MX2007002790A - Combinacion de un agonista del receptor 5-hidroxitriptamina (i) y un ligando alfa-2-delta para el tratamiento de migrana. - Google Patents

Combinacion de un agonista del receptor 5-hidroxitriptamina (i) y un ligando alfa-2-delta para el tratamiento de migrana.

Info

Publication number: MX2007002790A
Authority: MX; Mexico
Prior art keywords: pain; alpha; acid; combination; agonist
Prior art date: 2004-09-07

Application number

MX2007002790A

Other languages

English (en)

Spanish (es)

Inventor

Jayasena Hettiarachchi

Iradj Haji Mohamad Reza

Carolyn Rose Sikes

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-09-07

Filing date

2005-08-27

Publication date

2007-04-23

2004-09-07 Priority claimed from GBGB0419849.5A external-priority patent/GB0419849D0/en

2005-08-27 Application filed by Pfizer filed Critical Pfizer

2007-04-23 Publication of MX2007002790A publication Critical patent/MX2007002790A/es

Links

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LENZDBCJOHFCAS-UHFFFAOYSA-N tris Chemical compound OCC(N)(CO)CO LENZDBCJOHFCAS-UHFFFAOYSA-N 0.000 description 1
229910052722 tritium Inorganic materials 0.000 description 1
229960000281 trometamol Drugs 0.000 description 1
208000009852 uremia Diseases 0.000 description 1
230000002485 urinary effect Effects 0.000 description 1
238000001291 vacuum drying Methods 0.000 description 1
229960002004 valdecoxib Drugs 0.000 description 1
LNPDTQAFDNKSHK-UHFFFAOYSA-N valdecoxib Chemical compound CC=1ON=C(C=2C=CC=CC=2)C=1C1=CC=C(S(N)(=O)=O)C=C1 LNPDTQAFDNKSHK-UHFFFAOYSA-N 0.000 description 1
BDIAUFOIMFAIPU-UHFFFAOYSA-N valepotriate Natural products CC(C)CC(=O)OC1C=C(C(=COC2OC(=O)CC(C)C)COC(C)=O)C2C11CO1 BDIAUFOIMFAIPU-UHFFFAOYSA-N 0.000 description 1
229940102566 valproate Drugs 0.000 description 1
229960002381 vardenafil Drugs 0.000 description 1
229940124549 vasodilator Drugs 0.000 description 1
239000003071 vasodilator agent Substances 0.000 description 1
229960004688 venlafaxine Drugs 0.000 description 1
229960001255 viloxazine Drugs 0.000 description 1
230000009278 visceral effect Effects 0.000 description 1
208000030401 vitamin deficiency disease Diseases 0.000 description 1
230000004580 weight loss Effects 0.000 description 1
239000013585 weight reducing agent Substances 0.000 description 1
239000003871 white petrolatum Substances 0.000 description 1
MWLSOWXNZPKENC-SSDOTTSWSA-N zileuton Chemical compound C1=CC=C2SC([C@H](N(O)C(N)=O)C)=CC2=C1 MWLSOWXNZPKENC-SSDOTTSWSA-N 0.000 description 1
229960005332 zileuton Drugs 0.000 description 1
150000003751 zinc Chemical class 0.000 description 1
XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical compound [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
229960000607 ziprasidone Drugs 0.000 description 1
MVWVFYHBGMAFLY-UHFFFAOYSA-N ziprasidone Chemical compound C1=CC=C2C(N3CCN(CC3)CCC3=CC=4CC(=O)NC=4C=C3Cl)=NSC2=C1 MVWVFYHBGMAFLY-UHFFFAOYSA-N 0.000 description 1
229960003414 zomepirac Drugs 0.000 description 1
ZXVNMYWKKDOREA-UHFFFAOYSA-N zomepirac Chemical compound C1=C(CC(O)=O)N(C)C(C(=O)C=2C=CC(Cl)=CC=2)=C1C ZXVNMYWKKDOREA-UHFFFAOYSA-N 0.000 description 1
229960004496 zotepine Drugs 0.000 description 1
HDOZVRUNCMBHFH-UHFFFAOYSA-N zotepine Chemical compound CN(C)CCOC1=CC2=CC=CC=C2SC2=CC=C(Cl)C=C12 HDOZVRUNCMBHFH-UHFFFAOYSA-N 0.000 description 1
210000002517 zygapophyseal joint Anatomy 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents

Landscapes

Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

MX2007002790A 2004-09-07 2005-08-27 Combinacion de un agonista del receptor 5-hidroxitriptamina (i) y un ligando alfa-2-delta para el tratamiento de migrana. MX2007002790A (es)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB0419849.5A GB0419849D0 (en)	2004-09-07	2004-09-07	Pharmaceutical combination
US61460704P	2004-09-29	2004-09-29
PCT/IB2005/002684 WO2006027681A1 (fr)	2004-09-07	2005-08-27	Combinaison d'un agoniste du recepteur 5-ht(1) et d'un ligand alpha-2-delta pour traiter la migraine

Publications (1)

Publication Number	Publication Date
MX2007002790A true MX2007002790A (es)	2007-04-23

Family

ID=35116045

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MX2007002790A MX2007002790A (es)	2004-09-07	2005-08-27	Combinacion de un agonista del receptor 5-hidroxitriptamina (i) y un ligando alfa-2-delta para el tratamiento de migrana.

