NO20033413L - Krystallmodifisering av et syklisk depsipeptid med forbedret aktivitet - Google Patents

Krystallmodifisering av et syklisk depsipeptid med forbedret aktivitet

Info

Publication number: NO20033413L
Authority: NO; Norway
Prior art keywords: cyclic depsipeptide; enhanced activity; crystal modification; depsipeptide; cyclic
Prior art date: 2001-02-01

Application number

NO20033413A

Other languages

English (en)

Other versions

NO331289B1 (no

NO20033413D0 (no

Inventor

Jochen Kalbe

Michael Traeubel

Achim Harder

Georg Von Samson-Himmelstjerna

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-02-01

Filing date

2003-07-30

Publication date

2003-09-26

2003-07-30 Application filed by Bayer Ag filed Critical Bayer Ag

2003-07-30 Publication of NO20033413D0 publication Critical patent/NO20033413D0/no

2003-09-26 Publication of NO20033413L publication Critical patent/NO20033413L/no

2011-11-21 Publication of NO331289B1 publication Critical patent/NO331289B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Organic Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Gastroenterology & Hepatology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Tropical Medicine & Parasitology (AREA)
Epidemiology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO20033413A 2001-02-01 2003-07-30 Anvendelse av krystallmodifisert syklisk depsipeptid for a kontrollere patogene endoparasitter NO331289B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10104362A DE10104362A1 (de)	2001-02-01	2001-02-01	Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
PCT/EP2002/000541 WO2002066048A1 (de)	2001-02-01	2002-01-21	Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Publications (3)

Publication Number	Publication Date
NO20033413D0 NO20033413D0 (no)	2003-07-30
NO20033413L true NO20033413L (no)	2003-09-26
NO331289B1 NO331289B1 (no)	2011-11-21

Family

ID=7672376

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20033413A NO331289B1 (no)	2001-02-01	2003-07-30	Anvendelse av krystallmodifisert syklisk depsipeptid for a kontrollere patogene endoparasitter

Country Status (27)

Country	Link
US (1)	US20040115483A1 (no)
EP (1)	EP1357932B1 (no)
JP (1)	JP2004525111A (no)
KR (2)	KR20030081378A (no)
CN (1)	CN1278735C (no)
AT (1)	ATE284703T1 (no)
AU (1)	AU2002226415B2 (no)
BR (1)	BRPI0206841B8 (no)
CA (1)	CA2436832C (no)
CR (1)	CR7039A (no)
CZ (1)	CZ299564B6 (no)
DE (2)	DE10104362A1 (no)
EE (1)	EE05490B1 (no)
ES (1)	ES2233805T3 (no)
HR (1)	HRP20030635A2 (no)
HU (1)	HU229229B1 (no)
IL (2)	IL157026A0 (no)
MX (1)	MXPA03006866A (no)
NO (1)	NO331289B1 (no)
NZ (1)	NZ527230A (no)
PL (1)	PL213106B1 (no)
PT (1)	PT1357932E (no)
RU (1)	RU2300390C2 (no)
SK (1)	SK286280B6 (no)
UA (1)	UA74623C2 (no)
WO (1)	WO2002066048A1 (no)
ZA (1)	ZA200305864B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20080003546A1 (en) *	2006-06-29	2008-01-03	Dunbar Kimberly L	Animated digital charted yarncraft instruction
US10081656B2 (en)	2015-05-20	2018-09-25	Merial, Inc.	Anthelmintic depsipeptide compounds
HUE065907T2 (hu)	2015-12-28	2024-06-28	Boehringer Ingelheim Vetmedica Gmbh	Anthelmintikus hatású depszipeptid vegyületek
EP3541789A1 (en)	2016-11-16	2019-09-25	Boehringer Ingelheim Animal Health USA Inc.	Anthelmintic depsipeptide compounds
CN114195732A (zh) *	2022-01-04	2022-03-18	丽珠集团福州福兴医药有限公司	一种艾默德斯的单晶型iii及其制备方法
CN114262303A (zh) *	2022-01-04	2022-04-01	丽珠集团福州福兴医药有限公司	一种艾默德斯的单晶型ii及其制备方法
CN115010680A (zh) *	2022-07-13	2022-09-06	丽珠集团福州福兴医药有限公司	单晶型i的艾默德斯及其制备方法
CN114989110A (zh) *	2022-07-13	2022-09-02	丽珠集团福州福兴医药有限公司	单晶型ⅳ的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB2096907A (en) *	1981-04-22	1982-10-27	Exxon Research Engineering Co	Distillation column with steam stripping
ES2166359T3 (es) *	1992-03-17	2002-04-16	Fujisawa Pharmaceutical Co	Derivado de depsipeptido, su produccion y uso.
DE4317458A1 (de) *	1992-06-11	1993-12-16	Bayer Ag	Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) *	1994-01-11	1995-07-13	Bayer Ag	Endoparasitizide Mittel
JP3985050B2 (ja) *	1995-06-30	2007-10-03	アステラス製薬株式会社	デプシペプチド誘導体その製造法およびその新規中間体
CA2232668C (en) *	1995-09-22	2011-10-18	Meiji Seika Kaisha, Ltd.	Novel derivatives of cyclodepsipeptide pf1022 substance
DE69806800T2 (de) *	1997-11-10	2002-12-05	Fujisawa Pharmaceutical Co., Ltd.	Kristall eines depsipeptid-derivates und verfahren zu seiner herstellung
DE10008128A1 (de) *	2000-02-22	2001-08-23	Bayer Ag	Endoparasitizide Mittel
DE10031044A1 (de) *	2000-06-26	2002-01-03	Bayer Ag	Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

