FI20001109L - Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi - Google Patents

Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi Download PDF

Info

Publication number: FI20001109L
Authority: FI; Finland
Prior art keywords: resolving; racemic mixture; cis compound; cis; compound
Prior art date: 1991-01-03

Application number

FI20001109A

Other languages

English (en)

Swedish (sv)

Other versions

FI20001109A7 (fi

Inventor

Dennis M Godek

Charles W Murtiashaw

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-01-03

Filing date

2000-05-10

Publication date

2000-05-10

2000-05-10 Application filed by Pfizer filed Critical Pfizer

2000-05-10 Publication of FI20001109A7 publication Critical patent/FI20001109A7/fi

2000-05-10 Publication of FI20001109L publication Critical patent/FI20001109L/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Indole Compounds (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Apparatuses For Bulk Treatment Of Fruits And Vegetables And Apparatuses For Preparing Feeds (AREA)

FI20001109A 1991-01-03 2000-05-10 Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi FI20001109L (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/637,102 US5138060A (en)	1991-01-03	1991-01-03	Process and intermediates for preparing azabicyclo(2.2.2)octan-3-imines
PCT/US1991/009186 WO1992012152A1 (en)	1991-01-03	1991-12-18	Process and intermediates for preparing azabicyclo[2.2.2]octan-3-imines

Publications (2)

Publication Number	Publication Date
FI20001109A7 FI20001109A7 (fi)	2000-05-10
FI20001109L true FI20001109L (fi)	2000-05-10

Family

ID=24554545

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
FI933065A FI933065A7 (fi)	1991-01-03	1991-12-18	Menetelmä atsabisyklo(2.2.2)oktaani-3-imiinien valmistamiseksi ja menetelmässä käytetyt välituotteet
FI20001108A FI20001108L (fi)	1991-01-03	2000-05-10	Menetelmä raseemisen cis-yhdisteen valmistamiseksi
FI20001109A FI20001109L (fi)	1991-01-03	2000-05-10	Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
FI933065A FI933065A7 (fi)	1991-01-03	1991-12-18	Menetelmä atsabisyklo(2.2.2)oktaani-3-imiinien valmistamiseksi ja menetelmässä käytetyt välituotteet
FI20001108A FI20001108L (fi)	1991-01-03	2000-05-10	Menetelmä raseemisen cis-yhdisteen valmistamiseksi

Country Status (21)

Country	Link
US (1)	US5138060A (fi)
EP (1)	EP0565558B1 (fi)
JP (5)	JPH0768244B2 (fi)
KR (1)	KR970001157B1 (fi)
AT (1)	ATE115580T1 (fi)
AU (1)	AU653380B2 (fi)
CA (2)	CA2158130C (fi)
DE (1)	DE69106003T2 (fi)
DK (1)	DK0565558T3 (fi)
ES (1)	ES2065161T3 (fi)
FI (3)	FI933065A7 (fi)
GR (1)	GR3015021T3 (fi)
HU (1)	HU9301931D0 (fi)
IE (1)	IE65005B1 (fi)
IL (1)	IL100541A0 (fi)
MX (1)	MX9200003A (fi)
NO (1)	NO932431L (fi)
NZ (1)	NZ241161A (fi)
PT (1)	PT99970B (fi)
WO (1)	WO1992012152A1 (fi)
ZA (1)	ZA928B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5364943A (en) *	1991-11-27	1994-11-15	Pfizer Inc.	Preparation of substituted piperidines
ES2092113T3 (es) *	1991-06-20	1996-11-16	Pfizer	Derivados fluoroalcoxibencilamino de heterociclos que contienen nitrogeno.
HUT70741A (en) *	1991-11-12	1995-10-30	Pfizer	Acyclic ethylenediamine derivatives as substance p receptor antagonists
EP0641328B1 (en) *	1992-05-18	2001-11-21	Pfizer Inc.	Bridged aza-bicyclic derivatives as substance p antagonists
US6048859A (en)	1992-06-29	2000-04-11	Merck & Co., Inc.	Morpholine and thiomorpholine tachykinin receptor antagonists
US5719147A (en) *	1992-06-29	1998-02-17	Merck & Co., Inc.	Morpholine and thiomorpholine tachykinin receptor antagonists
US5637699A (en) *	1992-06-29	1997-06-10	Merck & Co., Inc.	Process for preparing morpholine tachykinin receptor antagonists
JPH07506379A (ja) *	1992-08-04	1995-07-13	ファイザー・インコーポレーテッド	物質ｐ受容体アンタゴニストとしての３−ベンジルアミノ−２−フェニル−ピペリジン
US5387595A (en) *	1992-08-26	1995-02-07	Merck & Co., Inc.	Alicyclic compounds as tachykinin receptor antagonists
US5518628A (en) *	1993-11-08	1996-05-21	Shipley Company Inc.	Purification process
TW385308B (en) *	1994-03-04	2000-03-21	Merck & Co Inc	Prodrugs of morpholine tachykinin receptor antagonists
US6861526B2 (en)	2002-10-16	2005-03-01	Pfizer Inc.	Process for the preparation of (S,S)-cis-2-benzhydryl-3-benzylaminoquinuclidine
US20050136487A1 (en) *	2003-10-27	2005-06-23	Meyer Donald W.	Transmissible spongiform encephalopathy detection in cervids, sheep and goats

