FI20001108L - Menetelmä raseemisen cis-yhdisteen valmistamiseksi - Google Patents

Menetelmä raseemisen cis-yhdisteen valmistamiseksi Download PDF

Info

Publication number: FI20001108L
Authority: FI; Finland
Prior art keywords: preparing; racemic cis; cis compound; compound; racemic
Prior art date: 1991-01-03

Application number

FI20001108A

Other languages

English (en)

Swedish (sv)

Other versions

FI20001108A7 (fi

Inventor

Dennis M Godek

Charles W Murtiashaw

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-01-03

Filing date

2000-05-10

Publication date

2000-05-10

2000-05-10 Application filed by Pfizer filed Critical Pfizer

2000-05-10 Publication of FI20001108A7 publication Critical patent/FI20001108A7/fi

2000-05-10 Publication of FI20001108L publication Critical patent/FI20001108L/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Indole Compounds (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Apparatuses For Bulk Treatment Of Fruits And Vegetables And Apparatuses For Preparing Feeds (AREA)

FI20001108A 1991-01-03 2000-05-10 Menetelmä raseemisen cis-yhdisteen valmistamiseksi FI20001108L (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/637,102 US5138060A (en)	1991-01-03	1991-01-03	Process and intermediates for preparing azabicyclo(2.2.2)octan-3-imines
PCT/US1991/009186 WO1992012152A1 (en)	1991-01-03	1991-12-18	Process and intermediates for preparing azabicyclo[2.2.2]octan-3-imines

Publications (2)

Publication Number	Publication Date
FI20001108A7 FI20001108A7 (fi)	2000-05-10
FI20001108L true FI20001108L (fi)	2000-05-10

Family

ID=24554545

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
FI933065A FI933065L (fi)	1991-01-03	1991-12-18	Foerfarande foer framstaellning av azabicyklo (2.2.2)oktan-3-iminer och foerfarandet anvaenda mellanprodukter
FI20001109A FI20001109A7 (fi)	1991-01-03	2000-05-10	Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi
FI20001108A FI20001108L (fi)	1991-01-03	2000-05-10	Menetelmä raseemisen cis-yhdisteen valmistamiseksi

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
FI933065A FI933065L (fi)	1991-01-03	1991-12-18	Foerfarande foer framstaellning av azabicyklo (2.2.2)oktan-3-iminer och foerfarandet anvaenda mellanprodukter
FI20001109A FI20001109A7 (fi)	1991-01-03	2000-05-10	Menetelmä cis-yhdisteen raseemisen seoksen resolvoimiseksi

Country Status (21)

Country	Link
US (1)	US5138060A (fi)
EP (1)	EP0565558B1 (fi)
JP (5)	JPH0768244B1 (fi)
KR (1)	KR970001157B1 (fi)
AT (1)	ATE115580T1 (fi)
AU (1)	AU653380B2 (fi)
CA (2)	CA2098989C (fi)
DE (1)	DE69106003T2 (fi)
DK (1)	DK0565558T3 (fi)
ES (1)	ES2065161T3 (fi)
FI (3)	FI933065L (fi)
GR (1)	GR3015021T3 (fi)
HU (1)	HU9301931D0 (fi)
IE (1)	IE65005B1 (fi)
IL (1)	IL100541A0 (fi)
MX (1)	MX9200003A (fi)
NO (1)	NO932431D0 (fi)
NZ (1)	NZ241161A (fi)
PT (1)	PT99970B (fi)
WO (1)	WO1992012152A1 (fi)
ZA (1)	ZA928B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5364943A (en) *	1991-11-27	1994-11-15	Pfizer Inc.	Preparation of substituted piperidines
EP0589924B1 (en) *	1991-06-20	1996-09-04	Pfizer Inc.	Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
DK0613458T3 (da) *	1991-11-12	1998-02-09	Pfizer	Acykliske ethylendiaminderivater som substans P receptorantagonister
PT641328E (pt) *	1992-05-18	2002-04-29	Pfizer	Derivados aza-biciclicos em ponte como antagonistas da substancia p
US5637699A (en) *	1992-06-29	1997-06-10	Merck & Co., Inc.	Process for preparing morpholine tachykinin receptor antagonists
US6048859A (en) *	1992-06-29	2000-04-11	Merck & Co., Inc.	Morpholine and thiomorpholine tachykinin receptor antagonists
US5719147A (en) *	1992-06-29	1998-02-17	Merck & Co., Inc.	Morpholine and thiomorpholine tachykinin receptor antagonists
JPH07506379A (ja) *	1992-08-04	1995-07-13	ファイザー・インコーポレーテッド	物質ｐ受容体アンタゴニストとしての３−ベンジルアミノ−２−フェニル−ピペリジン
US5387595A (en) *	1992-08-26	1995-02-07	Merck & Co., Inc.	Alicyclic compounds as tachykinin receptor antagonists
US5518628A (en) *	1993-11-08	1996-05-21	Shipley Company Inc.	Purification process
IL112778A0 (en) *	1994-03-04	1995-05-26	Merck & Co Inc	Substituted heterocycles, their preparation and pharmaceutical compositions containing them
US6861526B2 (en)	2002-10-16	2005-03-01	Pfizer Inc.	Process for the preparation of (S,S)-cis-2-benzhydryl-3-benzylaminoquinuclidine
US20050136487A1 (en) *	2003-10-27	2005-06-23	Meyer Donald W.	Transmissible spongiform encephalopathy detection in cervids, sheep and goats