2001
- 2001-02-01 DE DE10104362A patent/DE10104362A1/de not_active Withdrawn
2002
- 2002-01-21 MX MXPA03006866A patent/MXPA03006866A/es active IP Right Grant
- 2002-01-21 NZ NZ527230A patent/NZ527230A/xx not_active IP Right Cessation
- 2002-01-21 IL IL15702602A patent/IL157026A0/xx unknown
- 2002-01-21 AT AT02716073T patent/ATE284703T1/de active
- 2002-01-21 ES ES02716073T patent/ES2233805T3/es not_active Expired - Lifetime
- 2002-01-21 CZ CZ20032063A patent/CZ299564B6/cs not_active IP Right Cessation
- 2002-01-21 CN CNB028044843A patent/CN1278735C/zh not_active Expired - Lifetime
- 2002-01-21 WO PCT/EP2002/000541 patent/WO2002066048A1/de not_active Ceased
- 2002-01-21 PT PT02716073T patent/PT1357932E/pt unknown
- 2002-01-21 DE DE50201777T patent/DE50201777D1/de not_active Expired - Lifetime
- 2002-01-21 UA UA2003088108A patent/UA74623C2/uk unknown
- 2002-01-21 PL PL362389A patent/PL213106B1/pl unknown
- 2002-01-21 EP EP02716073A patent/EP1357932B1/de not_active Expired - Lifetime
- 2002-01-21 SK SK988-2003A patent/SK286280B6/sk not_active IP Right Cessation
- 2002-01-21 AU AU2002226415A patent/AU2002226415B2/en not_active Expired
- 2002-01-21 CA CA2436832A patent/CA2436832C/en not_active Expired - Lifetime
- 2002-01-21 EE EEP200300365A patent/EE05490B1/xx unknown
- 2002-01-21 KR KR10-2003-7009110A patent/KR20030081378A/ko not_active Ceased
- 2002-01-21 KR KR1020097006790A patent/KR20090041451A/ko not_active Ceased
- 2002-01-21 RU RU2003126589/15A patent/RU2300390C2/ru active
- 2002-01-21 HU HU0302880A patent/HU229229B1/hu unknown
- 2002-01-21 BR BRPI0206841-9 patent/BRPI0206841B8/pt not_active IP Right Cessation
- 2002-01-21 HR HR20030635A patent/HRP20030635A2/hr not_active Application Discontinuation
- 2002-01-21 JP JP2002565606A patent/JP2004525111A/ja active Pending
- 2002-01-21 US US10/470,853 patent/US20040115483A1/en not_active Abandoned
2003
- 2003-07-21 IL IL157026A patent/IL157026A/en unknown
- 2003-07-30 NO NO20033413A patent/NO331289B1/no not_active IP Right Cessation
- 2003-07-30 CR CR7039A patent/CR7039A/es unknown
- 2003-07-30 ZA ZA200305864A patent/ZA200305864B/en unknown

