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FI932206A0 - This heterocyclic compound is an antagonist of excitatory amino acid receptors, which can be used as an exciter - Google Patents

This heterocyclic compound is an antagonist of excitatory amino acid receptors, which can be used as an exciter

Info

Publication number
FI932206A0
FI932206A0 FI932206A FI932206A FI932206A0 FI 932206 A0 FI932206 A0 FI 932206A0 FI 932206 A FI932206 A FI 932206A FI 932206 A FI932206 A FI 932206A FI 932206 A0 FI932206 A0 FI 932206A0
Authority
FI
Finland
Prior art keywords
exciter
antagonist
amino acid
heterocyclic compound
excitatory amino
Prior art date
Application number
FI932206A
Other languages
Finnish (fi)
Other versions
FI932206A7 (en
FI932206L (en
Inventor
Alf Claesson
Britt-Marie Swahn
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Publication of FI932206A0 publication Critical patent/FI932206A0/en
Publication of FI932206A7 publication Critical patent/FI932206A7/en
Publication of FI932206L publication Critical patent/FI932206L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6509—Six-membered rings
    • C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/59—Hydrogenated pyridine rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Injection Moulding Of Plastics Or The Like (AREA)
FI932206A 1990-11-15 1991-11-07 Nya heterocykliska foereningar som antagonister mot excitatory aminosyrareceptorer, foerfaranden Foer deras framstaellning och anvaendning av desamma FI932206L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9003652A SE9003652D0 (en) 1990-11-15 1990-11-15 NEW HETEROCYCLIC COMPOUNDS
PCT/SE1991/000753 WO1992008724A1 (en) 1990-11-15 1991-11-07 New heterocyclic compounds as antagonists of excitatory amino acid receptors, processes for their preparation and their use

Publications (3)

Publication Number Publication Date
FI932206A0 true FI932206A0 (en) 1993-05-14
FI932206A7 FI932206A7 (en) 1993-05-14
FI932206L FI932206L (en) 1993-05-14

Family

ID=20380925

Family Applications (1)

Application Number Title Priority Date Filing Date
FI932206A FI932206L (en) 1990-11-15 1991-11-07 Nya heterocykliska foereningar som antagonister mot excitatory aminosyrareceptorer, foerfaranden Foer deras framstaellning och anvaendning av desamma

Country Status (17)

Country Link
EP (1) EP0557375A1 (en)
JP (1) JPH06502421A (en)
CN (1) CN1061595A (en)
AU (1) AU652399B2 (en)
CA (1) CA2095224A1 (en)
CZ (1) CZ80993A3 (en)
FI (1) FI932206L (en)
HU (1) HU9301417D0 (en)
IE (1) IE913922A1 (en)
IS (1) IS3782A7 (en)
LT (1) LTIP1718A (en)
MX (1) MX9101979A (en)
NO (1) NO931679D0 (en)
PT (1) PT99515A (en)
SE (1) SE9003652D0 (en)
SK (1) SK46993A3 (en)
WO (1) WO1992008724A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5194430A (en) * 1990-05-17 1993-03-16 Merrell Dow Pharmaceuticals Inc. Heterocyclic-nmda antagonists
TW281670B (en) * 1993-09-02 1996-07-21 Hoffmann La Roche
US5491241A (en) * 1993-10-18 1996-02-13 Eli Lilly And Company Bicyclic intermediates for excitatory amino acid receptor antagonists
US10508083B2 (en) 2016-02-04 2019-12-17 Takeda Pharmaceutical Company Limited Substituted piperidine compound and use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1248531A (en) * 1984-04-17 1989-01-10 Jeffrey C. Watkins 4-substituted piperazine-2-carboxylic acids
JPS612519A (en) * 1984-04-24 1986-01-08 Aron Kasei Co Ltd Method of injection molding
US4906621A (en) * 1985-05-24 1990-03-06 Ciba-Geigy Corporation Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
US4740346A (en) * 1986-02-26 1988-04-26 The Budd Company Perimeter resin feeding of composite structures
JPS63112129A (en) * 1986-10-30 1988-05-17 Toyoda Gosei Co Ltd Multi-color resin molding die
IL84492A0 (en) * 1986-11-21 1988-04-29 Ciba Geigy Ag Unsaturated phosphonic acids and derivatives

Also Published As

Publication number Publication date
CA2095224A1 (en) 1992-05-16
CN1061595A (en) 1992-06-03
NO931679L (en) 1993-05-07
FI932206A7 (en) 1993-05-14
LTIP1718A (en) 1995-07-25
JPH06502421A (en) 1994-03-17
AU652399B2 (en) 1994-08-25
SK46993A3 (en) 1993-10-06
WO1992008724A1 (en) 1992-05-29
NO931679D0 (en) 1993-05-07
HU9301417D0 (en) 1993-09-28
IS3782A7 (en) 1992-05-16
PT99515A (en) 1992-09-30
IE913922A1 (en) 1992-05-20
AU8939191A (en) 1992-06-11
FI932206L (en) 1993-05-14
SE9003652D0 (en) 1990-11-15
EP0557375A1 (en) 1993-09-01
CZ80993A3 (en) 1994-02-16
MX9101979A (en) 1992-07-08

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FI932206A0 (en) This heterocyclic compound is an antagonist of excitatory amino acid receptors, which can be used as an exciter
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Legal Events

Date Code Title Description
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