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DK0761218T3 - Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat - Google Patents

Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat

Info

Publication number
DK0761218T3
DK0761218T3 DK96202848T DK96202848T DK0761218T3 DK 0761218 T3 DK0761218 T3 DK 0761218T3 DK 96202848 T DK96202848 T DK 96202848T DK 96202848 T DK96202848 T DK 96202848T DK 0761218 T3 DK0761218 T3 DK 0761218T3
Authority
DK
Denmark
Prior art keywords
amoxycillin
clavulanate
polymer
preparation
coated tablets
Prior art date
Application number
DK96202848T
Other languages
English (en)
Inventor
Creighton Pierce Conley
Nigel Philip Davidson
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10754044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0761218(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Application granted granted Critical
Publication of DK0761218T3 publication Critical patent/DK0761218T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK96202848T 1994-04-23 1995-04-19 Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat DK0761218T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9408117A GB9408117D0 (en) 1994-04-23 1994-04-23 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
DK0761218T3 true DK0761218T3 (da) 2000-12-18

Family

ID=10754044

Family Applications (4)

Application Number Title Priority Date Filing Date
DK00204182T DK1093813T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til at fremstille polymer-overtrukket tablet, der omfatter amoxycillin og clavunalat, belagt med et vandigt polymerfilmovertræk
DK95917937T DK0758235T3 (da) 1994-04-23 1995-04-19 Polymercoatet tablet omfattende amoxycillin og clavulanat
DK99200891T DK0978276T3 (da) 1994-04-23 1995-04-19 Polymerovertrukken tablet omfattende amoxycillin og clavulanat
DK96202848T DK0761218T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat

Family Applications Before (3)

Application Number Title Priority Date Filing Date
DK00204182T DK1093813T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til at fremstille polymer-overtrukket tablet, der omfatter amoxycillin og clavunalat, belagt med et vandigt polymerfilmovertræk
DK95917937T DK0758235T3 (da) 1994-04-23 1995-04-19 Polymercoatet tablet omfattende amoxycillin og clavulanat
DK99200891T DK0978276T3 (da) 1994-04-23 1995-04-19 Polymerovertrukken tablet omfattende amoxycillin og clavulanat

Country Status (35)

Country Link
US (1) US6051255A (da)
EP (5) EP0761218B1 (da)
JP (1) JP3622975B2 (da)
CN (1) CN1134258C (da)
AP (2) AP564A (da)
AT (6) ATE196845T1 (da)
AU (1) AU684949B2 (da)
BG (1) BG62842B1 (da)
BR (1) BR9507502A (da)
CA (1) CA2188496A1 (da)
CZ (2) CZ294168B6 (da)
DE (5) DE29522153U1 (da)
DK (4) DK1093813T3 (da)
DZ (1) DZ1876A1 (da)
ES (4) ES2161288T3 (da)
FI (1) FI964249L (da)
GB (1) GB9408117D0 (da)
GR (2) GR3035031T3 (da)
HK (1) HK1050992A1 (da)
HU (1) HU228399B1 (da)
IL (1) IL113433A (da)
MA (1) MA23528A1 (da)
MY (1) MY115351A (da)
NO (1) NO310703B1 (da)
NZ (1) NZ285080A (da)
OA (1) OA10377A (da)
PL (1) PL316966A1 (da)
PT (4) PT758235E (da)
RO (1) RO116997B1 (da)
RU (1) RU2152213C1 (da)
SA (1) SA95160343B1 (da)
SI (1) SI0758235T1 (da)
SK (1) SK282594B6 (da)
WO (1) WO1995028927A1 (da)
ZA (1) ZA953236B (da)

