CZ109795A3 - Antimicrobial 5-hydrazine-quionolone derivatives - Google Patents
Antimicrobial 5-hydrazine-quionolone derivativesInfo
- Publication number
- CZ109795A3 CZ109795A3 CZ951097A CZ109795A CZ109795A3 CZ 109795 A3 CZ109795 A3 CZ 109795A3 CZ 951097 A CZ951097 A CZ 951097A CZ 109795 A CZ109795 A CZ 109795A CZ 109795 A3 CZ109795 A3 CZ 109795A3
- Authority
- CZ
- Czechia
- Prior art keywords
- quionolone
- hydrazine
- antimicrobial
- derivatives
- quionolone derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Quinoline Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US96896092A | 1992-10-30 | 1992-10-30 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CZ109795A3 true CZ109795A3 (en) | 1995-12-13 |
| CZ282581B6 CZ282581B6 (en) | 1997-08-13 |
Family
ID=25514997
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CZ951097A CZ282581B6 (en) | 1992-10-30 | 1993-10-22 | 5-hydrazine-choline derivatives and pharmaceutical compositions containing thereof |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP0666853A1 (en) |
| JP (1) | JPH08502750A (en) |
| KR (1) | KR950704301A (en) |
| CN (1) | CN1064357C (en) |
| AU (1) | AU687018B2 (en) |
| BR (1) | BR9307347A (en) |
| CA (1) | CA2148003A1 (en) |
| CZ (1) | CZ282581B6 (en) |
| EG (1) | EG20543A (en) |
| FI (1) | FI952049L (en) |
| HU (1) | HUT72072A (en) |
| IL (1) | IL107323A (en) |
| MX (1) | MX9306814A (en) |
| NO (1) | NO951640L (en) |
| NZ (1) | NZ257470A (en) |
| PL (1) | PL178094B1 (en) |
| RU (1) | RU2126000C1 (en) |
| SG (1) | SG59979A1 (en) |
| SK (1) | SK54795A3 (en) |
| WO (1) | WO1994010163A1 (en) |
| ZA (1) | ZA938089B (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5646163A (en) * | 1992-10-30 | 1997-07-08 | The Procter & Gamble Company | Quinolone 5-(N-heterosubstituted amino) antimicrobials |
| EP0775114B1 (en) * | 1994-08-02 | 2000-03-22 | The Procter & Gamble Company | Process for making antimicrobial compounds |
| NZ290722A (en) * | 1994-08-02 | 1999-03-29 | Procter & Gamble | A process for making derivatives of quinolonyl lactam (qla's); intermediates |
| ES2188890T3 (en) * | 1996-02-09 | 2003-07-01 | Toyama Chemical Co Ltd | DERIVATIVES OF THE QUINOLEINCARBOXILICO ACID AND ITS SALTS. |
| RU2248199C1 (en) * | 2003-06-02 | 2005-03-20 | Открытое Акционерное Общество "Акционерное Курганское общество медицинских препаратов и изделий "Синтез" (ОАО "Синтез") | Eye drops and method for their obtaining |
| RU2265437C2 (en) * | 2003-07-02 | 2005-12-10 | Суханов Александр Владимирович | Method for treating gastric and duodenal diseases caused by helicobacter pylori |
| RU2245134C1 (en) * | 2003-09-02 | 2005-01-27 | Открытое акционерное общество "Красфарма" | Ofloxacine composition for injections |
| WO2005026147A1 (en) | 2003-09-10 | 2005-03-24 | Kyorin Pharmaceutical Co., Ltd. | 7-(4-substituted 3- cyclopropylaminomethyl-1 pyrrolidinyl) quinolonecarboxylic acid derivative |
| RS55114B1 (en) * | 2005-05-18 | 2016-12-30 | Raptor Pharmaceuticals Inc | AEROSOLIZED FLUOROCHINOLONS AND THEIR USE |
| US8524735B2 (en) | 2005-05-18 | 2013-09-03 | Mpex Pharmaceuticals, Inc. | Aerosolized fluoroquinolones and uses thereof |
| CA2528849C (en) | 2005-06-08 | 2014-01-14 | Janssen Pharmaceutica N.V. | Quinoline derivatives as antibacterial agents |
| EA010601B1 (en) * | 2005-06-09 | 2008-10-30 | Янссен Фармацевтика Н.В. | Quinoline derivatives as antibacterial agents |
| CN101020647B (en) * | 2007-02-14 | 2011-03-30 | 杭州师范学院 | A kind of synthetic method of β-cyclopropylaminoacrylic acid (ester) |
| WO2008115890A2 (en) * | 2007-03-19 | 2008-09-25 | Takeda Pharmaceutical Company Limited | Mapk/erk kinase inhibitors |
| CA2701630C (en) * | 2007-10-05 | 2016-10-25 | Cylene Pharmaceuticals, Inc. | Quinolone analogs and methods related thereto |
| CN102046603B (en) * | 2008-06-03 | 2014-08-13 | 埃科特莱茵药品有限公司 | [4-(1-Amino-ethyl)-cyclohexyl]-methyl-amine and [6-(1-amino-ethyl)-tetrahydro-pyran-3-yl]-methanol as antibacterial agents base-amine derivatives |
| PT2346509T (en) | 2008-10-07 | 2020-08-05 | Horizon Orphan Llc | Inhalation of levofloxacin for reducing lung inflammation |
