DK2342197T3 - Radiomærkede inhibitorer af glycin 1-transportør - Google Patents
Radiomærkede inhibitorer af glycin 1-transportørInfo
- Publication number
- DK2342197T3 DK2342197T3 DK09737459.9T DK09737459T DK2342197T3 DK 2342197 T3 DK2342197 T3 DK 2342197T3 DK 09737459 T DK09737459 T DK 09737459T DK 2342197 T3 DK2342197 T3 DK 2342197T3
- Authority
- DK
- Denmark
- Prior art keywords
- glycin
- radio
- transport
- labeled inhibitors
- inhibitors
- Prior art date
Links
- DHMQDGOQFOQNFH-UHFFFAOYSA-N Glycine Chemical compound NCC(O)=O DHMQDGOQFOQNFH-UHFFFAOYSA-N 0.000 title 2
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/58—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances
- G01N33/60—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances involving radioactive labelled substances
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Physics & Mathematics (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Analytical Chemistry (AREA)
- Cell Biology (AREA)
- Epidemiology (AREA)
- Optics & Photonics (AREA)
- Microbiology (AREA)
- Pain & Pain Management (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Food Science & Technology (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- General Physics & Mathematics (AREA)
- Pathology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08168229 | 2008-11-04 | ||
| PCT/EP2009/064033 WO2010052143A1 (en) | 2008-11-04 | 2009-10-26 | Radiolabelled inhibitors of the glycine 1 transporter |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK2342197T3 true DK2342197T3 (da) | 2013-02-18 |
Family
ID=41402176
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK09737459.9T DK2342197T3 (da) | 2008-11-04 | 2009-10-26 | Radiomærkede inhibitorer af glycin 1-transportør |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US8153679B2 (da) |
| EP (1) | EP2342197B1 (da) |
| JP (1) | JP5543477B2 (da) |
| KR (1) | KR101307671B1 (da) |
| CN (1) | CN102186844B (da) |
| AR (1) | AR074084A1 (da) |
| AU (1) | AU2009312891B2 (da) |
| BR (1) | BRPI0921795B8 (da) |
| CA (1) | CA2739869C (da) |
| CL (1) | CL2011000982A1 (da) |
| DK (1) | DK2342197T3 (da) |
| ES (1) | ES2401221T3 (da) |
| IL (1) | IL211804A (da) |
| MX (1) | MX2011004350A (da) |
| PE (1) | PE20110434A1 (da) |
| PL (1) | PL2342197T3 (da) |
| RU (1) | RU2512529C2 (da) |
| SI (1) | SI2342197T1 (da) |
| TW (1) | TWI449537B (da) |
| WO (1) | WO2010052143A1 (da) |
| ZA (1) | ZA201102521B (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5618047B2 (ja) * | 2010-01-29 | 2014-11-05 | 国立大学法人千葉大学 | ポジトロン断層撮影法およびポジトロン放出化合物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005014563A1 (en) | 2003-08-11 | 2005-02-17 | F. Hoffmann-La Roche Ag | Piperazine with or-substituted phenyl group and their use as glyt1 inhibitors |
| DK1848694T3 (da) * | 2005-02-07 | 2010-01-25 | Hoffmann La Roche | Heterocykliske substituerede phenylmethanoner som inhibitorer af glycintransporter |
| EP1942733B1 (en) * | 2005-09-29 | 2012-03-21 | Merck Sharp & Dohme Corp. | Radiolabeled glycine transporter inhibitors |
-
2009
- 2009-10-26 PE PE2011000892A patent/PE20110434A1/es active IP Right Grant
- 2009-10-26 ES ES09737459T patent/ES2401221T3/es active Active
- 2009-10-26 JP JP2011533694A patent/JP5543477B2/ja not_active Expired - Fee Related
- 2009-10-26 RU RU2011118230/04A patent/RU2512529C2/ru active
- 2009-10-26 MX MX2011004350A patent/MX2011004350A/es active IP Right Grant
- 2009-10-26 EP EP09737459A patent/EP2342197B1/en active Active
- 2009-10-26 BR BRPI0921795A patent/BRPI0921795B8/pt not_active IP Right Cessation
- 2009-10-26 SI SI200930547T patent/SI2342197T1/sl unknown
- 2009-10-26 CN CN200980141350.7A patent/CN102186844B/zh not_active Expired - Fee Related
- 2009-10-26 KR KR1020117010147A patent/KR101307671B1/ko not_active Expired - Fee Related
- 2009-10-26 AU AU2009312891A patent/AU2009312891B2/en not_active Ceased
- 2009-10-26 CA CA2739869A patent/CA2739869C/en not_active Expired - Fee Related
- 2009-10-26 DK DK09737459.9T patent/DK2342197T3/da active
- 2009-10-26 WO PCT/EP2009/064033 patent/WO2010052143A1/en not_active Ceased
- 2009-10-26 PL PL09737459T patent/PL2342197T3/pl unknown
- 2009-10-28 US US12/607,111 patent/US8153679B2/en not_active Expired - Fee Related
- 2009-11-03 TW TW098137279A patent/TWI449537B/zh not_active IP Right Cessation
- 2009-11-03 AR ARP090104237A patent/AR074084A1/es not_active Application Discontinuation
-
2011
- 2011-03-17 IL IL211804A patent/IL211804A/en active IP Right Grant
- 2011-04-05 ZA ZA2011/02521A patent/ZA201102521B/en unknown
- 2011-05-03 CL CL2011000982A patent/CL2011000982A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2739869A1 (en) | 2011-05-14 |
| AR074084A1 (es) | 2010-12-22 |
| PE20110434A1 (es) | 2011-07-01 |
| ZA201102521B (en) | 2012-09-29 |
| SI2342197T1 (sl) | 2013-05-31 |
| JP5543477B2 (ja) | 2014-07-09 |
| CN102186844A (zh) | 2011-09-14 |
| KR101307671B1 (ko) | 2013-09-12 |
| AU2009312891A1 (en) | 2010-05-14 |
| CA2739869C (en) | 2016-09-27 |
| IL211804A0 (en) | 2011-06-30 |
| PL2342197T3 (pl) | 2013-06-28 |
| BRPI0921795B1 (pt) | 2020-10-20 |
| MX2011004350A (es) | 2011-05-23 |
| RU2512529C2 (ru) | 2014-04-10 |
| JP2012507486A (ja) | 2012-03-29 |
| TWI449537B (zh) | 2014-08-21 |
| WO2010052143A1 (en) | 2010-05-14 |
| KR20110063861A (ko) | 2011-06-14 |
| BRPI0921795A2 (pt) | 2016-01-12 |
| EP2342197A1 (en) | 2011-07-13 |
| CL2011000982A1 (es) | 2012-02-03 |
| TW201019964A (en) | 2010-06-01 |
| CN102186844B (zh) | 2014-08-13 |
| EP2342197B1 (en) | 2013-01-16 |
| IL211804A (en) | 2013-11-28 |
| US8153679B2 (en) | 2012-04-10 |
| AU2009312891B2 (en) | 2013-07-11 |
| BRPI0921795B8 (pt) | 2021-07-27 |
| RU2011118230A (ru) | 2012-12-20 |
| US20100111862A1 (en) | 2010-05-06 |
| ES2401221T3 (es) | 2013-04-17 |
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