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DK1881967T3 - Substituerede benzo (D) isoaxol-3-yl-amin-forbindelser som analgetika - Google Patents

Substituerede benzo (D) isoaxol-3-yl-amin-forbindelser som analgetika

Info

Publication number
DK1881967T3
DK1881967T3 DK06753695.3T DK06753695T DK1881967T3 DK 1881967 T3 DK1881967 T3 DK 1881967T3 DK 06753695 T DK06753695 T DK 06753695T DK 1881967 T3 DK1881967 T3 DK 1881967T3
Authority
DK
Denmark
Prior art keywords
isoaxol
analgesics
amine compounds
substituted benzo
compounds
Prior art date
Application number
DK06753695.3T
Other languages
English (en)
Inventor
Beatrix Merla
Robert Frank
Gregor Bahrenberg
Wolfgang Schroeder
Saskia Zemolka
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Application granted granted Critical
Publication of DK1881967T3 publication Critical patent/DK1881967T3/da

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
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    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
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    • A61P17/00Drugs for dermatological disorders
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    • A61P17/04Antipruritics
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    • A61P25/00Drugs for disorders of the nervous system
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36Opioid-abuse
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    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P3/00Drugs for disorders of the metabolism
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
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    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
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    • A61P9/00Drugs for disorders of the cardiovascular system
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Psychology (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
DK06753695.3T 2005-05-18 2006-05-18 Substituerede benzo (D) isoaxol-3-yl-amin-forbindelser som analgetika DK1881967T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102005023589 2005-05-18
DE102005038947A DE102005038947A1 (de) 2005-05-18 2005-08-16 Substituierte Benzo[d]isoxazol-3-yl-amin-Verbindungen und deren Verwendung in Arzneimitteln
PCT/EP2006/004700 WO2006122800A1 (de) 2005-05-18 2006-05-18 Substituierte benzo (d) isoaxol-3-yl-amin-verbindungen als analgetika

Publications (1)

Publication Number Publication Date
DK1881967T3 true DK1881967T3 (da) 2010-08-16

Family

ID=36699120

Family Applications (2)

Application Number Title Priority Date Filing Date
DK06753695.3T DK1881967T3 (da) 2005-05-18 2006-05-18 Substituerede benzo (D) isoaxol-3-yl-amin-forbindelser som analgetika
DK06742972T DK1888541T3 (da) 2005-05-18 2006-05-18 Benzo(d)isoxazol-3-yl-amin-forbindelser og anvendelse af disse som vanilloidreceptorligander

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK06742972T DK1888541T3 (da) 2005-05-18 2006-05-18 Benzo(d)isoxazol-3-yl-amin-forbindelser og anvendelse af disse som vanilloidreceptorligander

Country Status (15)

Country Link
US (2) US7977360B2 (da)
EP (2) EP1881967B1 (da)
JP (2) JP2008540597A (da)
AT (2) ATE466002T1 (da)
AU (1) AU2006249065B2 (da)
CA (2) CA2608386A1 (da)
CY (2) CY1109568T1 (da)
DE (3) DE102005038947A1 (da)
DK (2) DK1881967T3 (da)
ES (2) ES2344272T3 (da)
PL (2) PL1881967T3 (da)
PT (2) PT1888541E (da)
RU (1) RU2416607C2 (da)
SI (2) SI1881967T1 (da)
WO (2) WO2006122800A1 (da)

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EP1881967B1 (de) 2010-04-28
US7696238B2 (en) 2010-04-13
SI1888541T1 (sl) 2010-01-29
JP2008540598A (ja) 2008-11-20
CA2608386A1 (en) 2006-11-23
DE502006004453D1 (de) 2009-09-17
ATE466002T1 (de) 2010-05-15
US7977360B2 (en) 2011-07-12
HK1112238A1 (zh) 2008-08-29
US20090042945A1 (en) 2009-02-12
CY1109568T1 (el) 2014-08-13
WO2006122800A1 (de) 2006-11-23
PT1888541E (pt) 2009-11-10
DE502006006854D1 (de) 2010-06-10
ATE438633T1 (de) 2009-08-15
WO2006122799A1 (de) 2006-11-23
AU2006249065A1 (en) 2006-11-23
AU2006249065B2 (en) 2011-04-21
RU2416607C2 (ru) 2011-04-20
PL1881967T3 (pl) 2010-10-29
CY1110209T1 (el) 2015-01-14
RU2007146385A (ru) 2009-10-27
DE102005038947A1 (de) 2006-11-30
DK1888541T3 (da) 2009-12-07
EP1881967A1 (de) 2008-01-30
ES2331259T3 (es) 2009-12-28
ES2344272T3 (es) 2010-08-23
PL1888541T3 (pl) 2010-01-29
JP2008540597A (ja) 2008-11-20
CA2608773A1 (en) 2006-11-23
US20080176915A1 (en) 2008-07-24
EP1888541B1 (de) 2009-08-05
PT1881967E (pt) 2010-06-30
SI1881967T1 (sl) 2010-08-31
EP1888541A1 (de) 2008-02-20

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