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3560510A (en) *	1969-03-05	1971-02-02	Aldrich Chem Co Inc	2-benzhydrylquinuclidines
US3993652A (en) *	1973-07-09	1976-11-23	Air Products And Chemicals, Inc.	Cyclic quaternary hydroxyalkyl phenoxide catalysts for isocyanate reactions
US4203990A (en) *	1979-04-30	1980-05-20	G. D. Searle & Co.	Anti-diarrheal 2-substituted quinuclidines
FR2529548A1 (fr) *	1982-07-02	1984-01-06	Delalande Sa	Nouveaux derives de l'amino-3 quinuclidine, leur procede et leur application en therapeutique
JPS59110656A (ja) *	1982-12-15	1984-06-26	Hiroyuki Nohira	光学活性な１―フェニル―２―（パラ―トリル）エチルアミンの製造方法
DE3604591A1 (de) *	1986-02-14	1987-08-20	Degussa	Verfahren zur herstellung chiraler glycinderivate
JPS6354342A (ja) *	1986-08-26	1988-03-08	Daicel Chem Ind Ltd	（±）−α−エチルベンジルアミンの光学分割方法
JPS63145256A (ja) *	1986-12-09	1988-06-17	Nippon Kayaku Co Ltd	光学活性ホモフエニルアラニンの製造法及び中間体
MX18467A (es) *	1988-11-23	1993-07-01	Pfizer	Agentes terapeuticos de quinuclidinas
AU658898B2 (en) *	1991-05-22	1995-05-04	Pfizer Inc.	Substituted 3-aminoquinuclidines

1991
- 1991-01-03 US US07/637,102 patent/US5138060A/en not_active Expired - Lifetime
- 1991-12-18 HU HU9301931A patent/HU9301931D0/hu unknown
- 1991-12-18 JP JP4-502391A patent/JPH0768244B2/ja not_active Expired - Lifetime
- 1991-12-18 DE DE69106003T patent/DE69106003T2/de not_active Expired - Fee Related
- 1991-12-18 CA CA002158130A patent/CA2158130C/en not_active Expired - Fee Related
- 1991-12-18 DK DK92901603.8T patent/DK0565558T3/da active
- 1991-12-18 ES ES92901603T patent/ES2065161T3/es not_active Expired - Lifetime
- 1991-12-18 JP JP4502391A patent/JPH0768244B1/ja active Pending
- 1991-12-18 WO PCT/US1991/009186 patent/WO1992012152A1/en not_active Ceased
- 1991-12-18 KR KR1019930702007A patent/KR970001157B1/ko not_active Expired - Lifetime
- 1991-12-18 CA CA002098989A patent/CA2098989C/en not_active Expired - Fee Related
- 1991-12-18 EP EP92901603A patent/EP0565558B1/en not_active Expired - Lifetime
- 1991-12-18 AU AU91298/91A patent/AU653380B2/en not_active Expired - Fee Related
- 1991-12-18 AT AT92901603T patent/ATE115580T1/de not_active IP Right Cessation
- 1991-12-18 FI FI933065A patent/FI933065A7/fi not_active Application Discontinuation
- 1991-12-23 NZ NZ241161A patent/NZ241161A/en unknown
- 1991-12-27 IL IL100541A patent/IL100541A0/xx unknown
1992
- 1992-01-02 ZA ZA928A patent/ZA928B/xx unknown
- 1992-01-02 MX MX9200003A patent/MX9200003A/es unknown
- 1992-01-02 IE IE920001A patent/IE65005B1/en not_active IP Right Cessation
- 1992-01-02 PT PT99970A patent/PT99970B/pt not_active IP Right Cessation
1993
- 1993-07-02 NO NO93932431A patent/NO932431L/no unknown
1994
- 1994-12-26 JP JP6322350A patent/JP2845425B2/ja not_active Expired - Fee Related
- 1994-12-26 JP JP6322353A patent/JP2583026B2/ja not_active Expired - Fee Related
- 1994-12-26 JP JP6322355A patent/JP2703193B2/ja not_active Expired - Fee Related
1995
- 1995-02-08 GR GR950400264T patent/GR3015021T3/el unknown
2000
- 2000-05-10 FI FI20001108A patent/FI20001108L/fi not_active Application Discontinuation
- 2000-05-10 FI FI20001109A patent/FI20001109L/fi not_active Application Discontinuation