Country Status (6)

Country	Link
EP (1)	EP1791599A1 (fr)
JP (1)	JP2008512436A (fr)
BR (1)	BRPI0514983A (fr)
CA (1)	CA2578990A1 (fr)
MX (1)	MX2007002790A (fr)
WO (1)	WO2006027681A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2010046399A1 (fr) *	2008-10-22	2010-04-29	Novartis Ag	Combinaisons pour le traitement de la migraine
SI2627328T1 (sl) *	2010-10-15	2017-01-31	Contera Pharma Aps	Kombinacije agonistov receptorjev serotonina za zdravljenje motenj premikanja
RU2670272C2 (ru)	2012-04-18	2018-10-22	Контера Фарма Апс	Пероральная фармацевтическая композиция, подходящая для повышения эффективности лечения двигательных нарушений
US11975104B2 (en)	2016-07-11	2024-05-07	Contera Pharma A/S	Pulsatile drug delivery system for treating morning akinesia
EP4093395B1 (fr) *	2020-01-22	2023-10-25	Technophage, Investigação e Desenvolvimento em Biotecnologia, SA	Bromhydrate d'élétriptan destiné au traitement d'une lésion médullaire et à l'amélioration de la fonction locomotrice

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BR9911943A (pt) *	1998-07-09	2001-05-29	Warner Lambert Co	Composições compreendendo análogos gaba e um descongestionante para aliviar dor de cabeça de sino
TWI312285B (en) *	2001-10-25	2009-07-21	Depomed Inc	Methods of treatment using a gastric retained gabapentin dosage
GB0219024D0 (en) *	2002-08-15	2002-09-25	Pfizer Ltd	Synergistic combinations

2005
- 2005-08-27 BR BRPI0514983-5A patent/BRPI0514983A/pt not_active IP Right Cessation
- 2005-08-27 MX MX2007002790A patent/MX2007002790A/es unknown
- 2005-08-27 EP EP05775629A patent/EP1791599A1/fr not_active Withdrawn
- 2005-08-27 JP JP2007530789A patent/JP2008512436A/ja not_active Withdrawn
- 2005-08-27 CA CA002578990A patent/CA2578990A1/fr not_active Abandoned
- 2005-08-27 WO PCT/IB2005/002684 patent/WO2006027681A1/fr not_active Ceased

Also Published As

Publication number	Publication date
WO2006027681A1 (fr)	2006-03-16
EP1791599A1 (fr)	2007-06-06
JP2008512436A (ja)	2008-04-24
CA2578990A1 (fr)	2006-03-16
BRPI0514983A (pt)	2008-07-01

Publication	Publication Date	Title
US20070191462A1 (en)	2007-08-16	Combination of A 5-HT(1) Receptor Agonist and an Alpha-2-Delta Ligand for the Treatment of Migraine
CN103906746B (zh)	2015-12-09	用作钠通道调节剂的(4-苯基咪唑-2-基)乙胺衍生物
JP5069415B2 (ja)	2012-11-07	結晶形態のイミダゾール誘導体
JP2015509110A (ja)	2015-03-26	ナトリウムチャネルモジュレーターとしてのベンゾイミダゾールおよびイミダゾピリジン誘導体
BRPI0618129A2 (pt)	2011-08-16	derivados de pirazina como moduladores de canal de sódio para o tratamento de dor
MX2007000694A (es)	2007-03-12	Combinacion de un inhibidor selectivo de reabsorcion de noradrenalina y un inhibidor.
MX2007002790A (es)	2007-04-23	Combinacion de un agonista del receptor 5-hidroxitriptamina (i) y un ligando alfa-2-delta para el tratamiento de migrana.
JP5903681B2 (ja)	2016-04-13	多形形態
WO2006056874A1 (fr)	2006-06-01	Forme saline
US20090227680A1 (en)	2009-09-10	Amino Acid Derivatives
US20080293746A1 (en)	2008-11-27	Combinations comprising pregabalin
WO2025155874A1 (fr)	2025-07-24	Méthodes et composés pour moduler une réponse immunitaire
WO2024239001A2 (fr)	2024-11-21	Analogues d'isoandrographolide et méthode de traitement les utilisant
AU2024271399A1 (en)	2025-12-18	Isoandrographolide analogs and method for treatment using the same
JP2009516675A (ja)	2009-04-23	疼痛を治療するためのイソシステイン誘導体
HK1108831A (en)	2008-05-23	Combination of a selective noradrenaline reuptake inhibitor and a pdev inhibitor
HK1116348A (en)	2008-12-19	Crystal forms of an imidazole derivative
WO2007052134A1 (fr)	2007-05-10	Acide (2s)-2-aminomethyl-5-ethyl heptanoique et son utilisation pharmaceutique
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OA18626A (en)	2019-01-31	Sulfonamides as modulators of sodium channels.