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BRPI0509876A - métodos para controlar a angiogênese e a proliferação de células - Google Patents

métodos para controlar a angiogênese e a proliferação de células

Info

Publication number
BRPI0509876A
BRPI0509876A BRPI0509876-9A BRPI0509876A BRPI0509876A BR PI0509876 A BRPI0509876 A BR PI0509876A BR PI0509876 A BRPI0509876 A BR PI0509876A BR PI0509876 A BRPI0509876 A BR PI0509876A
Authority
BR
Brazil
Prior art keywords
methods
cell proliferation
angiogenesis
thrombin
administering
Prior art date
Application number
BRPI0509876-9A
Other languages
English (en)
Inventor
Cheng-Der Tony Yu
Original Assignee
Canyon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Canyon Pharmaceuticals Inc filed Critical Canyon Pharmaceuticals Inc
Publication of BRPI0509876A publication Critical patent/BRPI0509876A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • A61K38/57Protease inhibitors from animals; from humans
    • A61K38/58Protease inhibitors from animals; from humans from leeches, e.g. hirudin, eglin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)

Abstract

MéTODOS PARA CONTROLAR A ANGIOGêNESE E A PROLIFERAçãO DE CéLULAS. A presente invenção refere-se, de um modo geral, aos métodos de inibir a angiogênese em um paciente, por administração de uma quantidade efetiva inibidora da angiogênese de um inibidor da trombina, e ao tratamento de estados de doenças que resultam da proliferação descontrolada das células, por administração de um inibidor da trombina sozinho ou coadministração de um inibidor da trombina com um agente anticâncer ou citotóxico. Especificamente, os inibidores da trombina usados nos métodos da presente invenção são as hirudinas.
BRPI0509876-9A 2004-04-12 2005-04-05 métodos para controlar a angiogênese e a proliferação de células BRPI0509876A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56174104P 2004-04-12 2004-04-12
PCT/US2005/011549 WO2005099749A2 (en) 2004-04-12 2005-04-05 Methods for controlling angiogenesis and cell proliferation

Publications (1)

Publication Number Publication Date
BRPI0509876A true BRPI0509876A (pt) 2007-10-16

Family

ID=35150501

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0509876-9A BRPI0509876A (pt) 2004-04-12 2005-04-05 métodos para controlar a angiogênese e a proliferação de células

Country Status (13)

Country Link
US (3) US7795205B2 (pt)
EP (1) EP1753291A4 (pt)
JP (1) JP2007532646A (pt)
AU (1) AU2005232625B2 (pt)
BR (1) BRPI0509876A (pt)
CA (1) CA2562756C (pt)
IL (1) IL178578A (pt)
MY (1) MY146091A (pt)
NZ (1) NZ551146A (pt)
SG (1) SG160323A1 (pt)
TW (1) TWI362941B (pt)
WO (1) WO2005099749A2 (pt)
ZA (1) ZA200609219B (pt)

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US7795205B2 (en) * 2004-04-12 2010-09-14 Canyon Pharmaceuticals, Inc. Methods for effecting regression of tumor mass and size in a metastasized pancreatic tumor
CN102225966B (zh) 2004-10-19 2012-12-26 隆萨股份公司 用于固相肽合成的方法
US20100239650A1 (en) * 2009-03-20 2010-09-23 Wilson Kurt Whitekettle Isothiazolin biodelivery systems
US20100239630A1 (en) * 2009-03-20 2010-09-23 Wilson Kurt Whitekettle Phosphonium salts delivery systems
US20100239627A1 (en) * 2009-03-20 2010-09-23 Wilson Kurt Whitekettle Quarternary ammonium salts delivery systems
US20100239651A1 (en) * 2009-03-20 2010-09-23 Wilson Kurt Whitekettle Nitrilopropionamide delivery systems
US20100239626A1 (en) * 2009-03-20 2010-09-23 Wilson Kurt Whitekettle Propanediol delivery systems
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CN104906037A (zh) * 2015-06-23 2015-09-16 广西复鑫益生物科技有限公司平南分公司 一种重组水蛭素滴眼液及其制备方法
CN110404060A (zh) * 2018-04-28 2019-11-05 复旦大学 凝血酶抑制剂在制备抗肿瘤侵袭转移药物中的用途

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Also Published As

Publication number Publication date
TWI362941B (en) 2012-05-01
EP1753291A2 (en) 2007-02-21
AU2005232625B2 (en) 2011-07-28
EP1753291A4 (en) 2009-08-12
US20110224150A1 (en) 2011-09-15
MY146091A (en) 2012-06-29
WO2005099749A3 (en) 2006-08-03
NZ551146A (en) 2009-04-30
TW200538466A (en) 2005-12-01
US20090269422A1 (en) 2009-10-29
AU2005232625A1 (en) 2005-10-27
CA2562756C (en) 2011-08-23
US7795205B2 (en) 2010-09-14
US20050233966A1 (en) 2005-10-20
ZA200609219B (en) 2012-02-29
WO2005099749A2 (en) 2005-10-27
CA2562756A1 (en) 2005-10-27
IL178578A0 (en) 2007-02-11
SG160323A1 (en) 2010-04-29
JP2007532646A (ja) 2007-11-15
IL178578A (en) 2013-06-27

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 11A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.