DK0773921T3 - Fremgangsmåde til fremstilling af en substitueret 2,5-diamino-3-hydroxyhexan - Google Patents
Fremgangsmåde til fremstilling af en substitueret 2,5-diamino-3-hydroxyhexanInfo
- Publication number
- DK0773921T3 DK0773921T3 DK95926318T DK95926318T DK0773921T3 DK 0773921 T3 DK0773921 T3 DK 0773921T3 DK 95926318 T DK95926318 T DK 95926318T DK 95926318 T DK95926318 T DK 95926318T DK 0773921 T3 DK0773921 T3 DK 0773921T3
- Authority
- DK
- Denmark
- Prior art keywords
- independently selected
- loweralkyl
- image
- substituted
- preparation
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- GQYLTNRRTTVXGQ-UHFFFAOYSA-N 2,5-diaminohexan-3-ol Chemical class CC(N)CC(O)C(C)N GQYLTNRRTTVXGQ-UHFFFAOYSA-N 0.000 title 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 150000002431 hydrogen Chemical group 0.000 abstract 3
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 238000009903 catalytic hydrogenation reaction Methods 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- -1 loweralkyl Chemical group 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
- C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
- C07C215/30—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings containing hydroxy groups and carbon atoms of six-membered aromatic rings bound to the same carbon atom of the carbon skeleton
- C07C215/32—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings containing hydroxy groups and carbon atoms of six-membered aromatic rings bound to the same carbon atom of the carbon skeleton containing hydroxy groups and carbon atoms of two six-membered aromatic rings bound to the same carbon atom of the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28310994A | 1994-07-29 | 1994-07-29 | |
| PCT/US1995/009133 WO1996004232A1 (en) | 1994-07-29 | 1995-07-17 | Process for the preparation of a substituted 2.5-diamino-3-hydroxyhexane |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0773921T3 true DK0773921T3 (da) | 2000-05-08 |
Family
ID=23084563
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK95926318T DK0773921T3 (da) | 1994-07-29 | 1995-07-17 | Fremgangsmåde til fremstilling af en substitueret 2,5-diamino-3-hydroxyhexan |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US5672706A (da) |
| EP (1) | EP0773921B1 (da) |
| JP (1) | JPH10503772A (da) |
| AT (1) | ATE187160T1 (da) |
| CA (1) | CA2192836A1 (da) |
| DE (1) | DE69513667T2 (da) |
| DK (1) | DK0773921T3 (da) |
| ES (1) | ES2143058T3 (da) |
| GR (1) | GR3032553T3 (da) |
| PT (1) | PT773921E (da) |
| WO (1) | WO1996004232A1 (da) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60027131D1 (de) | 1999-01-06 | 2006-05-18 | Us Gov Health & Human Serv | Inhibitoren für asparagin-proteasen |
| IT1313624B1 (it) * | 1999-09-21 | 2002-09-09 | Archimica Spa Ora Clariant Lif | Procedimento per la sintesi del ritonavir |
| EP1411045B1 (en) * | 2002-10-18 | 2008-01-16 | Tohru Yokozawa | Process for production of optically active amino alcohols |
| JP2004346008A (ja) * | 2003-05-22 | 2004-12-09 | Sumitomo Chem Co Ltd | Ｎ−モノアルキル−３−ヒドロキシ−３−アリールプロピルアミン類の製造方法および中間体 |
| MX2007003858A (es) | 2004-10-07 | 2007-12-11 | Vitae Pharmaceuticals Inc | Diaminoalcanos inhibidores de proteasa asparticas. |
| JP2006248978A (ja) | 2005-03-10 | 2006-09-21 | Mebiopharm Co Ltd | 新規なリポソーム製剤 |
| TWI411607B (zh) | 2005-11-14 | 2013-10-11 | Vitae Pharmaceuticals Inc | 天門冬胺酸蛋白酶抑制劑 |
| CL2007002689A1 (es) | 2006-09-18 | 2008-04-18 | Vitae Pharmaceuticals Inc | Compuestos derivados de piperidin-1-carboxamida, inhibidores de la renina; compuestos intermediarios; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hipertension, insuficiencia cardiaca, fibrosis cardiaca, entre otras. |
| AR077692A1 (es) | 2009-08-06 | 2011-09-14 | Vitae Pharmaceuticals Inc | Sales de 2-((r)-(3-clorofenil) ((r)-1-((s) -2-(metilamino)-3-((r)-tetrahidro-2h-piran-3-il) propilcarbamoil) piperidin -3-il) metoxi) etilcarbamato de metilo |
| CN111393329A (zh) * | 2020-04-16 | 2020-07-10 | 安徽一帆香料有限公司 | 一种利托那韦和洛匹那韦中间体的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4360684A (en) * | 1981-04-08 | 1982-11-23 | Merck & Co., Inc. | Process for the preparation of (2S)-tetrahydro-2α-methyl-6-oxo-4βα-carboxylic acid |
| IE20010533A1 (en) * | 1990-11-20 | 2003-03-05 | Abbott Lab | Intermediates for preparing retroviral protease inhibiting compounds |
| EP1302468B1 (en) * | 1992-12-29 | 2008-12-17 | Abbott Laboratories | Processes and intermediates for manufacturing retroviral protease inhibiting compounds |
-
1995
- 1995-07-17 EP EP95926318A patent/EP0773921B1/en not_active Expired - Lifetime
- 1995-07-17 WO PCT/US1995/009133 patent/WO1996004232A1/en not_active Ceased
- 1995-07-17 DK DK95926318T patent/DK0773921T3/da active
- 1995-07-17 AT AT95926318T patent/ATE187160T1/de not_active IP Right Cessation
- 1995-07-17 DE DE69513667T patent/DE69513667T2/de not_active Expired - Fee Related
- 1995-07-17 CA CA002192836A patent/CA2192836A1/en not_active Abandoned
- 1995-07-17 PT PT95926318T patent/PT773921E/pt unknown
- 1995-07-17 JP JP8506551A patent/JPH10503772A/ja not_active Withdrawn
- 1995-07-17 ES ES95926318T patent/ES2143058T3/es not_active Expired - Lifetime
-
1996
- 1996-04-17 US US08/633,605 patent/US5672706A/en not_active Expired - Fee Related
-
2000
- 2000-02-02 GR GR20000400249T patent/GR3032553T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PT773921E (pt) | 2000-05-31 |
| US5672706A (en) | 1997-09-30 |
| ES2143058T3 (es) | 2000-05-01 |
| EP0773921B1 (en) | 1999-12-01 |
| JPH10503772A (ja) | 1998-04-07 |
| EP0773921A1 (en) | 1997-05-21 |
| DE69513667T2 (de) | 2000-07-06 |
| GR3032553T3 (en) | 2000-05-31 |
| WO1996004232A1 (en) | 1996-02-15 |
| MX9700720A (es) | 1997-09-30 |
| DE69513667D1 (de) | 2000-01-05 |
| ATE187160T1 (de) | 1999-12-15 |
| CA2192836A1 (en) | 1996-02-15 |
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