DK2315755T3 - Syntese af dihydrothieno[3,2-d]pyrimidindioler og lignende pyrimidindioler - Google Patents

Syntese af dihydrothieno[3,2-d]pyrimidindioler og lignende pyrimidindioler

Info

Publication number: DK2315755T3
Authority: DK; Denmark
Prior art keywords: pyrimidinediols; dihydrothieno; synthesis; similar; similar pyrimidinediols
Prior art date: 2008-05-13

Application number

DK09736709.8T

Other languages

English (en)

Inventor

Rogelio Perez Frutos

Thomas G Tampone

Jason Alan Mulder

Dhileepkumar Krishnamurthy

Chris Hugh Senanayake

Original Assignee

Boehringer Ingelheim Int

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-05-13

Filing date

2009-05-07

Publication date

2012-10-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41319263&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2315755(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-05-07 Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int

2012-10-15 Application granted granted Critical

2012-10-15 Publication of DK2315755T3 publication Critical patent/DK2315755T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Pulmonology (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK09736709.8T 2008-05-13 2009-05-07 Syntese af dihydrothieno[3,2-d]pyrimidindioler og lignende pyrimidindioler DK2315755T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US5281608P	2008-05-13	2008-05-13
PCT/US2009/043068 WO2009140127A2 (en)	2008-05-13	2009-05-07	SYNTHESIS OF DIHYDROTHIENO[3,2-d]PYRIMIDINE DIOLS AND SIMILAR PYRIMIDINE DIOLS

Publications (1)

Publication Number	Publication Date
DK2315755T3 true DK2315755T3 (da)	2012-10-15

Family

ID=41319263

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK09736709.8T DK2315755T3 (da)	2008-05-13	2009-05-07	Syntese af dihydrothieno[3,2-d]pyrimidindioler og lignende pyrimidindioler

Country Status (31)

Country	Link
US (1)	US8471010B2 (da)
EP (1)	EP2315755B1 (da)
JP (1)	JP5281153B2 (da)
KR (1)	KR20110021764A (da)
CN (1)	CN102026984B (da)
AR (1)	AR071720A1 (da)
AU (1)	AU2009246686B2 (da)
BR (1)	BRPI0912546A2 (da)
CA (1)	CA2722970A1 (da)
CL (1)	CL2009001149A1 (da)
CO (1)	CO6260135A2 (da)
CY (1)	CY1113577T1 (da)
DK (1)	DK2315755T3 (da)
EA (1)	EA019735B1 (da)
EC (1)	ECSP10010571A (da)
ES (1)	ES2392920T3 (da)
HR (1)	HRP20120860T1 (da)
IL (1)	IL208382A0 (da)
MA (1)	MA32312B1 (da)
ME (1)	ME01465B (da)
MX (1)	MX2010011025A (da)
MY (1)	MY152292A (da)
NZ (1)	NZ588484A (da)
PL (1)	PL2315755T3 (da)
PT (1)	PT2315755E (da)
RS (1)	RS52476B (da)
SI (1)	SI2315755T1 (da)
TW (1)	TWI421254B (da)
UA (1)	UA99964C2 (da)
WO (1)	WO2009140127A2 (da)
ZA (1)	ZA201006891B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SA08280783B1 (ar) *	2007-01-11	2011-04-24	استرازينيكا ايه بي	مشتقات بيريدوبيريميدين كمثبطات pde4
WO2013082275A1 (en) *	2011-11-30	2013-06-06	Trustees Of Boston College	Inhibitors of phosphodiesterases 11 (pde11) and methods of use to elevate cortisol production
WO2025131986A1 (en)	2023-12-19	2025-06-26	Boehringer Ingelheim International Gmbh	Novel synthetic steps for the manufacturing method of the pde4b-inhibitor 1-({(5r)-2-[4-(5-chloropyrimidine-2-yl)piperidine-1-yl]-5-oxido-6,7-dihydrothieno[3,2-d]pyrimidine-4-yl}amino)cyclobutyl]methanol

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1470336A1 (de) *	1962-07-04	1969-03-20	Thomae Gmbh Dr K	Neue Dihydrothieno-[3,4-d]-pyrimidine und Verfahren zu ihrer Herstellung
FR2029250A5 (da) *	1969-01-21	1970-10-16	Roussel Uclaf
AR044743A1 (es) *	2002-09-26	2005-10-05	Nihon Nohyaku Co Ltd	Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,
CN101163706A (zh) *	2005-04-21	2008-04-16	贝林格尔·英格海姆国际有限公司	用于治疗炎性疾病的二氢噻吩并嘧啶
US7851468B2 (en) *	2006-05-15	2010-12-14	Cephalon, Inc.	Substituted pyrazolo[3,4-d]pyrimidines

