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DE60119949D1 - 1,2,5,10-TETRAHYDROPYRIDAZINOi4,5-BöCHINOLIN-1,10-DIONE UND IHRE ANWENDUNG IN DER BEHANDLUNG VON SCHMERZEN - Google Patents

1,2,5,10-TETRAHYDROPYRIDAZINOi4,5-BöCHINOLIN-1,10-DIONE UND IHRE ANWENDUNG IN DER BEHANDLUNG VON SCHMERZEN

Info

Publication number
DE60119949D1
DE60119949D1 DE60119949T DE60119949T DE60119949D1 DE 60119949 D1 DE60119949 D1 DE 60119949D1 DE 60119949 T DE60119949 T DE 60119949T DE 60119949 T DE60119949 T DE 60119949T DE 60119949 D1 DE60119949 D1 DE 60119949D1
Authority
DE
Germany
Prior art keywords
pain
treatment
bochinoline
dione
structural diagram
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60119949T
Other languages
English (en)
Other versions
DE60119949T2 (de
Inventor
Megan Murphy
Wenhua Xiao
Gordon Brown
Ann Urbanek
Marie Mclaren
Edward Vacek
Thomas Bare
Lynn Horchler
Christine Barlaam
Banks Steelman
Vernon Alford
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
AstraZeneca AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AstraZeneca AB filed Critical AstraZeneca AB
Application granted granted Critical
Publication of DE60119949D1 publication Critical patent/DE60119949D1/de
Publication of DE60119949T2 publication Critical patent/DE60119949T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE60119949T 2000-09-29 2001-09-28 1,2,5,10-TETRAHYDROPYRIDAZINOi4,5-BöCHINOLIN-1,10-DIONE UND IHRE ANWENDUNG IN DER BEHANDLUNG VON SCHMERZEN Expired - Lifetime DE60119949T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23662900P 2000-09-29 2000-09-29
US236629P 2000-09-29
PCT/SE2001/002123 WO2002026738A1 (en) 2000-09-29 2001-09-28 1,2,5,10-TETRAHYDROPYRIDAZINO[4,5-b]QUINOLINE-1,10-DIONES AND THEIR USE FOR THE TREATMENT OF PAIN

Publications (2)

Publication Number Publication Date
DE60119949D1 true DE60119949D1 (de) 2006-06-29
DE60119949T2 DE60119949T2 (de) 2007-04-26

Family

ID=22890304

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60119949T Expired - Lifetime DE60119949T2 (de) 2000-09-29 2001-09-28 1,2,5,10-TETRAHYDROPYRIDAZINOi4,5-BöCHINOLIN-1,10-DIONE UND IHRE ANWENDUNG IN DER BEHANDLUNG VON SCHMERZEN

Country Status (8)

Country Link
US (1) US6833368B2 (de)
EP (1) EP1325002B1 (de)
JP (1) JP2004509962A (de)
AT (1) ATE327235T1 (de)
AU (1) AU2001292498A1 (de)
DE (1) DE60119949T2 (de)
ES (1) ES2263661T3 (de)
WO (1) WO2002026738A1 (de)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9420590D0 (en) 1993-10-22 1994-11-30 Zeneca Ltd Pyridazino quinoline compounds
GB9507318D0 (en) 1995-04-07 1995-05-31 Zeneca Ltd Alpha substituted pyridazino quinoline compounds
HK1048767A1 (zh) 1999-12-23 2003-04-17 阿斯特拉曾尼卡有限公司 治疗疼痛的方法和组合物
DE60013326T2 (de) 1999-12-23 2005-09-08 Astrazeneca Ab Verbindungen und verfahren zur behandlung von schmerz
JP2003519147A (ja) 1999-12-23 2003-06-17 アストラゼネカ・アクチエボラーグ 痛みの処置のための化合物および方法
AU2420001A (en) * 1999-12-23 2001-07-09 Astrazeneca Ab Methods and compositions for the treatment of pain
AU2420101A (en) 1999-12-23 2001-07-09 Astrazeneca Ab Method and composition for the treatment of pain
JP4197216B2 (ja) 1999-12-24 2008-12-17 Jsr株式会社 液状硬化性樹脂組成物およびその硬化物

Also Published As

Publication number Publication date
ATE327235T1 (de) 2006-06-15
AU2001292498A1 (en) 2002-04-08
US6833368B2 (en) 2004-12-21
EP1325002A1 (de) 2003-07-09
WO2002026738A1 (en) 2002-04-04
US20040058927A1 (en) 2004-03-25
JP2004509962A (ja) 2004-04-02
ES2263661T3 (es) 2006-12-16
DE60119949T2 (de) 2007-04-26
EP1325002B1 (de) 2006-05-24

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition