108638B (fi

FI952797A0 (fi

Inventor

Erik Torngaard Hansen

Andersen Niels Smidt Rastrup

Lene Hoffmeyer Ringborg

Original Assignee

Leo Pharm Prod Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-01-15

Filing date

1995-06-07

Publication date

1995-06-07

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10728784&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI952797(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1995-06-07 Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd

1995-06-07 Publication of FI952797L publication Critical patent/FI952797L/fi

1995-06-07 Publication of FI952797A0 publication Critical patent/FI952797A0/fi

2002-02-28 Application granted granted Critical

2002-02-28 Publication of FI108638B publication Critical patent/FI108638B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J19/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J19/02—Apparatus characterised by being constructed of material selected for its chemically-resistant properties
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C5/00—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms
- C07C5/32—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms by dehydrogenation with formation of free hydrogen
- C07C5/321—Catalytic processes
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C5/00—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms
- C07C5/32—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms by dehydrogenation with formation of free hydrogen
- C07C5/327—Formation of non-aromatic carbon-to-carbon double bonds only
- C07C5/333—Catalytic processes
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C5/00—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms
- C07C5/32—Preparation of hydrocarbons from hydrocarbons containing the same number of carbon atoms by dehydrogenation with formation of free hydrogen
- C07C5/327—Formation of non-aromatic carbon-to-carbon double bonds only
- C07C5/333—Catalytic processes
- C07C5/3335—Catalytic processes with metals
- C07C5/3337—Catalytic processes with metals of the platinum group
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/02—Apparatus characterised by their chemically-resistant properties
- B01J2219/0204—Apparatus characterised by their chemically-resistant properties comprising coatings on the surfaces in direct contact with the reactive components
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/02—Apparatus characterised by their chemically-resistant properties
- B01J2219/0204—Apparatus characterised by their chemically-resistant properties comprising coatings on the surfaces in direct contact with the reactive components
- B01J2219/0236—Metal based
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/02—Apparatus characterised by their chemically-resistant properties
- B01J2219/025—Apparatus characterised by their chemically-resistant properties characterised by the construction materials of the reactor vessel proper
- B01J2219/0277—Metal based
- B01J2219/0286—Steel
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2523/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00
- C07C2523/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00 of noble metals
- C07C2523/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00 of noble metals of the platinum group metals
- C07C2523/42—Platinum

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

FI952797A 1993-01-15 1995-06-07 Menetelmä D-vitamiinianalogin uuden kiteisen muodon valmistamiseksi FI108638B (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GB939300763A GB9300763D0 (en)	1993-01-15	1993-01-15	Chemical compound
GB9300763		1993-01-15
PCT/DK1994/000011 WO1994015912A1 (en)	1993-01-15	1994-01-07	New crystalline form of a vitamin d analogue
DK9400011		1994-01-07

Publications (3)

Publication Number	Publication Date
FI952797L true FI952797L (fi)	1995-06-07
FI952797A0 FI952797A0 (fi)	1995-06-07
FI108638B FI108638B (fi)	2002-02-28

Family

ID=10728784

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI952797A FI108638B (fi)	1993-01-15	1995-06-07	Menetelmä D-vitamiinianalogin uuden kiteisen muodon valmistamiseksi

Country Status (17)

