CA2860038A1 - Compositions a liberation prolongee - Google Patents

Compositions a liberation prolongee Download PDF

Info

Publication number: CA2860038A1
Authority: CA; Canada
Prior art keywords: desvenlafaxine; oxalate; composition; rate controlling; pharmaceutical composition
Prior art date: 2014-08-18
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA2860038A

Other languages

English (en)

Inventor

Subrata Kundu

Atul Patil

Nitin Borkar

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

GENERIC PARTNERS PTY Ltd

Original Assignee

GENERIC PARTNERS PTY Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2014-08-18

Filing date

2014-08-18

Publication date

2016-02-18

2014-08-18 Application filed by GENERIC PARTNERS PTY Ltd filed Critical GENERIC PARTNERS PTY Ltd

2014-08-18 Priority to CA2860038A priority Critical patent/CA2860038A1/fr

2016-02-18 Publication of CA2860038A1 publication Critical patent/CA2860038A1/fr

Status Abandoned legal-status Critical Current

Links

239000000203 mixture Substances 0.000 title claims description 45
238000013265 extended release Methods 0.000 title description 4
KYYIDSXMWOZKMP-UHFFFAOYSA-N O-desmethylvenlafaxine Chemical compound C1CCCCC1(O)C(CN(C)C)C1=CC=C(O)C=C1 KYYIDSXMWOZKMP-UHFFFAOYSA-N 0.000 claims abstract description 65
229960001623 desvenlafaxine Drugs 0.000 claims abstract description 56
MUBZPKHOEPUJKR-UHFFFAOYSA-N Oxalic acid Chemical compound OC(=O)C(O)=O MUBZPKHOEPUJKR-UHFFFAOYSA-N 0.000 claims abstract description 40
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AXZKOIWUVFPNLO-UHFFFAOYSA-N magnesium;oxygen(2-) Chemical compound [O-2].[Mg+2] AXZKOIWUVFPNLO-UHFFFAOYSA-N 0.000 description 2
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PNVNVHUZROJLTJ-UHFFFAOYSA-N venlafaxine Chemical compound C1=CC(OC)=CC=C1C(CN(C)C)C1(O)CCCCC1 PNVNVHUZROJLTJ-UHFFFAOYSA-N 0.000 description 2
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230000013275 serotonin uptake Effects 0.000 description 1
238000004513 sizing Methods 0.000 description 1
239000011734 sodium Substances 0.000 description 1
239000007787 solid Substances 0.000 description 1
239000002195 soluble material Substances 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
238000005563 spheronization Methods 0.000 description 1
239000008117 stearic acid Substances 0.000 description 1
150000003890 succinate salts Chemical class 0.000 description 1
208000024891 symptom Diseases 0.000 description 1
235000002906 tartaric acid Nutrition 0.000 description 1
239000011975 tartaric acid Substances 0.000 description 1
238000012360 testing method Methods 0.000 description 1
MHXBHWLGRWOABW-UHFFFAOYSA-N tetradecyl octadecanoate Chemical compound CCCCCCCCCCCCCCCCCC(=O)OCCCCCCCCCCCCCC MHXBHWLGRWOABW-UHFFFAOYSA-N 0.000 description 1
239000001069 triethyl citrate Substances 0.000 description 1
235000013769 triethyl citrate Nutrition 0.000 description 1
VMYFZRTXGLUXMZ-UHFFFAOYSA-N triethyl citrate Natural products CCOC(=O)C(O)(C(=O)OCC)C(=O)OCC VMYFZRTXGLUXMZ-UHFFFAOYSA-N 0.000 description 1
229960001947 tripalmitin Drugs 0.000 description 1
230000001457 vasomotor Effects 0.000 description 1
XLYOFNOQVPJJNP-UHFFFAOYSA-N water Chemical compound O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 description 1
230000004584 weight gain Effects 0.000 description 1
235000019786 weight gain Nutrition 0.000 description 1
238000005550 wet granulation Methods 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Emergency Medicine (AREA)
Medicinal Preparation (AREA)

