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EA200200942A1 - Фармацевтические композиции, содержащие производные 3-аминоазетидина, новые производные и способ их получения - Google Patents

Фармацевтические композиции, содержащие производные 3-аминоазетидина, новые производные и способ их получения

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Publication number
EA200200942A1
EA200200942A1 EA200200942A EA200200942A EA200200942A1 EA 200200942 A1 EA200200942 A1 EA 200200942A1 EA 200200942 A EA200200942 A EA 200200942A EA 200200942 A EA200200942 A EA 200200942A EA 200200942 A1 EA200200942 A1 EA 200200942A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
pharmaceutical compositions
compositions containing
denotes
radical
Prior art date
Application number
EA200200942A
Other languages
English (en)
Other versions
EA004649B1 (ru
Inventor
Даниель Ашар
Эрве Бушар
Жан Букерель
Брюно Филош
Серж Гризони
Огюстэн Иттэнжер
Майкл Майерс
Original Assignee
Авентис Фарма С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Авентис Фарма С.А. filed Critical Авентис Фарма С.А.
Publication of EA200200942A1 publication Critical patent/EA200200942A1/ru
Publication of EA004649B1 publication Critical patent/EA004649B1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
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    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
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    • A61P25/16—Anti-Parkinson drugs
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    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Anesthesiology (AREA)
  • Endocrinology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Reproductive Health (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Настоящее изобретение относится к фармацевтическим композициям, содержащим в качестве активного ингредиента соединение формулыв которой Rобозначает радикал -NHCORили -N(R)-Y-R, Y обозначает СО или SO, Rобозначает радикал alk-SO-R, alk-SO-CH=CH-R, Het, замещенный группой -SO-R, или фенил, замещенный группой -SO-Rили -alk-SO-R, Rобозначает атом водорода или радикал алкил, Rобозначает радикал фенилалкил, Het или Ar, новым производным формулы I и их получениям.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200200942A 2000-03-03 2001-03-01 Фармацевтические композиции, содержащие производные 3-аминоазетидина, новые производные и способ их получения EA004649B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0002777A FR2805810B1 (fr) 2000-03-03 2000-03-03 Compositions pharmaceutiques contenant des derives de 3- amino-azetidine, les nouveaux derives et leur preparation
PCT/FR2001/000601 WO2001064633A1 (fr) 2000-03-03 2001-03-01 Compositions pharmaceutiques contenant des derives de 3-amino-azetidine, les nouveaux derives et leur preparation

Publications (2)

Publication Number Publication Date
EA200200942A1 true EA200200942A1 (ru) 2003-02-27
EA004649B1 EA004649B1 (ru) 2004-06-24

Family

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EA200200942A EA004649B1 (ru) 2000-03-03 2001-03-01 Фармацевтические композиции, содержащие производные 3-аминоазетидина, новые производные и способ их получения

Country Status (35)

Country Link
EP (1) EP1263721B1 (ru)
JP (1) JP2003525269A (ru)
KR (1) KR100813740B1 (ru)
CN (1) CN1187325C (ru)
AR (1) AR034405A1 (ru)
AT (1) ATE478840T1 (ru)
AU (2) AU3752601A (ru)
BG (1) BG107057A (ru)
BR (1) BR0108894A (ru)
CA (1) CA2400138A1 (ru)
CY (1) CY1111075T1 (ru)
DE (1) DE60142890D1 (ru)
DK (1) DK1263721T3 (ru)
DZ (1) DZ3311A1 (ru)
EA (1) EA004649B1 (ru)
EE (1) EE05081B1 (ru)
ES (1) ES2351183T3 (ru)
FR (1) FR2805810B1 (ru)
HR (1) HRP20020710A2 (ru)
HU (1) HUP0300350A2 (ru)
IL (2) IL151209A0 (ru)
MA (1) MA26879A1 (ru)
MX (1) MXPA02008346A (ru)
NO (1) NO324523B1 (ru)
NZ (1) NZ521076A (ru)
OA (1) OA12221A (ru)
PL (1) PL365007A1 (ru)
PT (1) PT1263721E (ru)
SI (1) SI1263721T1 (ru)
SK (1) SK12442002A3 (ru)
TW (1) TWI294420B (ru)
UA (1) UA72319C2 (ru)
WO (1) WO2001064633A1 (ru)
YU (1) YU65902A (ru)
ZA (1) ZA200206916B (ru)

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