DE69920683D1 - Selektiv auf den cb2-rezeptor wirkende cannabinoide - Google Patents
Selektiv auf den cb2-rezeptor wirkende cannabinoideInfo
- Publication number
- DE69920683D1 DE69920683D1 DE69920683T DE69920683T DE69920683D1 DE 69920683 D1 DE69920683 D1 DE 69920683D1 DE 69920683 T DE69920683 T DE 69920683T DE 69920683 T DE69920683 T DE 69920683T DE 69920683 D1 DE69920683 D1 DE 69920683D1
- Authority
- DE
- Germany
- Prior art keywords
- receptor
- selective
- cannabinoids
- cannabinoid
- novel
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 229930003827 cannabinoid Natural products 0.000 title abstract 6
- 239000003557 cannabinoid Substances 0.000 title abstract 6
- 229940065144 cannabinoids Drugs 0.000 title abstract 3
- 102000009135 CB2 Cannabinoid Receptor Human genes 0.000 abstract 1
- 108010073376 CB2 Cannabinoid Receptor Proteins 0.000 abstract 1
- 125000002837 carbocyclic group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 210000000987 immune system Anatomy 0.000 abstract 1
- 230000001506 immunosuppresive effect Effects 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/78—Ring systems having three or more relevant rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8412998P | 1998-05-04 | 1998-05-04 | |
| US84129P | 1998-05-04 | ||
| PCT/US1999/009806 WO1999057107A2 (en) | 1998-05-04 | 1999-05-04 | Cannabinoids selective for the cb2 receptor |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69920683D1 true DE69920683D1 (de) | 2004-11-04 |
| DE69920683T2 DE69920683T2 (de) | 2005-04-07 |
Family
ID=22183058
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69920683T Expired - Fee Related DE69920683T2 (de) | 1998-05-04 | 1999-05-04 | Selektiv auf den CB2-Rezeptor wirkende Cannabinoide |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US6166066A (de) |
| EP (1) | EP1076653B1 (de) |
| AT (1) | ATE277921T1 (de) |
| CA (1) | CA2340444A1 (de) |
| DE (1) | DE69920683T2 (de) |
| ES (1) | ES2224658T3 (de) |
| WO (1) | WO1999057107A2 (de) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE277921T1 (de) * | 1998-05-04 | 2004-10-15 | Univ Connecticut | Selektiv auf den cb2-rezeptor wirkende cannabinoide |
| US20010009965A1 (en) * | 1998-05-04 | 2001-07-26 | Alexandros Makriyannis | Novel analgesic and immunomodulatory cannabinoids |
| US7897598B2 (en) | 1998-06-09 | 2011-03-01 | Alexandros Makriyannis | Inhibitors of the anandamide transporter |
| US7589220B2 (en) * | 1998-06-09 | 2009-09-15 | University Of Connecticut | Inhibitors of the anandamide transporter |
| US7276613B1 (en) | 1998-11-24 | 2007-10-02 | University Of Connecticut | Retro-anandamides, high affinity and stability cannabinoid receptor ligands |
| US7161016B1 (en) | 1998-11-24 | 2007-01-09 | University Of Connecticut | Cannabimimetic lipid amides as useful medications |
| US20070179135A1 (en) * | 2006-01-05 | 2007-08-02 | Travis Craig R | Cannabinoid derivatives |
| AU778159B2 (en) | 1999-10-18 | 2004-11-18 | University Of Connecticut, The | Peripheral cannabinoid receptor (CB2) selective ligands |
| US6900236B1 (en) | 1999-10-18 | 2005-05-31 | University Of Connecticut | Cannabimimetic indole derivatives |
| US8084467B2 (en) * | 1999-10-18 | 2011-12-27 | University Of Connecticut | Pyrazole derivatives as cannabinoid receptor antagonists |
| US7393842B2 (en) * | 2001-08-31 | 2008-07-01 | University Of Connecticut | Pyrazole analogs acting on cannabinoid receptors |
| US7741365B2 (en) * | 1999-10-18 | 2010-06-22 | University Of Connecticut | Peripheral cannabinoid receptor (CB2) selective ligands |
| US6943266B1 (en) * | 1999-10-18 | 2005-09-13 | University Of Connecticut | Bicyclic cannabinoid agonists for the cannabinoid receptor |
| US7119108B1 (en) * | 1999-10-18 | 2006-10-10 | University Of Connecticut | Pyrazole derivatives as cannabinoid receptor antagonists |
| KR20030008153A (ko) * | 2000-06-22 | 2003-01-24 | 파모스 코포레이션 | 신규 비-향정신성 카나비노이드 |
| US7235584B2 (en) * | 2000-06-22 | 2007-06-26 | Pharmos Corporation | Non-psychotropic cannabinoids |
| EP1361876A4 (de) | 2001-01-26 | 2004-03-31 | Univ Connecticut | Neue cannabimimetische liganden |
