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CR8559A - Pirazolopirimidinas - Google Patents

Pirazolopirimidinas

Info

Publication number
CR8559A
CR8559A CR8559A CR8559A CR8559A CR 8559 A CR8559 A CR 8559A CR 8559 A CR8559 A CR 8559A CR 8559 A CR8559 A CR 8559A CR 8559 A CR8559 A CR 8559A
Authority
CR
Costa Rica
Prior art keywords
pirazolopirimidinas
pyrazolopyrimidines
substances
formula
manufacturing process
Prior art date
Application number
CR8559A
Other languages
English (en)
Inventor
Gebauer Olaf
Gayer Herbert
Heinemann Ulrich
Herrmann Stefan
Elbe Hans-Ludwig
Ebbert Ronald
Wachendorf-Neumann Ulrike
Dahmen Peter
Kuck Karl-Heinz
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of CR8559A publication Critical patent/CR8559A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

El invento se refiere a los Pirazolopirimidinas de la formula (I), donde R1,R2,R3, R4,R5 y X tienen los significados indicados en la descripcion; a un procedimiento de fabricacion de estas sustancias y su uso para combatir los microorganismos no deseados.
CR8559A 2004-02-20 2006-08-14 Pirazolopirimidinas CR8559A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004008807A DE102004008807A1 (de) 2004-02-20 2004-02-20 Pyrazolopyrimidine

Publications (1)

Publication Number Publication Date
CR8559A true CR8559A (es) 2006-11-23

Family

ID=34832976

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8559A CR8559A (es) 2004-02-20 2006-08-14 Pirazolopirimidinas

Country Status (15)

Country Link
US (1) US7629294B2 (es)
EP (1) EP1718652A2 (es)
JP (1) JP2007524691A (es)
KR (1) KR20070015386A (es)
CN (1) CN1946293A (es)
AR (1) AR048857A1 (es)
BR (1) BRPI0507894A (es)
CA (1) CA2556798A1 (es)
CR (1) CR8559A (es)
DE (1) DE102004008807A1 (es)
EA (1) EA200601515A1 (es)
IL (1) IL177510A0 (es)
MX (1) MXPA06009311A (es)
TW (1) TW200538044A (es)
WO (1) WO2005082907A2 (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY143499A (en) * 2003-12-22 2011-05-31 Sb Pharmco Inc Crf receptor antagonist and methods relating thereto
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
EP1945220A1 (en) 2005-10-21 2008-07-23 Mitsubishi Tanabe Pharma Corporation Pyrazolo[1,5-a]pyrimidine compounds as cannabinoid receptor antagonists
JP4847275B2 (ja) * 2005-10-21 2011-12-28 田辺三菱製薬株式会社 ピラゾロ[1,5−a]ピリミジン化合物
AR061793A1 (es) 2006-07-05 2008-09-24 Mitsubishi Tanabe Pharma Corp Compuesto de pirazolo[1,5-a] pirimidina y composicion farmaceutica
TW201345908A (zh) * 2006-07-05 2013-11-16 Mitsubishi Tanabe Pharma Corp 吡唑并〔1,5-a〕嘧啶化合物
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
JP4837701B2 (ja) * 2007-04-20 2011-12-14 田辺三菱製薬株式会社 医薬組成物
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
US8507673B2 (en) * 2008-12-11 2013-08-13 Emory University Process for preparing 5,7 diaminopyrazolo [1,5-A] pyrimidine compounds
HRP20202008T1 (hr) 2013-03-14 2021-02-19 Epizyme, Inc. Inhibitori arginin-metiltransferaze i njihove uporabe
US9365527B2 (en) 2013-03-14 2016-06-14 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
CA2903264A1 (en) 2013-03-14 2014-11-06 Epizyme, Inc. Pyrazole derivatives as arginine methyltransferase inhibitors and uses thereof
WO2014153214A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyl transferase inhibtors and uses thereof
US9447079B2 (en) 2013-03-14 2016-09-20 Epizyme, Inc. PRMT1 inhibitors and uses thereof
US9120757B2 (en) 2013-03-14 2015-09-01 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
WO2014153235A2 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
WO2014153090A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Pyrazole derivatives asprmt1 inhibitors and uses thereof
EP2970181B1 (en) 2013-03-14 2017-06-07 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
US9023883B2 (en) 2013-03-14 2015-05-05 Epizyme, Inc. PRMT1 inhibitors and uses thereof
US11046698B2 (en) * 2017-07-28 2021-06-29 Nimbus Lakshmi, Inc. TYK2 inhibitors and uses thereof
US11414431B2 (en) * 2018-10-15 2022-08-16 Nimbus Lakshmi, Inc. Substituted pyrazolo[1,5-a]pyrimidines as TYK2 inhibitors