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* Cited by examiner, † Cited by third party
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DZ2028A1 (fr) * 1995-05-03 2002-10-23 Smithkline Beecham Plc Médicaments destinés au traitement d'infections bactériennes en pédiatrie.
US20030109503A1 (en) * 1995-06-06 2003-06-12 Smithkline Beecham P.L.C. Pharmaceutical formulations comprising clavulanic acid alone or in combination with other beta-lactam antibiotics
NZ337247A (en) * 1995-09-07 2001-05-25 Smithkline Beecham Corp Pharmaceutical tablet formulation comprising 875mg amoxycillin
AT403375B (de) * 1995-11-15 1998-01-26 Biochemie Gmbh Verfahren zur fällung von alkalisalzen der clavulansäure
AT407701B (de) * 1996-08-12 2001-05-25 Biochemie Gmbh Zur direkttablettierung geeignete mischung, die als wesentliche komponenten amoxicillin-trihydrat und das kaliumsalz der clavulansäure enthält und verfahren zur herstellung dieser mischung
TWI225402B (en) * 1996-03-13 2004-12-21 Biochemie Gmbh Auxiliary-free agglomerates
GB9613470D0 (en) 1996-06-27 1996-08-28 Ciba Geigy Ag Small solid oral dosage form
GB9616536D0 (en) 1996-08-06 1996-09-25 Quadrant Holdings Cambridge Co-amoxiclav dosage form
GB9617780D0 (en) * 1996-08-24 1996-10-02 Smithkline Beecham Plc Method of treatment
WO1998034598A2 (en) * 1997-02-07 1998-08-13 Gist-Brocades B.V. Homogeneous granulated formulations for dose sipping technology
CA2280857A1 (en) * 1997-02-14 1998-08-20 Smithkline Beecham Laboratoires Pharmaceutiques Pharmaceutical formulations comprising amoxocyllin and clavulanate
US20030124187A1 (en) * 1997-02-14 2003-07-03 Smithkline Beecham Laboratoires Pharmaceutiques, Pharmaceutical formulations comprising amoxycillin and clavulanate
AU9540898A (en) * 1997-08-29 1999-03-22 Dsm N.V. Granules free of excipients
US6395298B1 (en) 1997-10-31 2002-05-28 Pharmacia Corporation Gellan gum tablet coating
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EP1044680B1 (en) * 1999-04-13 2003-06-11 Beecham Pharmaceuticals (Pte) Limited Novel method of treatment using a high dosage regimen of amoxycillin and potassium clavulanate
US7250176B1 (en) * 1999-04-13 2007-07-31 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
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US20030070584A1 (en) * 2001-05-15 2003-04-17 Cynthia Gulian Dip coating compositions containing cellulose ethers
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AU2003210925A1 (en) * 2002-02-07 2003-09-02 Rutgers, The State University Antibiotic polymers
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ES2263949T3 (es) * 2002-02-14 2006-12-16 Glaxo Group Limited Composicion farmaceutica que comprende n-((1-n-butil-4-piperidinil)mentil)-3,4-dihidro-2h-(1,3)oxazino (3,2-aindol-10-carboxamida o una sal de la misma y procedimiento para su preparacon que comprende granulacion por via seca.
US20060083759A1 (en) * 2002-07-17 2006-04-20 Aleksander Resman Stabilization of the profile of release of active substances from a formulation
US8637512B2 (en) 2002-07-29 2014-01-28 Glaxo Group Limited Formulations and method of treatment
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US8778924B2 (en) * 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
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CL2008003230A1 (es) * 2007-11-01 2009-11-27 Sanofi Aventis Healthcare Pty Ltd Composicion de recubrimiento de tableta que comprende polimero celulosico, plastificante, edulcorante y composicion de sabor en polvo la que comprende saborizante asociado con portador solido; fluido de recubrimiento de tableta que comprende dicha composicion; tableta farmaceutica; proceso de preparacion de dicha tableta.
SI2477611T1 (sl) * 2009-09-18 2017-07-31 Sanofi Formulacije tablete (Z)-2-ciano-3-hidroksi-but-2-enojska kislina-(4'-trifluormetilfenil)-amida z izboljšano stabilnostjo
TR200909787A2 (tr) 2009-12-25 2011-07-21 Bi̇lgi̇ç Mahmut Üçüncü kuşak bir sefalosporin ve klavulanik asit içeren farmasötik formülasyonlar.
TR201000686A1 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Bakteriyel enfeksiyonların tedavisinde suda çözünebilir sefdinir ve klavulanik asit formülasyonları.@
TR201000687A1 (tr) 2010-01-29 2011-08-22 Bi̇lgi̇ç Mahmut Aktif madde olarak sefiksim ve klavulanik asit içeren efervesan formülasyonlar
TR201000688A2 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Aktif madde olarak sefaklor ve klavulanik asit içeren efervesan formülasyonlar.
JP6041591B2 (ja) * 2011-09-13 2016-12-14 大日本住友製薬株式会社 イルベサルタンとアムロジピンまたはその塩を含有する安定化された医薬組成物
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EP0080862B1 (en) * 1981-12-02 1985-09-25 Beecham Group Plc Pharmaceutical formulation comprising beta-lactam antibiotics
GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
EP1044680B1 (en) * 1999-04-13 2003-06-11 Beecham Pharmaceuticals (Pte) Limited Novel method of treatment using a high dosage regimen of amoxycillin and potassium clavulanate
AU2001292185A1 (en) * 2000-10-12 2002-04-22 Beecham Pharmaceuticals (Pte) Limited Formulation containing amoxicillin

