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BR9911487A - Composto de resina de fluorofenila, e, processos para preparar uma amida, um composto amina, o composto de resina de fluorofenila, um composto sulfonamida, um composto, um composto de amina dissubstituìda, o composto de resina de fluorofenila e um composto de carbonila substituìdo em a - Google Patents

Composto de resina de fluorofenila, e, processos para preparar uma amida, um composto amina, o composto de resina de fluorofenila, um composto sulfonamida, um composto, um composto de amina dissubstituìda, o composto de resina de fluorofenila e um composto de carbonila substituìdo em a

Info

Publication number
BR9911487A
BR9911487A BR9911487-9A BR9911487A BR9911487A BR 9911487 A BR9911487 A BR 9911487A BR 9911487 A BR9911487 A BR 9911487A BR 9911487 A BR9911487 A BR 9911487A
Authority
BR
Brazil
Prior art keywords
compound
fluorophenyl resin
amine
processes
fluorophenyl
Prior art date
Application number
BR9911487-9A
Other languages
English (en)
Inventor
Joseph M Salvino
Robert D Groneberg
John E Airey
Gregory B Poli
Gerard M Mcgeehan
Richard F Labaudiniere
Francois-Frederic Clerc
Daniel Noul Andre Bezard
Original Assignee
Aventis Pharm Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharm Prod Inc filed Critical Aventis Pharm Prod Inc
Publication of BR9911487A publication Critical patent/BR9911487A/pt

Links

Classifications

    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N24/00Investigating or analyzing materials by the use of nuclear magnetic resonance, electron paramagnetic resonance or other spin effects
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/14Esterification
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/18Introducing halogen atoms or halogen-containing groups
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/18Introducing halogen atoms or halogen-containing groups
    • C08F8/20Halogenation
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/26Removing halogen atoms or halogen-containing groups from the molecule
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/34Introducing sulfur atoms or sulfur-containing groups
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/34Introducing sulfur atoms or sulfur-containing groups
    • C08F8/36Sulfonation; Sulfation
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00Chemical modification by after-treatment
    • C08F8/40Introducing phosphorus atoms or phosphorus-containing groups
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F2800/00Copolymer characterised by the proportions of the comonomers expressed
    • C08F2800/20Copolymer characterised by the proportions of the comonomers expressed as weight or mass percentages
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08FMACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F2810/00Chemical modification of a polymer
    • C08F2810/20Chemical modification of a polymer leading to a crosslinking, either explicitly or inherently
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N24/00Investigating or analyzing materials by the use of nuclear magnetic resonance, electron paramagnetic resonance or other spin effects
    • G01N24/08Investigating or analyzing materials by the use of nuclear magnetic resonance, electron paramagnetic resonance or other spin effects by using nuclear magnetic resonance

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Analytical Chemistry (AREA)
  • Pathology (AREA)
  • High Energy & Nuclear Physics (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Physics & Mathematics (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Polyamides (AREA)
  • Polyurethanes Or Polyureas (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

"COMPOSTO DE RESINA DE FLUOROFENILA, E, PROCESSOS PARA PREPARAR UMA AMIDA, UM COMPOSTO AMINA, O COMPOSTO DE RESINA DE FLUOROFENILA, UM COMPOSTO SULFONAMIDA, UM COMPOSTO, UM COMPOSTO DE AMINA DISSUBSTITUìDA, O COMPOSTO DE RESINA DE FLUOROFENILA E UM COMPOSTO DE CARBONILA SUBSTITUìDO EM <244>" A invenção refere-se a um composto de resina de fluorofenila, a processos para sua preparação; e a seu uso na síntese de fase sólida de amidas, peptídeos, ácidos hidroxâmicos, aminas, uretanas, carbonatos carbamatos, sulfonamidas e compostos carbonila substituídos em <244>.
BR9911487-9A 1998-06-24 1999-06-23 Composto de resina de fluorofenila, e, processos para preparar uma amida, um composto amina, o composto de resina de fluorofenila, um composto sulfonamida, um composto, um composto de amina dissubstituìda, o composto de resina de fluorofenila e um composto de carbonila substituìdo em a BR9911487A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9055898P 1998-06-24 1998-06-24
PCT/US1999/014252 WO1999067228A1 (en) 1998-06-24 1999-06-23 Fluorophenyl resin compounds

