DK1638971T3 - Fremstilling af substitueret Quinoxaliner fra dianilinen med 2,3-dihydroxy-1,4-dioxan - Google Patents
Fremstilling af substitueret Quinoxaliner fra dianilinen med 2,3-dihydroxy-1,4-dioxanInfo
- Publication number
- DK1638971T3 DK1638971T3 DK04734570T DK04734570T DK1638971T3 DK 1638971 T3 DK1638971 T3 DK 1638971T3 DK 04734570 T DK04734570 T DK 04734570T DK 04734570 T DK04734570 T DK 04734570T DK 1638971 T3 DK1638971 T3 DK 1638971T3
- Authority
- DK
- Denmark
- Prior art keywords
- quinoxalins
- dianiline
- dihydroxy
- dioxane
- substituted
- Prior art date
Links
- YLVACWCCJCZITJ-UHFFFAOYSA-N 1,4-dioxane-2,3-diol Chemical compound OC1OCCOC1O YLVACWCCJCZITJ-UHFFFAOYSA-N 0.000 title 1
- QGMGHALXLXKCBD-UHFFFAOYSA-N 4-amino-n-(2-aminophenyl)benzamide Chemical compound C1=CC(N)=CC=C1C(=O)NC1=CC=CC=C1N QGMGHALXLXKCBD-UHFFFAOYSA-N 0.000 title 1
- XSCHRSMBECNVNS-UHFFFAOYSA-N quinoxaline Chemical class N1=CC=NC2=CC=CC=C21 XSCHRSMBECNVNS-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47558903P | 2003-06-04 | 2003-06-04 | |
| PCT/IB2004/001787 WO2004108725A1 (fr) | 2003-06-04 | 2004-05-24 | Preparation de quinoxalines substituees a partir de la dianiline avec du 2,3-dihydroxy-1,4-dioxane |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1638971T3 true DK1638971T3 (da) | 2008-10-27 |
Family
ID=33511699
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK04734570T DK1638971T3 (da) | 2003-06-04 | 2004-05-24 | Fremstilling af substitueret Quinoxaliner fra dianilinen med 2,3-dihydroxy-1,4-dioxan |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20070185327A1 (fr) |
| EP (1) | EP1638971B1 (fr) |
| JP (1) | JP2006526607A (fr) |
| AR (1) | AR044472A1 (fr) |
| AT (1) | ATE405566T1 (fr) |
| BR (1) | BRPI0410613A (fr) |
| CA (1) | CA2527337A1 (fr) |
| CL (1) | CL2004001271A1 (fr) |
| DE (1) | DE602004015986D1 (fr) |
| DK (1) | DK1638971T3 (fr) |
| ES (1) | ES2310730T3 (fr) |
| MX (1) | MXPA05013084A (fr) |
| PL (2) | PL1638971T3 (fr) |
| PT (1) | PT1638971E (fr) |
| SI (1) | SI1638971T1 (fr) |
| TW (1) | TWI251594B (fr) |
| WO (1) | WO2004108725A1 (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0607838A2 (pt) * | 2005-02-24 | 2009-06-13 | Pfizer Prod Inc | preparação de uma quinoxalina substituìda de pureza elevada |
| EP2268639A2 (fr) | 2008-05-22 | 2011-01-05 | Teva Pharmaceutical Industries Ltd. | Tosylate de varénicline, un intermédiaire dans le procédé de préparation du l-tartrate de varénicline |
| US20090318695A1 (en) * | 2008-06-19 | 2009-12-24 | Vinod Kumar Kansal | Processes for the preparation of varenicline and intermediates thereof |
| US8314235B2 (en) | 2008-09-01 | 2012-11-20 | Actavis Group Ptc Ehf | Process for preparing varenicline, varenicline intermediates, pharmaceutically acceptable salts thereof |
| US8178537B2 (en) | 2009-06-22 | 2012-05-15 | Teva Pharmaceutical Industries Ltd. | Solid state forms of varenicline salts and processes for preparation thereof |