Country	Link
US (2)	US5763426A (fi)
EP (1)	EP0679154B1 (fi)
JP (1)	JP3729847B2 (fi)
KR (1)	KR100309751B1 (fi)
CN (1)	CN1040746C (fi)
AT (1)	ATE159717T1 (fi)
AU (1)	AU663249B2 (fi)
CA (1)	CA2151730C (fi)
DE (1)	DE69406529T2 (fi)
DK (1)	DK0679154T3 (fi)
ES (1)	ES2111287T3 (fi)
FI (1)	FI108638B (fi)
GB (1)	GB9300763D0 (fi)
GR (1)	GR3025668T3 (fi)
NZ (1)	NZ259679A (fi)
RU (1)	RU2128646C1 (fi)
WO (1)	WO1994015912A1 (fi)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU710931B2 (en) *	1996-02-28	1999-09-30	Sumitomo Pharmaceuticals Company, Limited	Crystalline vitamin D derivative
US8263580B2 (en)	1998-09-11	2012-09-11	Stiefel Research Australia Pty Ltd	Vitamin formulation
CA2370565C (en) *	1999-04-23	2008-11-25	Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab)	Dermally applicable vitamin d-containing pharmaceutical compositions
US20090098065A1 (en) *	2000-01-11	2009-04-16	Avikam Harel	Composition and methods for the treatment of skin disorders
WO2004046097A1 (en) *	2002-11-18	2004-06-03	Teva Pharmaceutical Industries Ltd.	A crystallization method for purification of calcipotriene
US8362287B2 (en)	2004-03-18	2013-01-29	Leo Pharma A/S	Stereoselective synthesis of vitamin D analogues
JP4667450B2 (ja) *	2004-03-18	2011-04-13	レオファーマアクティーゼルスカブ	ビタミンｄ類似体の立体選択的合成
FR2871696B1 (fr) *	2004-06-17	2006-11-10	Galderma Sa	Composition topique pour le traitement du psoriasis
TWI318203B (en) *	2004-09-01	2009-12-11	Leo Pharma As	Epimerization of allylic alcohols
WO2006129161A2 (en)	2005-06-01	2006-12-07	Stiefel Research Australia Pty Ltd	Vitamin formulation
US7989631B2 (en) *	2006-02-10	2011-08-02	Amgen Inc.	Hydrate forms of AMG706
BRPI0621471A2 (pt) *	2006-03-17	2012-09-11	Leo Pharma As	métodos de isomerização de uma solução de um derivado de vitamina d, para produzir e preparar calcipotriol ou monoidrato de calcipotriol, e para a fabricação de uma formulação farmacêutica ou medicamento, e, uso de um reator foto-reator de fluxo direto ou foto-reator de fluxo contìnuo
US20080064669A1 (en) *	2006-08-29	2008-03-13	Rakefet Cohen	Stable pharmacologically active compositions including vitamin D-containing and corticosteroid compounds with low pH compatibility
US20100056644A1 (en) *	2006-11-29	2010-03-04	Nilendu Sen	Pharmaceutical compositions containing anhydrous calcipotriene
ES2272198B1 (es) *	2006-12-28	2008-06-01	Laboratorios Viñas S.A.	Procedimiento para la obtencion de hidrato de calcipotriol.
US10265265B2 (en) *	2007-03-15	2019-04-23	Drug Delivery Solutions Limited	Topical composition
EP1970048A1 (en) *	2007-03-15	2008-09-17	Drug Delivery Solutions Limited	Polyaphron topical composition with vitamin D
EP2008651A1 (en)	2007-06-26	2008-12-31	Drug Delivery Solutions Limited	A bioerodible patch
ES2575565T3 (es) *	2008-05-08	2016-06-29	United Therapeutics Corporation	Procedimiento para la preparación de monohidrato de treprostinilo y su utilización para el almacenamiento y el envío
WO2011002756A2 (en) *	2009-07-01	2011-01-06	Vitamin Derivatives, Inc.	Vitamin d compounds and methods for preparing same
CN102770121B (zh)	2009-12-22	2014-10-15	利奥制药有限公司	包含溶剂混合物和维生素d衍生物或类似物的药物组合物
US9254296B2 (en)	2009-12-22	2016-02-09	Leo Pharma A/S	Pharmaceutical composition comprising vitamin D analogue and cosolvent-surfactant mixture
WO2011076206A1 (en) *	2009-12-22	2011-06-30	Leo Pharma A/S	Pharmaceutical composition comprising vitamin d analogue and cosolvent-surfactant mixture
PL2515874T3 (pl) *	2009-12-22	2015-01-30	Leo Pharma As	Nanokryształy jednowodnego kalcypotriolu
AU2010335654B2 (en)	2009-12-22	2015-04-09	Leo Pharma A/S	Cutaneous composition comprising vitamin D analogue and a mixture of solvent and surfactants
JP5945268B2 (ja)	2010-06-11	2016-07-05	レオファーマアクティーゼルスカブ	ビタミンｄ類似体およびコルチコステロイドを含むスプレー医薬組成物
WO2012123515A1 (en)	2011-03-14	2012-09-20	Drug Delivery Solutions Limited	An ophthalmic composition
EP2688560A2 (en)	2011-03-24	2014-01-29	Leo Pharma A/S	A composition comprising lipid nanoparticles and a corticosteroid or vitamin d derivative
JP5652723B2 (ja) *	2012-08-17	2015-01-14	フォーモサ・ラボラトリーズ・インコーポレーテッド	マキサカルシトールの新しい結晶形態
CN103724162A (zh) *	2014-01-07	2014-04-16	成都医路康医学技术服务有限公司	一种银屑病治疗药物卡泊三醇溶剂化物的制备方法
MA41818A (fr)	2015-03-27	2018-01-30	Leo Pharma As	Timbre à micro-aiguilles pour administration d'un principe actif à la peau
EP3542788A1 (en)	2018-03-19	2019-09-25	MC2 Therapeutics Limited	Topical composition comprising calcipotriol and betamethasone dipropionate

