DK0837066T3 - Forbedret fremgangsmåde til fremstilling af penicillin G phenylester - Google Patents
Forbedret fremgangsmåde til fremstilling af penicillin G phenylesterInfo
- Publication number
- DK0837066T3 DK0837066T3 DK96917662T DK96917662T DK0837066T3 DK 0837066 T3 DK0837066 T3 DK 0837066T3 DK 96917662 T DK96917662 T DK 96917662T DK 96917662 T DK96917662 T DK 96917662T DK 0837066 T3 DK0837066 T3 DK 0837066T3
- Authority
- DK
- Denmark
- Prior art keywords
- penicillin
- phenyl ester
- preparation
- improved process
- chem
- Prior art date
Links
- JGSARLDLIJGVTE-MBNYWOFBSA-N Penicillin G Natural products N([C@H]1[C@H]2SC([C@@H](N2C1=O)C(O)=O)(C)C)C(=O)CC1=CC=CC=C1 JGSARLDLIJGVTE-MBNYWOFBSA-N 0.000 title abstract 2
- -1 penicillin G phenyl ester Chemical class 0.000 title abstract 2
- 229940056360 penicillin g Drugs 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/04—Preparation
- C07D499/08—Modification of a carboxyl radical directly attached in position 2, e.g. esterification
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP14752895 | 1995-06-14 | ||
| JP8078296 | 1996-03-07 | ||
| PCT/JP1996/001604 WO1997000259A1 (en) | 1995-06-14 | 1996-06-13 | Improved process for producing penicillin g phenyl ester |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0837066T3 true DK0837066T3 (da) | 2003-11-24 |
Family
ID=26421757
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK96917662T DK0837066T3 (da) | 1995-06-14 | 1996-06-13 | Forbedret fremgangsmåde til fremstilling af penicillin G phenylester |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP0837066B1 (da) |
| JP (1) | JP3377795B2 (da) |
| KR (1) | KR100402595B1 (da) |
| CN (1) | CN1092661C (da) |
| AT (1) | ATE248841T1 (da) |
| DE (1) | DE69629815T2 (da) |
| DK (1) | DK0837066T3 (da) |
| ES (1) | ES2205034T3 (da) |
| PT (1) | PT837066E (da) |
| WO (1) | WO1997000259A1 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5419119B2 (ja) * | 2007-08-20 | 2014-02-19 | 国立大学法人名古屋大学 | エステルの製造法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DD150393A3 (de) * | 1978-04-05 | 1981-09-02 | Wolfgang Krueger | Verfahren zur herstellung halbsynthetischer penicilline und ihrer alkalisalze |
| US5112967A (en) * | 1990-04-27 | 1992-05-12 | Hoffmann-La Roches Inc. | Process for synthesizing antibacterial cephalosporin compounds |
| JP2952015B2 (ja) * | 1990-08-28 | 1999-09-20 | 大塚化学株式会社 | ペニシリン類のエステル化方法 |
| JP2674315B2 (ja) * | 1991-10-15 | 1997-11-12 | 藤沢薬品工業株式会社 | ペニシリンｇエステル |
-
1996
- 1996-06-13 DK DK96917662T patent/DK0837066T3/da active
- 1996-06-13 EP EP96917662A patent/EP0837066B1/en not_active Expired - Lifetime
- 1996-06-13 CN CN96194750A patent/CN1092661C/zh not_active Expired - Fee Related
- 1996-06-13 AT AT96917662T patent/ATE248841T1/de not_active IP Right Cessation
- 1996-06-13 ES ES96917662T patent/ES2205034T3/es not_active Expired - Lifetime
- 1996-06-13 WO PCT/JP1996/001604 patent/WO1997000259A1/ja not_active Ceased
- 1996-06-13 JP JP50291397A patent/JP3377795B2/ja not_active Expired - Fee Related
- 1996-06-13 DE DE69629815T patent/DE69629815T2/de not_active Expired - Fee Related
- 1996-06-13 PT PT96917662T patent/PT837066E/pt unknown
- 1996-06-13 KR KR1019970708137A patent/KR100402595B1/ko not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP0837066A1 (en) | 1998-04-22 |
| DE69629815T2 (de) | 2004-04-08 |
| EP0837066A4 (en) | 1998-11-25 |
| EP0837066B1 (en) | 2003-09-03 |
| ATE248841T1 (de) | 2003-09-15 |
| KR100402595B1 (ko) | 2005-09-02 |
| ES2205034T3 (es) | 2004-05-01 |
| KR19990014793A (ko) | 1999-02-25 |
| CN1187822A (zh) | 1998-07-15 |
| JP3377795B2 (ja) | 2003-02-17 |
| DE69629815D1 (de) | 2003-10-09 |
| WO1997000259A1 (en) | 1997-01-03 |
| PT837066E (pt) | 2004-01-30 |
| CN1092661C (zh) | 2002-10-16 |
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