EP2291366A4 - Préparation de mésylate d imatinib - Google Patents
Préparation de mésylate d imatinibInfo
- Publication number
- EP2291366A4 EP2291366A4 EP09763190A EP09763190A EP2291366A4 EP 2291366 A4 EP2291366 A4 EP 2291366A4 EP 09763190 A EP09763190 A EP 09763190A EP 09763190 A EP09763190 A EP 09763190A EP 2291366 A4 EP2291366 A4 EP 2291366A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- preparation
- imatinib mesylate
- imatinib
- mesylate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 229960003685 imatinib mesylate Drugs 0.000 title 1
- YLMAHDNUQAMNNX-UHFFFAOYSA-N imatinib methanesulfonate Chemical compound CS(O)(=O)=O.C1CN(C)CCN1CC1=CC=C(C(=O)NC=2C=C(NC=3N=C(C=CN=3)C=3C=NC=CC=3)C(C)=CC=2)C=C1 YLMAHDNUQAMNNX-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1285CH2008 | 2008-05-26 | ||
| US9800308P | 2008-09-18 | 2008-09-18 | |
| PCT/US2009/044587 WO2009151899A2 (fr) | 2008-05-26 | 2009-05-20 | Préparation de mésylate d’imatinib |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP2291366A2 EP2291366A2 (fr) | 2011-03-09 |
| EP2291366A4 true EP2291366A4 (fr) | 2012-06-06 |
Family
ID=41417346
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP09763190A Withdrawn EP2291366A4 (fr) | 2008-05-26 | 2009-05-20 | Préparation de mésylate d imatinib |
Country Status (2)
| Country | Link |
|---|---|
| EP (1) | EP2291366A4 (fr) |
| WO (1) | WO2009151899A2 (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL390611A1 (pl) * | 2010-03-04 | 2011-09-12 | Tomasz Koźluk | Sposób otrzymywania polimorficznej formy alfa i nowa forma polimorficzna mesylanu imatinibu |
| WO2011158255A1 (fr) * | 2010-06-16 | 2011-12-22 | Aptuit Laurus Private Limited | Procédé pour la préparation de forme alpha de mésylate d'imatinib stable |
| SI2582689T1 (sl) | 2010-06-18 | 2017-05-31 | Krka, D.D., Novo Mesto | Nova polimorfna oblika imatinib baze in priprava njenih soli |
| EP2598499A2 (fr) * | 2010-07-29 | 2013-06-05 | Dr. Reddy's Laboratories Ltd. | Procédé de préparation de mésylate d'imatinib |
| WO2012014000A1 (fr) * | 2010-07-30 | 2012-02-02 | Ramesh Babu Potluri | Forme cristalline α stable de mésylate d'imatinib et son procédé de synthèse |
| CN102477031B (zh) | 2010-11-30 | 2015-07-15 | 浙江九洲药业股份有限公司 | 一种甲磺酸伊马替尼α晶型的制备方法 |
| JP2014509642A (ja) | 2011-03-31 | 2014-04-21 | アイエヌディー−スイフト ラボラトリーズ リミテッド | イマチニブ及びそのメシル酸塩の生成のための改良方法 |
| ITMI20111309A1 (it) | 2011-07-14 | 2013-01-15 | Italiana Sint Spa | Procedimento di preparazione di imatinib mesilato |
| IN2012DE00728A (fr) | 2012-03-13 | 2015-08-21 | Fresenius Kabi Oncology Ltd | |
| EP2749557A1 (fr) | 2012-12-31 | 2014-07-02 | Deva Holding Anonim Sirketi | Procédé de préparation d'alpha forme polymorphe de mesylate d'imatinib de isopropanol et THF solvatés de mésylate d'imatinib |
| US20160122315A1 (en) * | 2013-06-12 | 2016-05-05 | Shilpa Medicare Limited | Crystalline imatinib mesylate process |
| EP2927223B1 (fr) | 2014-04-04 | 2016-06-29 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Procédé de préparation de l'imatinib et de ses sels, exempt d'impureté génotoxique f |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080090833A1 (en) * | 2006-04-27 | 2008-04-17 | Alexandr Jegorov | Polymorphic forms of imatinib mesylate and processes for preparation of novel crystalline forms as well as amorphous and form alpha |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004106326A1 (fr) * | 2003-06-02 | 2004-12-09 | Hetero Drugs Limited | Nouveaux polymorphismes du mesylate d'imatinib |
