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CO6361912A2 - Compuestos que modulan selectivamenta el receptor cb2 - Google Patents

Compuestos que modulan selectivamenta el receptor cb2

Info

Publication number
CO6361912A2
CO6361912A2 CO11033548A CO11033548A CO6361912A2 CO 6361912 A2 CO6361912 A2 CO 6361912A2 CO 11033548 A CO11033548 A CO 11033548A CO 11033548 A CO11033548 A CO 11033548A CO 6361912 A2 CO6361912 A2 CO 6361912A2
Authority
CO
Colombia
Prior art keywords
compounds
receiver
agonists
modulate
selectively
Prior art date
Application number
CO11033548A
Other languages
English (en)
Inventor
Alessandra Bartolozzi
Angela Berry
Eugene Richard Hickey
Markus Ostermeier
Doris Riether
Achim Sauer
David S Thomson
Lifen Wu
Renee Zindell
Patricia Amouzegh
Nigel Blumire
Stephen Peter East
Monika Ermann
Someina Khor
Innocent Mushi
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of CO6361912A2 publication Critical patent/CO6361912A2/es

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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
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Abstract

Se describen compuestos de fórmula (I)Los compuestos de acuerdo con la invención se unen a y son agonistas, antagonistas o agonistas inversos del receptor CB2, y son útiles para tratar la inflamación. Los compuestos que son agonistas son útiles adicionalmente para tratar el dolor.
CO11033548A 2008-09-25 2011-03-17 Compuestos que modulan selectivamenta el receptor cb2 CO6361912A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10007708P 2008-09-25 2008-09-25

Publications (1)

Publication Number Publication Date
CO6361912A2 true CO6361912A2 (es) 2012-01-20

Family

ID=41698020

Family Applications (1)

Application Number Title Priority Date Filing Date
CO11033548A CO6361912A2 (es) 2008-09-25 2011-03-17 Compuestos que modulan selectivamenta el receptor cb2

Country Status (24)

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US (4) US8372874B2 (es)
EP (2) EP2342199B1 (es)
JP (2) JP4928650B2 (es)
KR (2) KR20110063485A (es)
CN (2) CN102164916A (es)
AP (1) AP2011005674A0 (es)
AR (2) AR073688A1 (es)
AU (2) AU2009296838A1 (es)
BR (2) BRPI0919172A2 (es)
CA (2) CA2737639A1 (es)
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US8048899B2 (en) 2011-11-01
US8372874B2 (en) 2013-02-12
AU2009296838A1 (en) 2010-04-01
EP2342200A2 (en) 2011-07-13
EP2342199A2 (en) 2011-07-13
CA2737645A1 (en) 2010-04-01
US20100076029A1 (en) 2010-03-25
UY32139A (es) 2010-04-30
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EP2342199B1 (en) 2014-02-26
WO2010036630A3 (en) 2010-05-20

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