CA2860038A 2014-08-18 2014-08-18 Compositions a liberation prolongee Abandoned CA2860038A1 (fr)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
CA2860038A CA2860038A1 (fr)	2014-08-18	2014-08-18	Compositions a liberation prolongee

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
CA2860038A CA2860038A1 (fr)	2014-08-18	2014-08-18	Compositions a liberation prolongee

Publications (1)

Publication Number	Publication Date
CA2860038A1 true CA2860038A1 (fr)	2016-02-18

Family

ID=55346398

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA2860038A Abandoned CA2860038A1 (fr)	2014-08-18	2014-08-18	Compositions a liberation prolongee

Country Status (1)

Country	Link
CA (1)	CA2860038A1 (fr)

2014
- 2014-08-18 CA CA2860038A patent/CA2860038A1/fr not_active Abandoned

Publication	Publication Date	Title
EP2286801A2 (fr)	2011-02-23	Formulation de comprimé à libération prolongée contenant du pramipexole ou l'un de ses sels pharmaceutiquement acceptable, son procédé de fabrication et utilisation associée
US20060051419A1 (en)	2006-03-09	Extended release pellet formulation containing pramipexole or a pharmaceutically acceptable salt thereof
CA2905011C (fr)	2019-08-27	Capsule de topiramate a liberation lente
JP7117975B2 (ja)	2022-08-15	テネリグリプチン含有医薬組成物、テネリグリプチン含有医薬組成物の製造方法、テネリグリプチン含有錠剤及びテネリグリプチン含有錠剤の製造方法
WO2008064202A2 (fr)	2008-05-29	Formulations à libération modifiée de composés actifs vis-à-vis du récepteur de calcium
JP5948648B2 (ja)	2016-07-06	安定化されたエペリゾンを含有する徐放性製剤
US20070009589A1 (en)	2007-01-11	Extended release compositions
WO2022144919A1 (fr)	2022-07-07	Compositions pharmaceutiques à libération prolongée de riociguat
WO2011037976A2 (fr)	2011-03-31	Formulations pharmaceutiques de pramipexole
WO2009057138A2 (fr)	2009-05-07	Compositions pharmaceutiques à libération régulée de toltérodine
EP2603207A2 (fr)	2013-06-19	Compositions orales de blonanserin a liberation controlee
US10172878B2 (en)	2019-01-08	Extended-release topiramate capsules
JP5973347B2 (ja)	2016-08-23	口腔内崩壊錠
JP2012515757A (ja)	2012-07-12	トリメタジジンの放出調節固形薬剤組成物及びその製造方法
SI22849A (sl)	2010-02-26	Ropinirolni pripravek
AU2009243734B2 (en)	2014-02-27	Granulate comprising escitalopram oxalate
MX2013010598A (es)	2014-01-08	Composiciones farmaceuticas de liberacion controlada de inhibidor de recaptacion de serotonina selectivo.
CN114053237A (zh)	2022-02-18	一种控释片剂及其制备方法
TWI823471B (zh)	2023-11-21	沙庫巴曲纈沙坦鈉緩釋組合物、其製備方法及應用
WO2020003196A1 (fr)	2020-01-02	Composition pharmaceutique d'axitinib
CA2860038A1 (fr)	2016-02-18	Compositions a liberation prolongee
WO2010089775A2 (fr)	2010-08-12	Forme galénique améliorée de médicament destiné à administrer de manière contrôlée un ou plusieurs agents pharmaceutiquement actifs
US20150050337A1 (en)	2015-02-19	Extended Release Compositions
AU2013200554A1 (en)	2013-08-22	Extended release compositions
EA033685B1 (ru)	2019-11-15	Фармацевтические лекарственные формы

Legal Events

Date	Code	Title	Description
2017-09-30	FZDE	Dead	Effective date: 20170818