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2457282A1 (fr) *	1979-05-23	1980-12-19	Roussel Uclaf	Nouveau derive du 1a,25 dihydroxy cholecalciferol, son procede de preparation et son application comme medicament
JPS59104358A (ja)	1982-12-03	1984-06-16	Teijin Ltd	１α，２４−ジヒドロキシコレカルシフエロ−ルの一水塩及びその製造法
JPH07100685B2 (ja) *	1985-08-02	1995-11-01	レオ・ファ−マシュ−ティカル・プロダクツ・リミテッド・エイ／エス（レ−ベンス・ケミスケ・ファブリック・プロデュクチオンスアクチ−セルスカブ）	新規ビタミンｄ類似体
GB9004544D0 (en) *	1990-03-01	1990-04-25	Leo Pharm Prod Ltd	Novel treatment ii

1993
- 1993-01-15 US US08/491,892 patent/US5763426A/en not_active Ceased
- 1993-01-15 GB GB939300763A patent/GB9300763D0/en active Pending
- 1993-01-15 US US10/986,575 patent/USRE39706E1/en not_active Expired - Lifetime
1994
- 1994-01-07 KR KR1019950702271A patent/KR100309751B1/ko not_active Expired - Lifetime
- 1994-01-07 WO PCT/DK1994/000011 patent/WO1994015912A1/en not_active Ceased
- 1994-01-07 NZ NZ259679A patent/NZ259679A/en not_active IP Right Cessation
- 1994-01-07 RU RU95116650A patent/RU2128646C1/ru active
- 1994-01-07 EP EP94904583A patent/EP0679154B1/en not_active Expired - Lifetime
- 1994-01-07 CA CA002151730A patent/CA2151730C/en not_active Expired - Lifetime
- 1994-01-07 AT AT94904583T patent/ATE159717T1/de active
- 1994-01-07 DE DE69406529T patent/DE69406529T2/de not_active Expired - Lifetime
- 1994-01-07 ES ES94904583T patent/ES2111287T3/es not_active Expired - Lifetime
- 1994-01-07 AU AU58573/94A patent/AU663249B2/en not_active Expired
- 1994-01-07 CN CN94190817A patent/CN1040746C/zh not_active Expired - Lifetime
- 1994-01-07 JP JP51560694A patent/JP3729847B2/ja not_active Expired - Lifetime
- 1994-01-07 DK DK94904583.5T patent/DK0679154T3/da active
1995
- 1995-06-07 FI FI952797A patent/FI108638B/fi not_active IP Right Cessation
1997
- 1997-12-16 GR GR970403317T patent/GR3025668T3/el unknown