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS423174Y1 (es) * 1964-01-17 1967-02-24
JPS423173Y1 (es) * 1964-01-24 1967-02-24
US3515715A (en) * 1967-01-23 1970-06-02 Eastman Kodak Co Quaternized pyrazolylazo dyes
US3634391A (en) * 1969-07-25 1972-01-11 Eastman Kodak Co Pyrazolyl-azo-indole dyestuffs
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
FR2537137B1 (fr) 1982-12-03 1985-07-19 Roussel Uclaf Procede de preparation de derives de l'acide 2-thiophene acetique et produits intermediaires necessaires pour leur preparation
DE3338292A1 (de) 1983-10-21 1985-05-02 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)-pyrimidine und diese enthaltende fungizide
DE3533050A1 (de) * 1985-09-17 1987-03-26 Basf Ag 7-amino-azolo(1,5-a)pyrimidine, verfahren zu ihrer herstellung und diese enthaltende fungizide, bzw. deren verwendung als fungizide
GB9510459D0 (en) * 1995-05-24 1995-07-19 Zeneca Ltd Bicyclic amines
FR2750048B1 (fr) * 1996-06-21 1998-08-14 Oreal Compositions de teinture des fibres keratiniques contenant des derives pyrazolo-(1, 5-a)-pyrimidine, procede de teinture, nouveaux derives pyrazolo-(1, 5-a)-pyrimidine et leur procede de preparation
GB9624611D0 (en) * 1996-11-26 1997-01-15 Zeneca Ltd Bicyclic amine compounds
WO1998025924A1 (en) 1996-11-26 1998-06-18 Zeneca Limited 8-azabicyclo[3.2.1]octane-, 8-azabicyclo[3.2.1]oct-6-ene-, 9-azabicyclo[3.3.1]nonane-, 9-aza-3-oxabicyclo[3.3.1]nonane- and 9-aza-3-thiabicyclo[3.3.1]nonane derivatives, their preparation and their use as insecticides
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6552026B2 (en) * 1999-06-14 2003-04-22 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
JP2001019693A (ja) * 1999-06-14 2001-01-23 American Cyanamid Co 殺菌・殺カビ性6−フェニル−ピラゾロピリミジン
JP2004515551A (ja) * 2000-12-11 2004-05-27 ビーエーエスエフ アクチェンゲゼルシャフト 6−フェニル−ピラゾロピリミジン
ATE357142T1 (de) 2001-07-26 2007-04-15 Basf Ag 7-aminotriazolopyrimidine zur bekämpfung von schadpilzen
DE10223917A1 (de) * 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine
MXPA05008955A (es) * 2003-02-28 2006-02-22 Teijin Pharma Ltd Derivados de pirazolo [1,5-a] pirimidina.
EA200501888A1 (ru) 2003-06-03 2006-06-30 Басф Акциенгезельшафт Замещённые пиразолопиримидины, способ их получения и их применение для борьбы с патогенными грибами, а также содержащие их средства
US20070037828A1 (en) * 2003-06-27 2007-02-15 Olaf Gebauer Pyrazolopyrimidines

Also Published As

Publication number Publication date
CN1946293A (zh) 2007-04-11
JP2007524691A (ja) 2007-08-30
CA2556798A1 (en) 2005-09-09
EA200601515A1 (ru) 2006-12-29
WO2005082907A3 (de) 2006-06-29
AR048857A1 (es) 2006-06-07
BRPI0507894A (pt) 2007-07-24
WO2005082907A2 (de) 2005-09-09
TW200538044A (en) 2005-12-01
US7629294B2 (en) 2009-12-08
DE102004008807A1 (de) 2005-09-08
KR20070015386A (ko) 2007-02-02
US20050187224A1 (en) 2005-08-25
EP1718652A2 (de) 2006-11-08
IL177510A0 (en) 2006-12-10
MXPA06009311A (es) 2007-03-01

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)