Also Published As

Publication number	Publication date
FI933065A0 (fi)	1993-07-02
FI20001109A7 (fi)	2000-05-10
JPH07330766A (ja)	1995-12-19
IE65005B1 (en)	1995-10-04
JPH07316154A (ja)	1995-12-05
JP2845425B2 (ja)	1999-01-13
FI20001108A7 (fi)	2000-05-10
ES2065161T3 (es)	1995-02-01
US5138060A (en)	1992-08-11
JP2703193B2 (ja)	1998-01-26
JPH07316153A (ja)	1995-12-05
GR3015021T3 (en)	1995-05-31
JP2583026B2 (ja)	1997-02-19
WO1992012152A1 (en)	1992-07-23
CA2098989C (en)	1998-02-03
DE69106003T2 (de)	1995-04-27
ATE115580T1 (de)	1994-12-15
DE69106003D1 (de)	1995-01-26
PT99970B (pt)	1999-06-30
KR930703312A (ko)	1993-11-29
JPH0768244B1 (fi)	1995-07-26
CA2158130C (en)	1998-07-14
DK0565558T3 (da)	1995-03-06
AU653380B2 (en)	1994-09-29
NZ241161A (en)	1994-10-26
FI20001108L (fi)	2000-05-10
NO932431D0 (no)	1993-07-02
KR970001157B1 (ko)	1997-01-29
MX9200003A (es)	1992-07-01
FI933065L (fi)	1993-07-02
PT99970A (pt)	1993-02-26
IL100541A0 (en)	1992-09-06
CA2098989A1 (en)	1992-07-04
HU9301931D0 (en)	1993-12-28
EP0565558B1 (en)	1994-12-14
JPH05508867A (ja)	1993-12-09
ZA928B (en)	1993-07-02
FI933065A7 (fi)	1993-07-02
AU9129891A (en)	1992-08-17
JPH0768244B2 (ja)	1995-07-26
IE920001A1 (en)	1992-07-15
EP0565558A1 (en)	1993-10-20
CA2158130A1 (en)	1992-07-04
NO932431L (no)	1993-07-02

Publication	Publication Date	Title
FI20030932A7 (fi)	2003-06-24	Menetelmä cis-FTC:n enantiomeerien erottamiseksi
ES538152A0 (es)	1986-02-01	Un derivado de dihidropiridina
FI933789A7 (fi)	1993-08-30	Menetelmä kemiallisen yhdisteen lisäämiseksi kuituun
FI20001109L (fi)	2000-05-10	Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi
FI882875A7 (fi)	1988-12-23	Menetelmä valmistaa farmakologisesti arvokasta substituoitua aminokarbonyylioksipropionyyli-histidyyliaminoalkoholiyhdistettä
ES542023A0 (es)	1986-09-01	Un procedimiento para preparar un compuesto de n-aril-n- -(4-piperidinil)-alcoxialquilamida
FI882253L (fi)	1988-11-15	Menetelmä kefuroksiimiaksetiilikoostumuksen valmistamiseksi
FI945441L (fi)	1994-11-18	Uusi menetelmä 7beta-substituoitu-4-atsa-5alfa-androstan-3-onien valmistamiseksi
FI943117A7 (fi)	1994-06-29	Menetelmä harjaskimppujen kiinnittämiseksi harjasalustaan
ES556503A0 (es)	1987-07-16	Un metodo para sintetizar compuestos de ascorbato-2-polifosfato
ES538891A0 (es)	1986-01-01	Un metodo de preparar un compuesto de beta-fluoropiridina
ES529031A0 (es)	1985-04-01	Un metodo de preparar nuevos compuestos de benzoilurea
FI951656A7 (fi)	1995-06-01	Menetelmä enantiomeerien erottamiseksi raseemisesta seoksesta
FI911420L (fi)	1991-09-27	Menetelmä terapeuttisesti käyttökelpoisten yhdisteiden valmistamiseksi
ES538736A0 (es)	1985-11-01	Un metodo de sintetizar un silicofosfoaluminato cristalino
HUT40607A (en)	1987-01-28	New process for the optical resolving of racemic mixtures of alpha-naphthyl-propionic acids
ES539062A0 (es)	1986-04-16	Un compuesto de tiofensulfonamida
ZA848639B (en)	1985-06-26	A new process for the optical resolution of racemic mixture of alpha-naphthyl-propionic acids
FI950155L (fi)	1995-01-13	Stereospesifisten GABA-T-inhibiittoreiden raseemisen seoksen entsymaattinen erotus
FI902110A7 (fi)	1990-10-30	Menetelmä peneemiyhdisteiden valmistamiseksi
ES538867A0 (es)	1986-02-01	Un derivado de 5-fluor-3-oxa-prostaciclina
FI942797A7 (fi)	1994-07-25	Menetelmä karbonaattikoostumuksen valmistamiseksi
FI941039A0 (fi)	1994-03-04	Lajittelurummun valmistusmenetelmä
FI893576A7 (fi)	1990-01-28	Uusi menetelmä raseemisten spirohydantoiinien isomeerien erottamiseksi
ES530247A0 (es)	1985-11-01	Un metodo para preparar compuestos de 1, 4-dihidropiridina

Legal Events

Date	Code	Title	Description
2006-03-25	FD	Application lapsed