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3560510A (en) *	1969-03-05	1971-02-02	Aldrich Chem Co Inc	2-benzhydrylquinuclidines
US3993652A (en) *	1973-07-09	1976-11-23	Air Products And Chemicals, Inc.	Cyclic quaternary hydroxyalkyl phenoxide catalysts for isocyanate reactions
US4203990A (en) *	1979-04-30	1980-05-20	G. D. Searle & Co.	Anti-diarrheal 2-substituted quinuclidines
FR2529548A1 (fr) *	1982-07-02	1984-01-06	Delalande Sa	Nouveaux derives de l'amino-3 quinuclidine, leur procede et leur application en therapeutique
JPS59110656A (ja) *	1982-12-15	1984-06-26	Hiroyuki Nohira	光学活性な１―フェニル―２―（パラ―トリル）エチルアミンの製造方法
DE3604591A1 (de) *	1986-02-14	1987-08-20	Degussa	Verfahren zur herstellung chiraler glycinderivate
JPS6354342A (ja) *	1986-08-26	1988-03-08	Daicel Chem Ind Ltd	（±）−α−エチルベンジルアミンの光学分割方法
JPS63145256A (ja) *	1986-12-09	1988-06-17	Nippon Kayaku Co Ltd	光学活性ホモフエニルアラニンの製造法及び中間体
WO1990005525A1 (en) *	1988-11-23	1990-05-31	Pfizer Inc.	Quinuclidine derivatives as substance p antagonists
DK0585328T3 (da) *	1991-05-22	2002-02-11	Pfizer	Substituerede 3-aminoquinuclidiner

1991
- 1991-01-03 US US07/637,102 patent/US5138060A/en not_active Expired - Lifetime
- 1991-12-18 JP JP4502391A patent/JPH0768244B1/ja active Pending
- 1991-12-18 EP EP92901603A patent/EP0565558B1/en not_active Expired - Lifetime
- 1991-12-18 AT AT92901603T patent/ATE115580T1/de not_active IP Right Cessation
- 1991-12-18 DE DE69106003T patent/DE69106003T2/de not_active Expired - Fee Related
- 1991-12-18 CA CA002098989A patent/CA2098989C/en not_active Expired - Fee Related
- 1991-12-18 DK DK92901603.8T patent/DK0565558T3/da active
- 1991-12-18 AU AU91298/91A patent/AU653380B2/en not_active Expired - Fee Related
- 1991-12-18 JP JP4-502391A patent/JPH0768244B2/ja not_active Expired - Lifetime
- 1991-12-18 ES ES92901603T patent/ES2065161T3/es not_active Expired - Lifetime
- 1991-12-18 WO PCT/US1991/009186 patent/WO1992012152A1/en not_active Ceased
- 1991-12-18 KR KR1019930702007A patent/KR970001157B1/ko not_active Expired - Lifetime
- 1991-12-18 HU HU9301931A patent/HU9301931D0/hu unknown
- 1991-12-18 FI FI933065A patent/FI933065L/fi not_active Application Discontinuation
- 1991-12-18 CA CA002158130A patent/CA2158130C/en not_active Expired - Fee Related
- 1991-12-23 NZ NZ241161A patent/NZ241161A/en unknown
- 1991-12-27 IL IL100541A patent/IL100541A0/xx unknown
1992
- 1992-01-02 IE IE920001A patent/IE65005B1/en not_active IP Right Cessation
- 1992-01-02 PT PT99970A patent/PT99970B/pt not_active IP Right Cessation
- 1992-01-02 ZA ZA928A patent/ZA928B/xx unknown
- 1992-01-02 MX MX9200003A patent/MX9200003A/es unknown
1993
- 1993-07-02 NO NO932431A patent/NO932431D0/no unknown
1994
- 1994-12-26 JP JP6322350A patent/JP2845425B2/ja not_active Expired - Fee Related
- 1994-12-26 JP JP6322353A patent/JP2583026B2/ja not_active Expired - Fee Related
- 1994-12-26 JP JP6322355A patent/JP2703193B2/ja not_active Expired - Fee Related
1995
- 1995-02-08 GR GR950400264T patent/GR3015021T3/el unknown
2000
- 2000-05-10 FI FI20001109A patent/FI20001109A7/fi not_active Application Discontinuation
- 2000-05-10 FI FI20001108A patent/FI20001108L/fi not_active Application Discontinuation