Also Published As

Publication number	Publication date
FI108638B (fi)	2002-02-28
JPH08505612A (ja)	1996-06-18
AU5857394A (en)	1994-08-15
DE69406529D1 (de)	1997-12-04
FI952797A0 (fi)	1995-06-07
ATE159717T1 (de)	1997-11-15
CN1115979A (zh)	1996-01-31
ES2111287T3 (es)	1998-03-01
RU95116650A (ru)	1997-06-10
KR950704249A (ko)	1995-11-17
EP0679154B1 (en)	1997-10-29
NZ259679A (en)	1996-11-26
CA2151730A1 (en)	1994-07-21
RU2128646C1 (ru)	1999-04-10
GR3025668T3 (en)	1998-03-31
US5763426A (en)	1998-06-09
DK0679154T3 (da)	1998-03-30
CA2151730C (en)	2005-01-04
CN1040746C (zh)	1998-11-18
GB9300763D0 (en)	1993-03-03
USRE39706E1 (en)	2007-06-26
JP3729847B2 (ja)	2005-12-21
WO1994015912A1 (en)	1994-07-21
KR100309751B1 (ko)	2002-11-08
AU663249B2 (en)	1995-09-28
DE69406529T2 (de)	1998-05-28
EP0679154A1 (en)	1995-11-02

Publication	Publication Date	Title
FI952797L (fi)	1995-06-07	D-vitamiinianalogin uusi kiteinen muoto
FR2630637B1 (fr)	1997-09-12	Nouvelle prothese alveolaire
FI934261L (fi)	1994-03-30	Foerfarande foer framstaellning av en bilvindruta foersedd med elastram av bestaemd form
PT1066828E (pt)	2003-10-31	Composicao de aerossol
FI935219L (fi)	1994-05-26	Kompositioner foer avskiljningskontroll foer med UV-straolning haerdbara agenser av epoxisilikon
FI945556A7 (fi)	1995-05-27	Tulehdustenvastaiset 3-aryyli-2-isoksatsoliinijohdannaiset
FI930657L (fi)	1993-08-18	Foerfarande foer framstaellning av doseringsformer med foerlaengd aktivaemnesfrigivning
FI932865A0 (fi)	1993-06-21	Kaernelektrod med aongminskning
DE69326663D1 (de)	1999-11-11	Unterschneidungsverfahren
FI961797L (fi)	1996-04-26	Stabiloitu prostaglandiini E1
FI931946L (fi)	1993-11-02	Alkylering av olefiner med isoparaffiner
FI930757A7 (fi)	1993-08-22	Bestrykningsmekanism foer bestrykning av en pappersbana med bestrykningssmet
FI924478L (fi)	1992-10-05	24-oxa-derivat i vitamin d-serien
DE69328310D1 (de)	2000-05-11	Prothetische schliessmuskeleinrichtung
FI931945L (fi)	1993-11-02	Alkylering av olefiner med isoparaffiner
DE69207786D1 (de)	1996-03-07	Analogweltzeituhr
FI931322L (fi)	1993-09-25	Stabilisering av peroxidblekningsvaetskor med klordioxid
FI216U1 (fi)	1992-08-12	Foerlaengningsholk foersedd med momentskruvar
FI933487L (fi)	1994-02-08	Jaestvaerdstammor med defekter i N-glykosyleringen
FI932350L (fi)	1993-11-26	Foerfarande foer separering av katalysatorfri arbetsloesning ur hydreringskretsloppet vid framstaellning av vaeteperoxid med antrakinonfoerfarandet
NO952485D0 (no)	1995-06-21	Antiinflammatorisk difluorpentapeptidderivat
FI931997L (fi)	1993-11-08	Spindeldrift med snabbutloesning av drivspindeln
FI922716L (fi)	1993-12-12	Foerfarande i samband med framstaellning av plaststycken
FI932658A0 (fi)	1993-06-10	Foerfarande foer framstaellning av viskosfibrer med bandformade tvaersnitt
FI925493A0 (fi)	1992-12-03	Rumselementsystem foer ersaettning av vaotutrymmen med tillfaelligutrymmeni samband med byggnadsarbeten

Legal Events

Date	Code	Title	Description
2014-02-18	MA	Patent expired