DK0788500T3 - Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on - Google Patents
Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-onInfo
- Publication number
- DK0788500T3 DK0788500T3 DK95929199T DK95929199T DK0788500T3 DK 0788500 T3 DK0788500 T3 DK 0788500T3 DK 95929199 T DK95929199 T DK 95929199T DK 95929199 T DK95929199 T DK 95929199T DK 0788500 T3 DK0788500 T3 DK 0788500T3
- Authority
- DK
- Denmark
- Prior art keywords
- benzisoxazol
- benzylpiperidin
- pyrrolo
- dihydro
- intermediates
- Prior art date
Links
- -1 1-benzylpiperidin-4-yl Chemical group 0.000 title 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 2
- HUMNYLRZRPPJDN-UHFFFAOYSA-N benzaldehyde Chemical compound O=CC1=CC=CC=C1 HUMNYLRZRPPJDN-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000006719 (C6-C10) aryl (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 239000003638 chemical reducing agent Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 238000010438 heat treatment Methods 0.000 abstract 1
- 229910052500 inorganic mineral Inorganic materials 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000011707 mineral Substances 0.000 abstract 1
- QNGNSVIICDLXHT-UHFFFAOYSA-N para-ethylbenzaldehyde Natural products CCC1=CC=C(C=O)C=C1 QNGNSVIICDLXHT-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32935294A | 1994-10-26 | 1994-10-26 | |
| PCT/IB1995/000755 WO1996013505A1 (en) | 1994-10-26 | 1995-09-13 | PROCESSES AND INTERMEDIATES FOR PREPARING 5,7-DIHYDRO-3-[2-{1-BENZYLPIPERIDIN-4-YL}ETHYL]-6H-PYRROLO-[4,5-f]-1,2-BENZISOXAZOL-6-ONE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0788500T3 true DK0788500T3 (da) | 2004-06-07 |
Family
ID=23284993
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK95929199T DK0788500T3 (da) | 1994-10-26 | 1995-09-13 | Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP0788500B1 (da) |
| JP (1) | JP3048643B2 (da) |
| AT (1) | ATE260922T1 (da) |
| CA (1) | CA2200607C (da) |
| DE (1) | DE69532641T2 (da) |
| DK (1) | DK0788500T3 (da) |
| ES (1) | ES2214506T3 (da) |
| FI (2) | FI113869B (da) |
| PT (1) | PT788500E (da) |
| WO (1) | WO1996013505A1 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1048302A3 (en) * | 1999-04-30 | 2002-07-17 | Pfizer Products Inc. | Radiotracers for in vivo study of acetylcholinesterase and Alzheimer's disease |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI934223L (fi) * | 1991-03-28 | 1993-09-27 | Pfizer | Heterocykliscykliska aminderivat |
-
1995
- 1995-09-13 ES ES95929199T patent/ES2214506T3/es not_active Expired - Lifetime
- 1995-09-13 JP JP8514409A patent/JP3048643B2/ja not_active Expired - Fee Related
- 1995-09-13 CA CA002200607A patent/CA2200607C/en not_active Expired - Fee Related
- 1995-09-13 WO PCT/IB1995/000755 patent/WO1996013505A1/en not_active Ceased
- 1995-09-13 EP EP95929199A patent/EP0788500B1/en not_active Expired - Lifetime
- 1995-09-13 DE DE69532641T patent/DE69532641T2/de not_active Expired - Fee Related
- 1995-09-13 AT AT95929199T patent/ATE260922T1/de not_active IP Right Cessation
- 1995-09-13 DK DK95929199T patent/DK0788500T3/da active
- 1995-09-13 PT PT95929199T patent/PT788500E/pt unknown
-
1997
- 1997-04-25 FI FI971785A patent/FI113869B/fi not_active IP Right Cessation
-
2004
- 2004-04-06 FI FI20040505A patent/FI115301B/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FI971785A0 (fi) | 1997-04-25 |
| DE69532641D1 (de) | 2004-04-08 |
| CA2200607A1 (en) | 1996-05-09 |
| FI20040505A7 (fi) | 2004-04-06 |
| ATE260922T1 (de) | 2004-03-15 |
| JPH10502939A (ja) | 1998-03-17 |
| PT788500E (pt) | 2004-05-31 |
| FI113869B (fi) | 2004-06-30 |
| WO1996013505A1 (en) | 1996-05-09 |
| FI115301B (fi) | 2005-04-15 |
| ES2214506T3 (es) | 2004-09-16 |
| EP0788500B1 (en) | 2004-03-03 |
| FI971785L (fi) | 1997-04-25 |
| EP0788500A1 (en) | 1997-08-13 |
| JP3048643B2 (ja) | 2000-06-05 |
| CA2200607C (en) | 2003-03-18 |
| MX9703076A (es) | 1997-07-31 |
| DE69532641T2 (de) | 2004-08-05 |
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