| CA2791460A1 (fr) | 2010-03-09 | 2011-09-15 | Actavis Group Ptc Ehf | Varenicline de haute purete ou son sel pharmaceutiquement acceptable sensiblement exempt d'impurete methylvarenicline |
| US20120004239A1 (en) | 2010-06-11 | 2012-01-05 | Medichem, S.A. | Process for Preparing Quinoxaline Derivatives |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6605610B1 (en) * | 1997-12-31 | 2003-08-12 | Pfizer Inc | Aryl fused azapolycyclic compounds |
| EA003190B1 (ru) * | 1997-12-31 | 2003-02-27 | Пфайзер Продактс Инк. | Азаполициклические соединения, конденсированные с арилом |
| CA2443946A1 (fr) * | 2001-04-20 | 2002-10-31 | Pfizer Products Inc. | Procede de preparation d'indenes 1,3-substitues et composes azapolycycliques d'aryle fondus |
-
2004
- 2004-05-24 PL PL04734570T patent/PL1638971T3/pl unknown
- 2004-05-24 ES ES04734570T patent/ES2310730T3/es not_active Expired - Lifetime
- 2004-05-24 DK DK04734570T patent/DK1638971T3/da active
- 2004-05-24 BR BRPI0410613-0A patent/BRPI0410613A/pt not_active IP Right Cessation
- 2004-05-24 CA CA002527337A patent/CA2527337A1/fr not_active Abandoned
- 2004-05-24 PT PT04734570T patent/PT1638971E/pt unknown
- 2004-05-24 JP JP2006508421A patent/JP2006526607A/ja not_active Withdrawn
- 2004-05-24 SI SI200430846T patent/SI1638971T1/sl unknown
- 2004-05-24 DE DE602004015986T patent/DE602004015986D1/de not_active Expired - Fee Related
- 2004-05-24 WO PCT/IB2004/001787 patent/WO2004108725A1/fr not_active Ceased
- 2004-05-24 PL PL378491A patent/PL378491A1/pl not_active Application Discontinuation
- 2004-05-24 MX MXPA05013084A patent/MXPA05013084A/es unknown
- 2004-05-24 EP EP04734570A patent/EP1638971B1/fr not_active Expired - Lifetime
- 2004-05-24 AT AT04734570T patent/ATE405566T1/de not_active IP Right Cessation
- 2004-05-25 CL CL200401271A patent/CL2004001271A1/es unknown
- 2004-06-01 TW TW093115706A patent/TWI251594B/zh not_active IP Right Cessation
- 2004-06-02 US US10/858,600 patent/US20070185327A1/en not_active Abandoned
- 2004-06-03 AR ARP040101901A patent/AR044472A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1638971A1 (fr) | 2006-03-29 |
| SI1638971T1 (sl) | 2008-12-31 |
| TW200500365A (en) | 2005-01-01 |
| TWI251594B (en) | 2006-03-21 |
| CA2527337A1 (fr) | 2004-12-16 |
| WO2004108725A1 (fr) | 2004-12-16 |
| CL2004001271A1 (es) | 2005-04-22 |
| BRPI0410613A (pt) | 2006-06-20 |
| ES2310730T3 (es) | 2009-01-16 |
| PT1638971E (pt) | 2008-10-23 |
| ATE405566T1 (de) | 2008-09-15 |
| US20070185327A1 (en) | 2007-08-09 |
| MXPA05013084A (es) | 2006-03-02 |
| PL378491A1 (pl) | 2006-05-02 |
| PL1638971T3 (pl) | 2009-01-30 |
| EP1638971B1 (fr) | 2008-08-20 |
| JP2006526607A (ja) | 2006-11-24 |
| AR044472A1 (es) | 2005-09-14 |
| DE602004015986D1 (de) | 2008-10-02 |
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