Also Published As

Publication number	Publication date
MX9200003A (es)	1992-07-01
GR3015021T3 (en)	1995-05-31
JPH07316154A (ja)	1995-12-05
HU9301931D0 (en)	1993-12-28
AU9129891A (en)	1992-08-17
JP2703193B2 (ja)	1998-01-26
ATE115580T1 (de)	1994-12-15
JPH07316153A (ja)	1995-12-05
EP0565558A1 (en)	1993-10-20
NO932431L (no)	1993-07-02
FI20001109L (fi)	2000-05-10
JP2845425B2 (ja)	1999-01-13
PT99970B (pt)	1999-06-30
NO932431D0 (no)	1993-07-02
FI20001108A7 (fi)	2000-05-10
KR930703312A (ko)	1993-11-29
JPH0768244B2 (ja)	1995-07-26
CA2158130A1 (en)	1992-07-04
PT99970A (pt)	1993-02-26
DE69106003T2 (de)	1995-04-27
FI933065A0 (fi)	1993-07-02
JP2583026B2 (ja)	1997-02-19
IE920001A1 (en)	1992-07-15
FI933065A7 (fi)	1993-07-02
JPH0768244B1 (fi)	1995-07-26
CA2098989C (en)	1998-02-03
CA2158130C (en)	1998-07-14
DK0565558T3 (da)	1995-03-06
EP0565558B1 (en)	1994-12-14
FI933065L (fi)	1993-07-02
CA2098989A1 (en)	1992-07-04
AU653380B2 (en)	1994-09-29
IE65005B1 (en)	1995-10-04
IL100541A0 (en)	1992-09-06
US5138060A (en)	1992-08-11
JPH07330766A (ja)	1995-12-19
ZA928B (en)	1993-07-02
ES2065161T3 (es)	1995-02-01
NZ241161A (en)	1994-10-26
WO1992012152A1 (en)	1992-07-23
FI20001109A7 (fi)	2000-05-10
DE69106003D1 (de)	1995-01-26
KR970001157B1 (ko)	1997-01-29
JPH05508867A (ja)	1993-12-09

Publication	Publication Date	Title
FI964106L (fi)	1996-10-14	Makeutusaineena käyttökelpoisen aspartaamista johdetun yhdisteen parannettu valmistusmenetelmä
FI932831A7 (fi)	1993-06-18	Menetelmä synteettisen johtosekvenssin valmistamiseksi
FI921021A7 (fi)	1992-09-10	Menetelmä trans-Pt(IV)-yhdisteiden valmistamiseksi
FI925529L (fi)	1992-12-04	En foerbaettrad syntesmetod
FI20000648A7 (fi)	2000-03-20	Menetelmä terapeuttisesti käyttökelpoisen yhdisteen valmistamiseksi, joka sisältää 1-okso-2-isokinoliiniin perustuvan keskuksen
FI943117A7 (fi)	1994-06-29	Menetelmä harjaskimppujen kiinnittämiseksi harjasalustaan
FI925988A7 (fi)	1992-12-31	Menetelmä B-laktaamien valmistamiseksi
FI20001108L (fi)	2000-05-10	Menetelmä raseemisen cis-yhdisteen valmistamiseksi
FI914988A7 (fi)	1992-04-27	Menetelmä ravintoseoksen valmistamiseksi
NO302292B1 (no)	1998-02-16	Forbedret fremgangsmåte for fremstilling av en lineær glukamidsurfaktant
FI942907A7 (fi)	1994-06-17	Menetelmä lipaasin valmistamiseksi
FI920993A7 (fi)	1992-09-07	Menetelmä galliumyhdisteiden valmistamiseksi
FI942954A0 (fi)	1994-06-20	Menetelmä hartsin säätämiseksi
FI940106L (fi)	1994-01-10	Menetelmä sertraliinin valmistamiseksi
FI911207L (fi)	1991-09-28	Menetelmä uuden terapeuttisesti käyttökelpoisen retinoidin valmistamiseksi
FI963050L (fi)	1996-10-01	Menetelmä klavulaanihapposuolan valmistamiseksi
NO922637D0 (no)	1992-07-03	Fremgangsmaate for fremstilling av en kornforfinende tilsats
FI935019L (fi)	1995-05-13	Menetelmä klodronaattivalmisteen valmistamiseksi
FI951656A7 (fi)	1995-06-01	Menetelmä enantiomeerien erottamiseksi raseemisesta seoksesta
FI942797A7 (fi)	1994-07-25	Menetelmä karbonaattikoostumuksen valmistamiseksi
FI923360A7 (fi)	1993-01-25	Menetelmä dimetyyliasetoasetamidin valmistamiseksi
FI972694L (fi)	1997-06-23	Uusi menetelmä sameridiinin valmistamiseksi
IT1260537B (it)	1996-04-09	Guarnizione per un albero
FI922515A7 (fi)	1992-12-01	Parannettu menetelmä glykosyylitransferaasien tuottamiseksi
FI942767A7 (fi)	1994-06-10	Menetelmä ketoni-enantiomeerin valmistamiseksi

Legal Events

Date	Code	Title	Description
2006-03-25	FD	Application lapsed