CA2578990A1 - Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine - Google Patents

Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine Download PDF

Info

Publication number: CA2578990A1
Authority: CA; Canada
Prior art keywords: pain; combination; alpha; pharmaceutically acceptable; agonist
Prior art date: 2004-09-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002578990A

Other languages

English (en)

Inventor

Jayasena Hettiarachchi

Iradj Haji Mohamad Reza

Carolyn Rose Sikes

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Corp SRL

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-09-07

Filing date

2005-08-27

Publication date

2006-03-16

2004-09-07 Priority claimed from GBGB0419849.5A external-priority patent/GB0419849D0/en

2005-08-27 Application filed by Individual filed Critical Individual

2006-03-16 Publication of CA2578990A1 publication Critical patent/CA2578990A1/fr

Status Abandoned legal-status Critical Current

Links

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210000000836 trigeminal nuclei Anatomy 0.000 description 1
LENZDBCJOHFCAS-UHFFFAOYSA-N tris Chemical compound OCC(N)(CO)CO LENZDBCJOHFCAS-UHFFFAOYSA-N 0.000 description 1
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239000003071 vasodilator agent Substances 0.000 description 1
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MWLSOWXNZPKENC-SSDOTTSWSA-N zileuton Chemical compound C1=CC=C2SC([C@H](N(O)C(N)=O)C)=CC2=C1 MWLSOWXNZPKENC-SSDOTTSWSA-N 0.000 description 1
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HDOZVRUNCMBHFH-UHFFFAOYSA-N zotepine Chemical compound CN(C)CCOC1=CC2=CC=CC=C2SC2=CC=C(Cl)C=C12 HDOZVRUNCMBHFH-UHFFFAOYSA-N 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents

Landscapes

Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
Neurosurgery (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

CA002578990A 2004-09-07 2005-08-27 Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine Abandoned CA2578990A1 (fr)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
GBGB0419849.5A GB0419849D0 (en)	2004-09-07	2004-09-07	Pharmaceutical combination
GB0419849.5		2004-09-07
US61460704P	2004-09-29	2004-09-29
US60/614,607		2004-09-29
PCT/IB2005/002684 WO2006027681A1 (fr)	2004-09-07	2005-08-27	Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine

Publications (1)

Publication Number	Publication Date
CA2578990A1 true CA2578990A1 (fr)	2006-03-16

Family

ID=35116045

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002578990A Abandoned CA2578990A1 (fr)	2004-09-07	2005-08-27	Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine

Country Status (6)

Country	Link
EP (1)	EP1791599A1 (fr)
JP (1)	JP2008512436A (fr)
BR (1)	BRPI0514983A (fr)
CA (1)	CA2578990A1 (fr)
MX (1)	MX2007002790A (fr)
WO (1)	WO2006027681A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2010046399A1 (fr) *	2008-10-22	2010-04-29	Novartis Ag	Combinaisons pour le traitement de la migraine
EP2627328B1 (fr)	2010-10-15	2016-09-14	Contera Pharma APS	Combinaisons d'agonistes de récepteurs de sérotonine pour le traitement de troubles du mouvement
HUE037732T2 (hu) *	2012-04-18	2018-09-28	Contera Pharma Aps	A mozgászavarok fejlett kezelésére alkalmas, szájon át szedhetõ gyógyszerészeti készítmény
EP3481385B1 (fr)	2016-07-11	2025-09-03	Contera Pharma A/S	Système d'administration de médicament pulsatile pour le traitement de l'akinésie matinale
CA3157466A1 (fr) *	2020-01-22	2021-07-29	Diana Sofia CHAPELA DUARTE PIRES	Bromhydrate d'eletriptan destine au traitement d'une lesion medullaire et a l'amelioration de la fonction locomotrice

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NZ508491A (en) *	1998-07-09	2003-09-26	Warner Lambert Co	Compositions comprising GABA analogs and a decongestant to relieve sinus headache pain
TWI312285B (en) *	2001-10-25	2009-07-21	Depomed Inc	Methods of treatment using a gastric retained gabapentin dosage
GB0219024D0 (en) *	2002-08-15	2002-09-25	Pfizer Ltd	Synergistic combinations

2005
- 2005-08-27 CA CA002578990A patent/CA2578990A1/fr not_active Abandoned
- 2005-08-27 BR BRPI0514983-5A patent/BRPI0514983A/pt not_active IP Right Cessation
- 2005-08-27 JP JP2007530789A patent/JP2008512436A/ja not_active Withdrawn
- 2005-08-27 MX MX2007002790A patent/MX2007002790A/es unknown
- 2005-08-27 EP EP05775629A patent/EP1791599A1/fr not_active Withdrawn
- 2005-08-27 WO PCT/IB2005/002684 patent/WO2006027681A1/fr not_active Ceased

Also Published As

Publication number	Publication date
JP2008512436A (ja)	2008-04-24
EP1791599A1 (fr)	2007-06-06
BRPI0514983A (pt)	2008-07-01
MX2007002790A (es)	2007-04-23
WO2006027681A1 (fr)	2006-03-16

Publication	Publication Date	Title
US20070191462A1 (en)	2007-08-16	Combination of A 5-HT(1) Receptor Agonist and an Alpha-2-Delta Ligand for the Treatment of Migraine
CA2850925C (fr)	2017-01-10	Derives de (4-phenylimidazol-2-yl) ethylamine utiles comme modulateurs de canal de sodium
CA2600510C (fr)	2010-11-02	Formes cristallines d'un derive d'imidazole
WO2007129188A1 (fr)	2007-11-15	Composé de cyclopropanecarboxamide
WO2012120398A1 (fr)	2012-09-13	Dérivés de carboxamide substitués par aryle en tant que modulateurs de trpm8
CA2578990A1 (fr)	2006-03-16	Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine
US20090227680A1 (en)	2009-09-10	Amino Acid Derivatives
WO2011077313A1 (fr)	2011-06-30	Pipéridinecarboxamides en tant qu'inhibiteurs de mpges - 1
WO2006056874A1 (fr)	2006-06-01	Forme saline
WO2013093688A1 (fr)	2013-06-27	Dérivés sulfonamides et leur utilisation en tant qu'inhibiteurs de vgsc
US20080293746A1 (en)	2008-11-27	Combinations comprising pregabalin
WO2025155874A1 (fr)	2025-07-24	Méthodes et composés pour moduler une réponse immunitaire
WO2024239001A2 (fr)	2024-11-21	Analogues d'isoandrographolide et méthode de traitement les utilisant
US20090286875A1 (en)	2009-11-19	Isocystene derivatives for the treatment of pain
WO2007052134A1 (fr)	2007-05-10	Acide (2s)-2-aminomethyl-5-ethyl heptanoique et son utilisation pharmaceutique
HK1108831A (en)	2008-05-23	Combination of a selective noradrenaline reuptake inhibitor and a pdev inhibitor
OA18626A (en)	2019-01-31	Sulfonamides as modulators of sodium channels.
HK1116348A (en)	2008-12-19	Crystal forms of an imidazole derivative

Legal Events

Date	Code	Title	Description
2007-03-02	EEER	Examination request
2010-08-27	FZDE	Dead