| TR200701870T1 (tr) * | 2004-09-02 | 2007-05-21 | Cipla Limited | İmatinib mesilatın kararlı kristal formu ve bu formun hazırlanması için işlem. |
| US20060223816A1 (en) * | 2006-05-08 | 2006-10-05 | Chemagis Ltd. | Imatinib mesylate alpha form and production process therefor |
-
2009
- 2009-05-20 EP EP09763190A patent/EP2291366A4/fr not_active Withdrawn
- 2009-05-20 WO PCT/US2009/044587 patent/WO2009151899A2/fr not_active Ceased
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080090833A1 (en) * | 2006-04-27 | 2008-04-17 | Alexandr Jegorov | Polymorphic forms of imatinib mesylate and processes for preparation of novel crystalline forms as well as amorphous and form alpha |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009151899A2 (fr) | 2009-12-17 |
| EP2291366A2 (fr) | 2011-03-09 |
| WO2009151899A3 (fr) | 2010-02-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP2291366A4 (fr) | Préparation de mésylate d imatinib | |
| ZA201006252B (en) | Preparation of lenalidomide | |
| GB0818498D0 (en) | Provision of inserts | |
| ZA201006679B (en) | Orally-disintergrating solid preparation | |
| EP2438246A4 (fr) | Aspects de construction | |
| IL237160A0 (en) | Stable amorphous forms of imatinib mesylate | |
| GB0922063D0 (en) | Porous silicon | |
| IL212119A0 (en) | Alkylcyclohexylethers of dihydrotetraazabenzoazulenes | |
| IL210149A0 (en) | Isolation of cyclopamine | |
| PL2133419T3 (pl) | Zastosowania beta-dipeptydów cyjanoficyny | |
| PL2401244T3 (pl) | Sposoby produkcji ceramicznych struktur | |
| IL221471A0 (en) | Process for the preparation of alpha form of imatinib mesylate | |
| EP2212251A4 (fr) | Procédés de préparation du clusterboron ® | |
| EP2370414A4 (fr) | Préparation de capécitabine | |
| EP2328873A4 (fr) | Préparation de ranolazine | |
| GB2471253B (en) | Hairdye preparation composition | |
| PL390611A1 (pl) | Sposób otrzymywania polimorficznej formy alfa i nowa forma polimorficzna mesylanu imatinibu | |
| PL385805A1 (pl) | Sposób wytwarzania imatinibu | |
| PL2278890T3 (pl) | Kompozycje fitosteroli o zwiększonej dostępności biologicznej | |
| EP2358693A4 (fr) | Préparation de docétaxel | |
| EP2205525A4 (fr) | Procédé de préparation du clusterboron | |
| EP2205524A4 (fr) | Procédés de fabrication de bore en grappe | |
| ZA201004979B (en) | Extracts of sclerocarya birrea | |
| IL208918A0 (en) | Methods of preparing substituted heterocycles-149 | |
| GB0922023D0 (en) | Preparation of n-monofluoroalkyl compounds |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
| 17P | Request for examination filed |
Effective date: 20101216 |
|
| AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR |
|
| AX | Request for extension of the european patent |
Extension state: AL BA RS |
|
| DAX | Request for extension of the european patent (deleted) | ||
| A4 | Supplementary search report drawn up and despatched |
Effective date: 20120507 |
|
| RIC1 | Information provided on ipc code assigned before grant |
Ipc: C07D 403/08 20060101ALI20120427BHEP Ipc: C07D 403/10 20060101AFI20120427BHEP Ipc: C07D 401/04 20060101ALN20120427BHEP Ipc: C07D 403/02 20060101ALI20120427BHEP |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
| 18D | Application deemed to be withdrawn |
Effective date: 20121201 |