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EE200400015A - Asendatud asaindoolid, neid sisaldav ravimkompositsioon ning ühendite ja kompositsiooni kasutamine proteiini kinaaside inhibeerimiseks - Google Patents

Asendatud asaindoolid, neid sisaldav ravimkompositsioon ning ühendite ja kompositsiooni kasutamine proteiini kinaaside inhibeerimiseks

Info

Publication number
EE200400015A
EE200400015A EEP200400015A EEP200400015A EE200400015A EE 200400015 A EE200400015 A EE 200400015A EE P200400015 A EEP200400015 A EE P200400015A EE P200400015 A EEP200400015 A EE P200400015A EE 200400015 A EE200400015 A EE 200400015A
Authority
EE
Estonia
Prior art keywords
compounds
protein kinases
inhibiting protein
pharmaceutical composition
composition containing
Prior art date
Application number
EEP200400015A
Other languages
English (en)
Estonian (et)
Inventor
Joseph Cox Paul
Nadeem Majid Tahir
Yeun Quai Lai Justine
David Morley Andrew
Amendola Shelley
Daniele Deprets Stephanie
Edlin Chris
J. Gardner Charles
Kominos Dorothea
Leslie Pedgrift Brian
Halley Frank
Alan Gillespy Timothy
Edwards Michael
Frederic Clerc Francois
Nemecek Conception
Houille Olivier
Damour Dominique
Bouchard Herv
Bezard Daniel
Carrez Chantal
Original Assignee
Aventis Pharma Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Limited filed Critical Aventis Pharma Limited
Publication of EE200400015A publication Critical patent/EE200400015A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EEP200400015A 2001-06-21 2002-06-20 Asendatud asaindoolid, neid sisaldav ravimkompositsioon ning ühendite ja kompositsiooni kasutamine proteiini kinaaside inhibeerimiseks EE200400015A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0115109.1A GB0115109D0 (en) 2001-06-21 2001-06-21 Chemical compounds
US30025701P 2001-06-22 2001-06-22
PCT/GB2002/002799 WO2003000688A1 (en) 2001-06-21 2002-06-20 Azaindoles

Publications (1)

Publication Number Publication Date
EE200400015A true EE200400015A (et) 2004-04-15

Family

ID=9917016

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200400015A EE200400015A (et) 2001-06-21 2002-06-20 Asendatud asaindoolid, neid sisaldav ravimkompositsioon ning ühendite ja kompositsiooni kasutamine proteiini kinaaside inhibeerimiseks

Country Status (37)

Country Link
US (2) US6897207B2 (xx)
EP (2) EP1397360A1 (xx)
JP (1) JP4409938B2 (xx)
KR (2) KR100977344B1 (xx)
CN (1) CN100509811C (xx)
AP (1) AP1739A (xx)
AR (1) AR036106A1 (xx)
BG (1) BG108481A (xx)
BR (1) BR0210507A (xx)
CA (1) CA2451678C (xx)
CZ (1) CZ20033444A3 (xx)
EC (1) ECSP034914A (xx)
EE (1) EE200400015A (xx)
GB (1) GB0115109D0 (xx)
HN (1) HN2002000154A (xx)
HR (1) HRP20031069A2 (xx)
HU (1) HUP0400247A2 (xx)
IL (1) IL159445A0 (xx)
JO (1) JO2327B1 (xx)
MA (1) MA27043A1 (xx)
MY (1) MY137099A (xx)
NO (1) NO20035476D0 (xx)
NZ (2) NZ529205A (xx)
OA (1) OA12637A (xx)
PA (1) PA8548701A1 (xx)
PE (1) PE20030155A1 (xx)
PL (1) PL365067A1 (xx)
RU (1) RU2326880C2 (xx)
SI (1) SI21462A (xx)
SK (1) SK15902003A3 (xx)
TN (1) TNSN03110A1 (xx)
TW (1) TWI334417B (xx)
UA (1) UA85660C2 (xx)
UY (1) UY27350A1 (xx)
WO (1) WO2003000688A1 (xx)
YU (1) YU96903A (xx)
ZA (1) ZA200309648B (xx)

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TW202430528A (zh) 2023-01-18 2024-08-01 美商拜歐米富士恩股份有限公司 Ｎ－［４－［４－（４－嗎啉基）－７ｈ－吡咯並［２，３－ｄ］嘧啶－６－基］苯基］－４－［［３（ｒ）－［（１－氧代－２－丙烯－１－基）氨基］－１－哌啶基］甲基］－２－吡啶甲醯胺的結晶形式作為ｍｅｎｉｎ－ｍｌｌ相互作用的共價抑制劑

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RU2326880C2 (ru) 2008-06-20
YU96903A (sh) 2006-08-17
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CN100509811C (zh) 2009-07-08
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US7943616B2 (en) 2011-05-17
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