2009
- 2009-05-07 RS RS20120445A patent/RS52476B/sr unknown
- 2009-05-07 EA EA201001775A patent/EA019735B1/ru not_active IP Right Cessation
- 2009-05-07 ME MEP-2012-113A patent/ME01465B/me unknown
- 2009-05-07 EP EP09736709A patent/EP2315755B1/en active Active
- 2009-05-07 BR BRPI0912546A patent/BRPI0912546A2/pt not_active IP Right Cessation
- 2009-05-07 JP JP2011509563A patent/JP5281153B2/ja active Active
- 2009-05-07 HR HRP20120860AT patent/HRP20120860T1/hr unknown
- 2009-05-07 PT PT09736709T patent/PT2315755E/pt unknown
- 2009-05-07 ES ES09736709T patent/ES2392920T3/es active Active
- 2009-05-07 WO PCT/US2009/043068 patent/WO2009140127A2/en not_active Ceased
- 2009-05-07 DK DK09736709.8T patent/DK2315755T3/da active
- 2009-05-07 CA CA2722970A patent/CA2722970A1/en not_active Abandoned
- 2009-05-07 PL PL09736709T patent/PL2315755T3/pl unknown
- 2009-05-07 AU AU2009246686A patent/AU2009246686B2/en not_active Ceased
- 2009-05-07 MX MX2010011025A patent/MX2010011025A/es active IP Right Grant
- 2009-05-07 MY MYPI20105081 patent/MY152292A/en unknown
- 2009-05-07 SI SI200930337T patent/SI2315755T1/sl unknown
- 2009-05-07 CN CN2009801169809A patent/CN102026984B/zh not_active Expired - Fee Related
- 2009-05-07 US US12/989,575 patent/US8471010B2/en active Active
- 2009-05-07 KR KR1020107025268A patent/KR20110021764A/ko not_active Withdrawn
- 2009-05-07 NZ NZ588484A patent/NZ588484A/en not_active IP Right Cessation
- 2009-05-12 TW TW098115740A patent/TWI421254B/zh not_active IP Right Cessation
- 2009-05-12 AR ARP090101712A patent/AR071720A1/es unknown
- 2009-05-12 CL CL2009001149A patent/CL2009001149A1/es unknown
- 2009-07-05 UA UAA201014583A patent/UA99964C2/ru unknown
2010
- 2010-09-28 ZA ZA2010/06891A patent/ZA201006891B/en unknown
- 2010-10-03 IL IL208382A patent/IL208382A0/en unknown
- 2010-10-26 EC EC2010010571A patent/ECSP10010571A/es unknown
- 2010-11-10 CO CO10140646A patent/CO6260135A2/es active IP Right Grant
- 2010-11-12 MA MA33361A patent/MA32312B1/fr unknown
2012
- 2012-10-31 CY CY20121101046T patent/CY1113577T1/el unknown

Also Published As

Publication number	Publication date
TWI421254B (zh)	2014-01-01
CO6260135A2 (es)	2011-03-22
BRPI0912546A2 (pt)	2016-10-18
SI2315755T1 (sl)	2012-10-30
EP2315755B1 (en)	2012-08-08
AR071720A1 (es)	2010-07-07
CN102026984B (zh)	2013-12-25
HK1151524A1 (en)	2012-02-03
MA32312B1 (fr)	2011-05-02
ME01465B (me)	2014-04-20
AU2009246686A1 (en)	2009-11-19
CL2009001149A1 (es)	2010-07-23
US20110130563A1 (en)	2011-06-02
WO2009140127A3 (en)	2010-01-28
JP5281153B2 (ja)	2013-09-04
CN102026984A (zh)	2011-04-20
KR20110021764A (ko)	2011-03-04
EA019735B1 (ru)	2014-05-30
WO2009140127A2 (en)	2009-11-19
PT2315755E (pt)	2012-10-03
RS52476B (sr)	2013-02-28
EP2315755A2 (en)	2011-05-04
US8471010B2 (en)	2013-06-25
ZA201006891B (en)	2011-06-29
CA2722970A1 (en)	2009-11-19
NZ588484A (en)	2012-06-29
AU2009246686B2 (en)	2014-02-13
IL208382A0 (en)	2010-12-30
HRP20120860T1 (hr)	2012-11-30
UA99964C2 (en)	2012-10-25
MY152292A (en)	2014-09-15
ES2392920T3 (es)	2012-12-17
PL2315755T3 (pl)	2013-01-31
TW201006841A (en)	2010-02-16
ECSP10010571A (es)	2010-11-30
MX2010011025A (es)	2010-11-05
JP2011520886A (ja)	2011-07-21
CY1113577T1 (el)	2016-06-22
EA201001775A1 (ru)	2011-06-30

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DK2205608T3 (da)	2013-07-01	Fremstilling af dihydrothieno[3,2-d]pyrimidiner og intermediære anvendt deri
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DK2315755T3 (da)	2012-10-15	Syntese af dihydrothieno[3,2-d]pyrimidindioler og lignende pyrimidindioler
ES1066957Y (es)	2008-07-01	Pulsera
FI20075663A0 (fi)	2007-09-21	Suljettu silta
FR2896995B1 (fr)	2008-04-18	Raquette de paddleball
BRPI0906053A2 (pt)	2015-06-30	"enzima artificial"
FR2932377B1 (fr)	2010-06-25	Prothese d'epaule inversee
ES1075351Y (es)	2011-12-23	Identificador de copas, vasos y similares
ATE516287T1 (de)	2011-07-15	Neuartige chromen-2-on-derivate
FR2938285B1 (fr)	2010-12-03	Panneton d'espagnolette
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UA18696S (uk)	2009-04-10	Браслет
UY3831Q (es)	2009-09-30	Pulsera