EE200300365A - Parendatud toimega tsüklilise depsipeptiidi kristallivorm - Google Patents

Parendatud toimega tsüklilise depsipeptiidi kristallivorm

Info

Publication number: EE200300365A
Authority: EE; Estonia
Prior art keywords: crystalline form; cyclic depsipeptide; improved cyclic; improved; depsipeptide
Prior art date: 2001-02-01

Application number

EEP200300365A

Other languages

English (en)

Inventor

Kalbe Jochen

Traeubel Michael

Harder Achim

Von Samson-Himmelstjerna Georg

Original Assignee

Bayer Aktiengesellschaft

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-02-01

Filing date

2002-01-21

Publication date

2003-10-15

2002-01-21 Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft

2003-10-15 Publication of EE200300365A publication Critical patent/EE200300365A/et

2011-12-15 Publication of EE05490B1 publication Critical patent/EE05490B1/et

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Organic Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Gastroenterology & Hepatology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Tropical Medicine & Parasitology (AREA)
Epidemiology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

EEP200300365A 2001-02-01 2002-01-21 Parendatud toimega tsklilise depsipeptiidi kristallivorm EE05490B1 (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10104362A DE10104362A1 (de)	2001-02-01	2001-02-01	Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
PCT/EP2002/000541 WO2002066048A1 (de)	2001-02-01	2002-01-21	Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Publications (2)

Publication Number	Publication Date
EE200300365A true EE200300365A (et)	2003-10-15
EE05490B1 EE05490B1 (et)	2011-12-15

Family

ID=7672376

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200300365A EE05490B1 (et)	2001-02-01	2002-01-21	Parendatud toimega tsklilise depsipeptiidi kristallivorm

Country Status (27)

Country	Link
US (1)	US20040115483A1 (et)
EP (1)	EP1357932B1 (et)
JP (1)	JP2004525111A (et)
KR (2)	KR20030081378A (et)
CN (1)	CN1278735C (et)
AT (1)	ATE284703T1 (et)
AU (1)	AU2002226415B2 (et)
BR (1)	BRPI0206841B8 (et)
CA (1)	CA2436832C (et)
CR (1)	CR7039A (et)
CZ (1)	CZ299564B6 (et)
DE (2)	DE10104362A1 (et)
EE (1)	EE05490B1 (et)
ES (1)	ES2233805T3 (et)
HR (1)	HRP20030635A2 (et)
HU (1)	HU229229B1 (et)
IL (2)	IL157026A0 (et)
MX (1)	MXPA03006866A (et)
NO (1)	NO331289B1 (et)
NZ (1)	NZ527230A (et)
PL (1)	PL213106B1 (et)
PT (1)	PT1357932E (et)
RU (1)	RU2300390C2 (et)
SK (1)	SK286280B6 (et)
UA (1)	UA74623C2 (et)
WO (1)	WO2002066048A1 (et)
ZA (1)	ZA200305864B (et)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20080003546A1 (en) *	2006-06-29	2008-01-03	Dunbar Kimberly L	Animated digital charted yarncraft instruction
US10081656B2 (en)	2015-05-20	2018-09-25	Merial, Inc.	Anthelmintic depsipeptide compounds
HUE065907T2 (hu)	2015-12-28	2024-06-28	Boehringer Ingelheim Vetmedica Gmbh	Anthelmintikus hatású depszipeptid vegyületek
EP3541789A1 (en)	2016-11-16	2019-09-25	Boehringer Ingelheim Animal Health USA Inc.	Anthelmintic depsipeptide compounds
CN114195732A (zh) *	2022-01-04	2022-03-18	丽珠集团福州福兴医药有限公司	一种艾默德斯的单晶型iii及其制备方法
CN114262303A (zh) *	2022-01-04	2022-04-01	丽珠集团福州福兴医药有限公司	一种艾默德斯的单晶型ii及其制备方法
CN115010680A (zh) *	2022-07-13	2022-09-06	丽珠集团福州福兴医药有限公司	单晶型i的艾默德斯及其制备方法
CN114989110A (zh) *	2022-07-13	2022-09-02	丽珠集团福州福兴医药有限公司	单晶型ⅳ的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB2096907A (en) *	1981-04-22	1982-10-27	Exxon Research Engineering Co	Distillation column with steam stripping
ES2166359T3 (es) *	1992-03-17	2002-04-16	Fujisawa Pharmaceutical Co	Derivado de depsipeptido, su produccion y uso.
DE4317458A1 (de) *	1992-06-11	1993-12-16	Bayer Ag	Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) *	1994-01-11	1995-07-13	Bayer Ag	Endoparasitizide Mittel
JP3985050B2 (ja) *	1995-06-30	2007-10-03	アステラス製薬株式会社	デプシペプチド誘導体その製造法およびその新規中間体
CA2232668C (en) *	1995-09-22	2011-10-18	Meiji Seika Kaisha, Ltd.	Novel derivatives of cyclodepsipeptide pf1022 substance
DE69806800T2 (de) *	1997-11-10	2002-12-05	Fujisawa Pharmaceutical Co., Ltd.	Kristall eines depsipeptid-derivates und verfahren zu seiner herstellung
DE10008128A1 (de) *	2000-02-22	2001-08-23	Bayer Ag	Endoparasitizide Mittel
DE10031044A1 (de) *	2000-06-26	2002-01-03	Bayer Ag	Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

