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CN113166135A - 苯并噻吩类衍生物调节剂、其制备方法和应用 - Google Patents

苯并噻吩类衍生物调节剂、其制备方法和应用 Download PDF

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Publication number
CN113166135A
CN113166135A CN202080006349.XA CN202080006349A CN113166135A CN 113166135 A CN113166135 A CN 113166135A CN 202080006349 A CN202080006349 A CN 202080006349A CN 113166135 A CN113166135 A CN 113166135A
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cycloalkyl
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haloalkyl
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CN113166135B (zh
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苏熠东
李松
陈晓坡
汪军
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Jiangsu Hansoh Pharmaceutical Group Co Ltd
Shanghai Hansoh Biomedical Co Ltd
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Jiangsu Hansoh Pharmaceutical Group Co Ltd
Shanghai Hansoh Biomedical Co Ltd
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Abstract

一种含氮环类衍生物调节剂、其制备方法和应用。特别地，涉及通式(I)所示的化合物、其制备方法及含有该化合物的药物组合物，及其作为G蛋白耦联受体调节剂在治疗或预防中枢神经系统疾病和/或精神疾病的用途。

Description

PCT国内申请，说明书已公开。

Claims (16)

  1. PCT国内申请，权利要求书已公开。
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WO2024072930A1 (en) * 2022-09-30 2024-04-04 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Dopamine d3/d2 receptor partial agonists for the treatment of neuropsychiatric disorders
WO2024075813A1 (ja) * 2022-10-07 2024-04-11 学校法人中部大学 ジケトピペラジン化合物を用いるポリペプチド合成
KR20240112213A (ko) * 2023-01-11 2024-07-18 리히터 게데온 닐트. 도파민 d3/d2 수용체 조절 화합물
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CN102159557A (zh) * 2008-09-22 2011-08-17 弗·哈夫曼-拉罗切有限公司 哌嗪d3和5-ht2a受体调节剂
WO2017045599A1 (zh) * 2015-09-15 2017-03-23 浙江京新药业股份有限公司 环己烷衍生物或其立体异构体或盐及其制备与应用

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