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DK3789042T3 - Fremgangsmåde til fremstilling af anti-her3-antistof-lægemiddelkonjugat - Google Patents

Fremgangsmåde til fremstilling af anti-her3-antistof-lægemiddelkonjugat Download PDF

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Publication number
DK3789042T3
DK3789042T3 DK20200710.0T DK20200710T DK3789042T3 DK 3789042 T3 DK3789042 T3 DK 3789042T3 DK 20200710 T DK20200710 T DK 20200710T DK 3789042 T3 DK3789042 T3 DK 3789042T3
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Prior art keywords
her3
antibiotics
drug conjugate
preparing anti
preparing
Prior art date
Application number
DK20200710.0T
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English (en)
Inventor
Thore Hettmann
Reimar Abraham
Sabine Blum
Suguru Ueno
Original Assignee
Daiichi Sankyo Co Ltd
Daiichi Sankyo Europe Gmbh
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Application filed by Daiichi Sankyo Co Ltd, Daiichi Sankyo Europe Gmbh filed Critical Daiichi Sankyo Co Ltd
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Publication of DK3789042T3 publication Critical patent/DK3789042T3/da

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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
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