2001
- 2001-02-01 DE DE10104362A patent/DE10104362A1/de not_active Withdrawn
2002
- 2002-01-21 MX MXPA03006866A patent/MXPA03006866A/es active IP Right Grant
- 2002-01-21 NZ NZ527230A patent/NZ527230A/xx not_active IP Right Cessation
- 2002-01-21 IL IL15702602A patent/IL157026A0/xx unknown
- 2002-01-21 AT AT02716073T patent/ATE284703T1/de active
- 2002-01-21 ES ES02716073T patent/ES2233805T3/es not_active Expired - Lifetime
- 2002-01-21 CZ CZ20032063A patent/CZ299564B6/cs not_active IP Right Cessation
- 2002-01-21 CN CNB028044843A patent/CN1278735C/zh not_active Expired - Lifetime
- 2002-01-21 WO PCT/EP2002/000541 patent/WO2002066048A1/de not_active Ceased
- 2002-01-21 PT PT02716073T patent/PT1357932E/pt unknown
- 2002-01-21 DE DE50201777T patent/DE50201777D1/de not_active Expired - Lifetime
- 2002-01-21 UA UA2003088108A patent/UA74623C2/uk unknown
- 2002-01-21 PL PL362389A patent/PL213106B1/pl unknown
- 2002-01-21 EP EP02716073A patent/EP1357932B1/de not_active Expired - Lifetime
- 2002-01-21 SK SK988-2003A patent/SK286280B6/sk not_active IP Right Cessation
- 2002-01-21 AU AU2002226415A patent/AU2002226415B2/en not_active Expired
- 2002-01-21 CA CA2436832A patent/CA2436832C/en not_active Expired - Lifetime
- 2002-01-21 EE EEP200300365A patent/EE05490B1/et unknown
- 2002-01-21 KR KR10-2003-7009110A patent/KR20030081378A/ko not_active Ceased
- 2002-01-21 KR KR1020097006790A patent/KR20090041451A/ko not_active Ceased
- 2002-01-21 RU RU2003126589/15A patent/RU2300390C2/ru active
- 2002-01-21 HU HU0302880A patent/HU229229B1/hu unknown
- 2002-01-21 BR BRPI0206841-9 patent/BRPI0206841B8/pt not_active IP Right Cessation
- 2002-01-21 HR HR20030635A patent/HRP20030635A2/hr not_active Application Discontinuation
- 2002-01-21 JP JP2002565606A patent/JP2004525111A/ja active Pending
- 2002-01-21 US US10/470,853 patent/US20040115483A1/en not_active Abandoned
2003
- 2003-07-21 IL IL157026A patent/IL157026A/en unknown
- 2003-07-30 NO NO20033413A patent/NO331289B1/no not_active IP Right Cessation
- 2003-07-30 CR CR7039A patent/CR7039A/es unknown
- 2003-07-30 ZA ZA200305864A patent/ZA200305864B/en unknown