Also Published As

Publication number Publication date
DE69528204D1 (de) 2002-10-17
EP0978276B1 (en) 2002-09-11
DE29522153U1 (de) 2000-04-06
FI964249A7 (fi) 1996-10-22
HK1027024A1 (en) 2001-01-05
DE69519093T2 (de) 2001-07-19
WO1995028927A1 (en) 1995-11-02
JPH09512027A (ja) 1997-12-02
ZA953236B (en) 1995-12-27
AT5349U1 (de) 2002-06-25
DE69528608T2 (de) 2003-06-26
EP0978276A3 (en) 2000-04-12
ATE226074T1 (de) 2002-11-15
DE69528204T2 (de) 2003-08-07
CN1149829A (zh) 1997-05-14
IL113433A (en) 2003-06-24
DK1093813T3 (da) 2003-02-17
NZ285080A (en) 1998-05-27
EP1243267A2 (en) 2002-09-25
CZ309096A3 (en) 1997-04-16
EP1243267A3 (en) 2002-10-30
HK1009936A1 (en) 1999-06-11
BG100933A (en) 1997-07-31
DK0758235T3 (da) 2001-10-29
HK1036404A1 (en) 2002-01-04
OA10377A (en) 2001-11-21
AT5350U1 (de) 2002-06-25
IL113433A0 (en) 1995-07-31
HUT76335A (en) 1997-08-28
DE69521799D1 (de) 2001-08-23
NO964488D0 (no) 1996-10-22
ATE196845T1 (de) 2000-10-15
AP9600868A0 (en) 1996-10-31
PT758235E (pt) 2001-10-31
GR3035031T3 (en) 2001-03-30
SK135496A3 (en) 1997-05-07
DE69521799T2 (de) 2002-06-13
SA95160343B1 (ar) 2005-05-04
US6051255A (en) 2000-04-18
AP564A (en) 1996-11-21
EP0758235A1 (en) 1997-02-19
GR3036844T3 (en) 2002-01-31
HU9602922D0 (en) 1996-12-30
CA2188496A1 (en) 1995-11-02
CN1134258C (zh) 2004-01-14
JP3622975B2 (ja) 2005-02-23
EP1093813A3 (en) 2001-05-30
EP1093813B1 (en) 2002-10-16
ATE223706T1 (de) 2002-09-15
PL316966A1 (en) 1997-03-03
PT761218E (pt) 2001-03-30
HK1021860A1 (en) 2000-07-07
CZ11376U1 (cs) 2001-07-12
AU684949B2 (en) 1998-01-08
ES2161288T3 (es) 2001-12-01
DZ1876A1 (fr) 2002-02-17
MY115351A (en) 2003-05-31
ES2182754T3 (es) 2003-03-16
EP0758235B1 (en) 2001-07-18
ATE203161T1 (de) 2001-08-15
DK0978276T3 (da) 2003-01-20
FI964249A0 (fi) 1996-10-22
RO116997B1 (ro) 2001-09-28
BG62842B1 (bg) 2000-09-29
EP0978276A2 (en) 2000-02-09
CZ294168B6 (cs) 2004-10-13
BR9507502A (pt) 1997-09-02
GB9408117D0 (en) 1994-06-15
FI964249L (fi) 1996-10-22
MA23528A1 (fr) 1995-12-31
HK1050992A1 (en) 2003-07-18
ES2180251T3 (es) 2003-02-01
DE69519093D1 (de) 2000-11-16
PT978276E (pt) 2003-01-31
ES2152485T3 (es) 2001-02-01
SK282594B6 (sk) 2002-10-08
PT1093813E (pt) 2003-02-28
SI0758235T1 (en) 2001-10-31
EP0761218B1 (en) 2000-10-11
NO310703B1 (no) 2001-08-20
HU228399B1 (en) 2013-03-28
NO964488L (no) 1996-12-17
EP0761218A1 (en) 1997-03-12
AU2406895A (en) 1995-11-16
AP9500733A0 (en) 1995-04-30
RU2152213C1 (ru) 2000-07-10
EP1093813A2 (en) 2001-04-25
DE69528608D1 (de) 2002-11-21

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