| NO2344129T3 (en) | 2008-10-07 | 2018-07-21 | ||
| AR076222A1 (en) * | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | DERIVATIVES 2-HYDROXIETIL-1H-QUINOLIN-ONA AND ITS AZAISOTHERAL ANALOGS WITH ANTIBACTERIAL ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| BR112012004692B8 (en) | 2009-09-04 | 2021-05-25 | Mpex Pharmaceuticals Inc | solution comprising levofloxacin for use in a method of treating cystic fibrosis in a human. |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4668680A (en) * | 1985-12-12 | 1987-05-26 | Warner-Lambert Company | 5-amino-6,8-difluoroquinolones as antibacterial agents |
| JPH0228178A (en) * | 1988-04-23 | 1990-01-30 | Toyama Chem Co Ltd | Novel pyridonecarboxylic acid derivative and salt thereof |
| DE3906365A1 (en) * | 1988-07-15 | 1990-01-18 | Bayer Ag | 7- (1-PYRROLIDINYL) -3-CHINOLONE AND NAPHTHYRIDONE CARBOXYLIC ACID DERIVATIVES, METHOD AND SUBSTITUTED (OXA) DIAZABICYCLOOCTANES AND NONANESE AS INTERMEDIATE PRODUCTS, AND ANTIBACTERIAL AGENTS AND FOOD ADDITIVES CONTAINING THEM |
| HU219403B (en) * | 1989-08-16 | 2001-04-28 | Pfizer Inc. | Azabicyclo-substituted quinolone and naphthyridone carboxylic acids and process for producing them |
| EP0525057B1 (en) * | 1990-04-18 | 2000-06-14 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactams |
| AU658384B2 (en) * | 1990-11-30 | 1995-04-13 | Warner-Lambert Company | Individual stereoisomers of 7-{3-(1-aminoalkyl)-1-pyrrolidinyl}-quinolones and naphthyridones as antibacterial agents |
-
1993
- 1993-01-30 EG EG68693A patent/EG20543A/en active
- 1993-10-19 IL IL10732393A patent/IL107323A/en not_active IP Right Cessation
- 1993-10-22 BR BR9307347A patent/BR9307347A/en not_active Application Discontinuation
- 1993-10-22 NZ NZ257470A patent/NZ257470A/en unknown
- 1993-10-22 EP EP93924393A patent/EP0666853A1/en not_active Withdrawn
- 1993-10-22 PL PL93308671A patent/PL178094B1/en unknown
- 1993-10-22 HU HU9501237A patent/HUT72072A/en unknown
- 1993-10-22 SG SG1996007851A patent/SG59979A1/en unknown
- 1993-10-22 CA CA002148003A patent/CA2148003A1/en not_active Abandoned
- 1993-10-22 WO PCT/US1993/010091 patent/WO1994010163A1/en not_active Ceased
- 1993-10-22 KR KR1019950701690A patent/KR950704301A/en not_active Abandoned
- 1993-10-22 CZ CZ951097A patent/CZ282581B6/en not_active IP Right Cessation
- 1993-10-22 RU RU95110762A patent/RU2126000C1/en active
- 1993-10-22 JP JP6511167A patent/JPH08502750A/en active Pending
- 1993-10-22 AU AU54097/94A patent/AU687018B2/en not_active Ceased
- 1993-10-22 SK SK547-95A patent/SK54795A3/en unknown
- 1993-10-22 FI FI952049A patent/FI952049L/en unknown
- 1993-10-29 ZA ZA938089A patent/ZA938089B/en unknown
- 1993-10-29 MX MX9306814A patent/MX9306814A/en not_active IP Right Cessation
- 1993-10-30 CN CN93120224A patent/CN1064357C/en not_active Expired - Fee Related
-
1995
- 1995-04-28 NO NO951640A patent/NO951640L/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA938089B (en) | 1994-06-07 |
| SG59979A1 (en) | 1999-02-22 |
| CZ282581B6 (en) | 1997-08-13 |
| BR9307347A (en) | 1999-05-25 |
| FI952049A7 (en) | 1995-04-28 |
| NZ257470A (en) | 1997-08-22 |
| KR950704301A (en) | 1995-11-17 |
| AU5409794A (en) | 1994-05-24 |
| NO951640L (en) | 1995-06-30 |
| CN1064357C (en) | 2001-04-11 |
| MX9306814A (en) | 1994-07-29 |
| HUT72072A (en) | 1996-03-28 |
| HU9501237D0 (en) | 1995-06-28 |
| FI952049A0 (en) | 1995-04-28 |
| EG20543A (en) | 1999-07-31 |
| NO951640D0 (en) | 1995-04-28 |
| IL107323A (en) | 2000-06-01 |
| RU2126000C1 (en) | 1999-02-10 |
| PL178094B1 (en) | 2000-02-29 |
| AU687018B2 (en) | 1998-02-19 |
| IL107323A0 (en) | 1994-01-25 |
| FI952049L (en) | 1995-04-28 |
| CA2148003A1 (en) | 1994-05-11 |
| PL308671A1 (en) | 1995-08-21 |
| CN1092773A (en) | 1994-09-28 |
| WO1994010163A1 (en) | 1994-05-11 |
| SK54795A3 (en) | 1995-12-06 |
| EP0666853A1 (en) | 1995-08-16 |
| JPH08502750A (en) | 1996-03-26 |
| RU95110762A (en) | 1997-01-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| IF00 | In force as of 2000-06-30 in czech republic | ||
| MM4A | Patent lapsed due to non-payment of fee |
Effective date: 20011022 |