Also Published As

Publication number	Publication date
CN1592631A (zh)	2005-03-09
BR0206841A (pt)	2004-02-25
NO331289B1 (no)	2011-11-21
WO2002066048A1 (de)	2002-08-29
EP1357932B1 (de)	2004-12-15
HU229229B1 (en)	2013-09-30
DE10104362A1 (de)	2002-08-08
BRPI0206841B1 (pt)	2018-02-14
CA2436832C (en)	2013-06-11
CN1278735C (zh)	2006-10-11
HK1075013A1 (en)	2005-12-02
ZA200305864B (en)	2004-08-27
CR7039A (es)	2004-06-08
WO2002066048A8 (de)	2003-11-20
NZ527230A (en)	2005-04-29
PL362389A1 (en)	2004-11-02
ATE284703T1 (de)	2005-01-15
KR20030081378A (ko)	2003-10-17
EE05490B1 (et)	2011-12-15
IL157026A0 (en)	2004-02-08
DE50201777D1 (de)	2005-01-20
HUP0302880A2 (hu)	2003-12-29
JP2004525111A (ja)	2004-08-19
HUP0302880A3 (en)	2005-05-30
CZ20032063A3 (cs)	2003-11-12
HRP20030635A2 (en)	2005-10-31
BRPI0206841B8 (pt)	2021-05-25
CA2436832A1 (en)	2002-08-29
PL213106B1 (pl)	2013-01-31
NO20033413D0 (no)	2003-07-30
EP1357932A1 (de)	2003-11-05
UA74623C2 (en)	2006-01-16
RU2003126589A (ru)	2005-02-27
SK286280B6 (sk)	2008-06-06
MXPA03006866A (es)	2004-05-31
PT1357932E (pt)	2005-04-29
RU2300390C2 (ru)	2007-06-10
CZ299564B6 (cs)	2008-09-03
US20040115483A1 (en)	2004-06-17
ES2233805T3 (es)	2005-06-16
IL157026A (en)	2010-11-30
NO20033413L (no)	2003-09-26
SK9882003A3 (en)	2003-12-02
KR20090041451A (ko)	2009-04-28
AU2002226415B2 (en)	2007-03-22

Publication	Publication Date	Title
SE0200920D0 (sv)	2002-03-25	Novel compounds
ATE433447T1 (de)	2009-06-15	Pyrimiidinverbindungen
SE0301700D0 (sv)	2003-06-10	Novel compounds
JO2282B1 (en)	2005-09-12	Oxazole derivatives
NO20070224L (no)	2007-04-02	2-karbamid-4-fenyltiazolderivater, fremstilling og terapeutisk anvendelse derav
SE0202133D0 (sv)	2002-07-08	Novel compounds
SE0302811D0 (sv)	2003-10-23	Novel compounds
TW200510325A (en)	2005-03-16	2-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof
EA200500203A1 (ru)	2005-08-25	Новый способ синтеза и новая кристаллическая форма агомелатина и фармацевтические композиции, которые её содержат
NO20071642L (no)	2007-06-01	N-Benzensulfonylsubstituerte anilino-pyrimidinanaloger
ATE324371T1 (de)	2006-05-15	N-substituierte heterocyclische nichtaryl- nmda/nr2b-antagonisten
NO20066055L (no)	2007-01-24	Pyridinderivater
NO20050088L (no)	2005-01-06	Kationisk substituerte difenylazefidinoner, fremgangsmate for deres fremstilling, medikamenter inneholdende nevnte forbindelser og anvendelse derav
WO2004069793A3 (en)	2005-01-20	Novel 2-substituted cyclic amines as calcium sensing receptor modulators
NO20062020L (no)	2006-07-10	1-amino-2-oksysubstituerte tetrahydronaftalenderivater, fremgangsmate for fremstilling derav, og deres anvendelse som antiflogistika
SE0401762D0 (sv)	2004-07-05	Novel compounds
MY142044A (en)	2010-08-30	Endoparasiticidal compositions for topical application
MY135850A (en)	2008-07-31	Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds and their use
SE0302139D0 (sv)	2003-07-28	Novel compounds
NO20043016L (no)	2004-07-15	6-aminomorfinan-derivater, fremgangsmate for fremstilling og anvendelse derav
SE0303541D0 (sv)	2003-12-22	New compounds
EE200300365A (et)	2003-10-15	Parendatud toimega tsüklilise depsipeptiidi kristallivorm
SE0303280D0 (sv)	2003-12-05	Novel compounds
SE0403086D0 (sv)	2004-12-17	Compounds
SE0303090D0 (sv)	2003-11-20	Novel compounds

Legal Events

Date	Code	Title	Description
2009-04-15	GB1A	Change in the ownership or in the address of the owner
2013-02-15	GB1A	Change in the ownership or in the address of the owner