| WO2002060447A1 (en) | 2001-01-29 | 2002-08-08 | University Of Connecticut | Receptor selective cannabimimetic aminoalkylindoles |
| AU2002320430A1 (en) * | 2001-07-13 | 2003-01-29 | University Of Connecticut | Novel bicyclic and tricyclic cannabinoids |
| US7666867B2 (en) * | 2001-10-26 | 2010-02-23 | University Of Connecticut | Heteroindanes: a new class of potent cannabimimetic ligands |
| CA2468794A1 (en) * | 2001-12-07 | 2003-06-19 | Virginia Commonwealth University | Treatment of neoplasia |
| WO2003075917A1 (en) | 2002-03-08 | 2003-09-18 | Signal Pharmaceuticals, Inc. | Combination therapy for treating, preventing or managing proliferative disorders and cancers |
| WO2004103410A1 (en) | 2002-06-06 | 2004-12-02 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Methods compositions and articles of manufacture for modulating bone growth |
| US7183313B2 (en) | 2002-08-23 | 2007-02-27 | University Of Connecticut | Keto cannabinoids with therapeutic indications |
| IL160420A0 (en) * | 2004-02-16 | 2004-07-25 | Yissum Res Dev Co | Treating or preventing diabetes with cannabidiol |
| WO2005123053A2 (en) * | 2004-06-22 | 2005-12-29 | Pharmos Limited | Use of cb2 receptors agonists for the treatment of huntington’s disease |
| US7781650B2 (en) * | 2007-04-30 | 2010-08-24 | Monsanto Technology Llc | Plants and seeds of corn variety CV202909 |
| US9575319B2 (en) | 2014-03-10 | 2017-02-21 | Ion Virtual Technology Corporation | Method and system for reducing motion blur when experiencing virtual or augmented reality environments |
| US10239808B1 (en) | 2016-12-07 | 2019-03-26 | Canopy Holdings, LLC | Cannabis extracts |
| JP2020524679A (ja) | 2017-06-20 | 2020-08-20 | イッサム リサーチ デベロップメント カンパニー オブ ザ ヘブリュー ユニバーシティー オブ エルサレム エルティーディー． | カンナビジオール酸エステル組成物およびその使用 |
| EP3745884A1 (de) | 2018-01-31 | 2020-12-09 | Canopy Holdings, Llc | Hanfpulver |
| US11040932B2 (en) | 2018-10-10 | 2021-06-22 | Treehouse Biotech, Inc. | Synthesis of cannabigerol |
| MX2021010875A (es) | 2019-03-12 | 2021-12-10 | Epm Ip Inc | Composiciones de éster de ácido cannabinoide y sus usos. |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3915996A (en) * | 1972-10-16 | 1975-10-28 | Abbott Lab | Process for making benzopyrans |
| US3886184A (en) * | 1973-08-03 | 1975-05-27 | Lilly Co Eli | Aminodibenzo(b,d)pyrans |
| US4833073A (en) * | 1987-01-27 | 1989-05-23 | Hoffmann-La Roche Inc. | Immunoassay for tetrahydrocannabinol metabolites |
| US5440052A (en) * | 1993-08-06 | 1995-08-08 | University Of Connecticut | Compositions useful as a cannabinoid receptor probe |
| FR2735774B1 (fr) * | 1995-06-21 | 1997-09-12 | Sanofi Sa | Utilisation de composes agonistes du recepteur cb2 humain pour la preparation de medicaments immunomodulateurs, nouveaux composes agonistes du recepteur cb2 et les compositions pharmaceutiques les contenant |
| US5688825A (en) * | 1996-05-31 | 1997-11-18 | University Of Connecticut | Anandamide amidase inhibitors as analgesic agents |
| US20010009965A1 (en) * | 1998-05-04 | 2001-07-26 | Alexandros Makriyannis | Novel analgesic and immunomodulatory cannabinoids |
| ATE277921T1 (de) * | 1998-05-04 | 2004-10-15 | Univ Connecticut | Selektiv auf den cb2-rezeptor wirkende cannabinoide |
-
1999
- 1999-05-04 AT AT99921676T patent/ATE277921T1/de not_active IP Right Cessation
- 1999-05-04 CA CA002340444A patent/CA2340444A1/en not_active Abandoned
- 1999-05-04 US US09/304,718 patent/US6166066A/en not_active Expired - Fee Related
- 1999-05-04 EP EP99921676A patent/EP1076653B1/de not_active Expired - Lifetime
- 1999-05-04 WO PCT/US1999/009806 patent/WO1999057107A2/en not_active Ceased
- 1999-05-04 ES ES99921676T patent/ES2224658T3/es not_active Expired - Lifetime
- 1999-05-04 DE DE69920683T patent/DE69920683T2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| WO1999057107A3 (en) | 2000-02-03 |
| WO1999057107A2 (en) | 1999-11-11 |
| EP1076653B1 (de) | 2004-09-29 |
| ATE277921T1 (de) | 2004-10-15 |
| EP1076653A2 (de) | 2001-02-21 |
| US6166066A (en) | 2000-12-26 |
| ES2224658T3 (es) | 2005-03-01 |
| DE69920683T2 (de) | 2005-04-07 |
| CA2340444A1 (en) | 1999-11-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition | ||
| 8339 | Ceased/non-payment of the annual fee |