Also Published As

Publication number	Publication date
CN1592631A (zh)	2005-03-09
BR0206841A (pt)	2004-02-25
NO331289B1 (no)	2011-11-21
WO2002066048A1 (de)	2002-08-29
EP1357932B1 (de)	2004-12-15
HU229229B1 (en)	2013-09-30
DE10104362A1 (de)	2002-08-08
BRPI0206841B1 (pt)	2018-02-14
CA2436832C (en)	2013-06-11
CN1278735C (zh)	2006-10-11
HK1075013A1 (en)	2005-12-02
ZA200305864B (en)	2004-08-27
CR7039A (es)	2004-06-08
WO2002066048A8 (de)	2003-11-20
NZ527230A (en)	2005-04-29
PL362389A1 (en)	2004-11-02
ATE284703T1 (de)	2005-01-15
KR20030081378A (ko)	2003-10-17
EE05490B1 (et)	2011-12-15
IL157026A0 (en)	2004-02-08
DE50201777D1 (de)	2005-01-20
HUP0302880A2 (hu)	2003-12-29
JP2004525111A (ja)	2004-08-19
HUP0302880A3 (en)	2005-05-30
EE200300365A (et)	2003-10-15
CZ20032063A3 (cs)	2003-11-12
HRP20030635A2 (en)	2005-10-31
BRPI0206841B8 (pt)	2021-05-25
CA2436832A1 (en)	2002-08-29
PL213106B1 (pl)	2013-01-31
NO20033413D0 (no)	2003-07-30
EP1357932A1 (de)	2003-11-05
UA74623C2 (en)	2006-01-16
RU2003126589A (ru)	2005-02-27
SK286280B6 (sk)	2008-06-06
MXPA03006866A (es)	2004-05-31
PT1357932E (pt)	2005-04-29
RU2300390C2 (ru)	2007-06-10
CZ299564B6 (cs)	2008-09-03
US20040115483A1 (en)	2004-06-17
ES2233805T3 (es)	2005-06-16
IL157026A (en)	2010-11-30
SK9882003A3 (en)	2003-12-02
KR20090041451A (ko)	2009-04-28
AU2002226415B2 (en)	2007-03-22

Publication	Publication Date	Title
JO2282B1 (en)	2005-09-12	Oxazole derivatives
MX2007000505A (es)	2007-06-25	Derivados de oxindol sustituidos y medicamentos que contienen los mismos.
TW200510325A (en)	2005-03-16	2-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof
MXPA03010134A (es)	2004-03-10	Derivados de ciclohexan-1-4-diamina sustituidos.
MY134892A (en)	2007-12-31	Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and their use
SE0302811D0 (sv)	2003-10-23	Novel compounds
BR0211473A (pt)	2004-10-26	Novos compostos
TW200621737A (en)	2006-07-01	2-carbamide-4-phenylthiazole derivatives, preparation thereof and therapeutic use thereof
SE0401762D0 (sv)	2004-07-05	Novel compounds
NO20065904L (no)	2007-02-20	Terapeutiske forbindelser
NO20050088L (no)	2005-01-06	Kationisk substituerte difenylazefidinoner, fremgangsmate for deres fremstilling, medikamenter inneholdende nevnte forbindelser og anvendelse derav
MX2007003031A (es)	2007-05-23	Compuestos heteroarilo para uso como betamimeticos en el tratamiento de enfermedades de vias respiratorias.
DE50202504D1 (de)	2005-04-21	Neue 4-aminofuropyrimidine und ihre verwendung
MY135850A (en)	2008-07-31	Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds and their use
TW200738658A (en)	2007-10-16	Novel compounds
DK1246808T3 (da)	2011-12-05	1,2-diarylbenzimidazoler til behandling af sygdomme, som er associeret med en mikroglia-aktivering
ATE202483T1 (de)	2001-07-15	Immuntolerante prothrombinkomplex-präparation
DE502005008057D1 (de)	2009-10-15	Substituierte cyclopenten-verbindungen
NO20033413D0 (no)	2003-07-30	Krystallmodifisering av et syklisk depsipeptid med forbedret aktivitet
DE60128100D1 (de)	2007-06-06	Analgetisches arzneimittel
SE0200198D0 (sv)	2002-01-23	New use
MXPA04004090A (es)	2004-07-08	Compuestos substituidos de 1h-quinolin-2-ona.
TW200609222A (en)	2006-03-16	Diazole derivatives
NO20064298L (no)	2006-11-24	Piperazinureaderivater til behandling av endometriose
MXPA03003466A (es)	2004-09-10	Derivados de piranosido.

Legal Events

Date	Code	Title	Description
2014-07-07	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: BAYER INTELLECTUAL PROPERTY GMBH, DE
2022-02-07	MK1K	Patent expired