Publications (1)

Publication Number Publication Date
BR9911487A true BR9911487A (pt) 2001-03-20

Family

ID=22223315

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9911487-9A BR9911487A (pt) 1998-06-24 1999-06-23 Composto de resina de fluorofenila, e, processos para preparar uma amida, um composto amina, o composto de resina de fluorofenila, um composto sulfonamida, um composto, um composto de amina dissubstituìda, o composto de resina de fluorofenila e um composto de carbonila substituìdo em a

Country Status (22)

Country Link
US (1) US6639023B1 (pt)
EP (1) EP1089988B1 (pt)
JP (1) JP2002518555A (pt)
KR (1) KR100634035B1 (pt)
CN (1) CN1185259C (pt)
AP (1) AP1347A (pt)
AT (1) ATE439351T1 (pt)
AU (1) AU764153B2 (pt)
BG (1) BG65208B1 (pt)
BR (1) BR9911487A (pt)
CA (1) CA2335760A1 (pt)
CZ (1) CZ20004794A3 (pt)
DE (1) DE69941260D1 (pt)
EA (1) EA004061B1 (pt)
HU (1) HUP0201967A3 (pt)
IL (2) IL140001A0 (pt)
NO (1) NO20006662D0 (pt)
OA (1) OA11575A (pt)
PL (1) PL345116A1 (pt)
SK (1) SK20132000A3 (pt)
UA (1) UA57153C2 (pt)
WO (1) WO1999067228A1 (pt)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6281227B1 (en) * 1996-12-13 2001-08-28 Aventis Pharma Deutschland Gmbh Sulfonic acid sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
JP4669933B2 (ja) * 2000-12-07 2011-04-13 国立大学法人東京工業大学 スルホン誘導体及びその製造方法
JP4598403B2 (ja) 2001-11-14 2010-12-15 ルミネックス コーポレーション 固定化の改善ための官能化組成物
CN100334120C (zh) * 2002-07-12 2007-08-29 东华大学 含杂环结构的氟树脂、制造方法及其用途
US6861473B2 (en) * 2003-02-28 2005-03-01 Baxter International Inc. Macromolecular ketoaldehydes
WO2006058720A2 (en) 2003-11-03 2006-06-08 Probiodrug Ag Novel compounds for the treatment of neurological disorders
JP2007509898A (ja) 2003-11-03 2007-04-19 プロビオドルグ エージー 神経障害治療に有用な組合せ
US7867774B2 (en) 2004-10-12 2011-01-11 Luminex Corporation Methods for altering surface characteristics of microspheres
EP1971614A1 (en) 2005-11-14 2008-09-24 Probiodrug AG Cyclopropyl-fused pyrrolidine derivatives as dipeptidyl peptidase iv inhibitors
KR20090004950A (ko) 2006-04-12 2009-01-12 프로비오드룩 아게 효소 억제제
CN101668525A (zh) 2007-03-01 2010-03-10 前体生物药物股份公司 谷氨酰胺酰环化酶抑制剂的新用途
CN111187407B (zh) * 2019-05-15 2022-04-29 江苏冰城氢能科技有限公司 一种燃料电池用耐高温高透气性磺化微孔聚合物及其铂碳复合膜的制备方法
EP3871665B1 (en) 2020-02-28 2025-12-24 Martin-Luther-Universität Halle-Wittenberg Inhibitors of rna-binding proteins as anti-cancer drugs
CN118084741A (zh) * 2024-03-29 2024-05-28 天津众泰材料科技有限公司 一种感光化合物tppa-pac的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4786684A (en) * 1986-08-21 1988-11-22 The Mount Sinai School Of Medicine Of The City University Of New York Benzylthioether-linked solid support-bound thiol compounds and method for peptide synthesis
US5116994A (en) * 1989-04-19 1992-05-26 Fuji Photo Film Co., Ltd. Deacylating agent and deacylating method
SU1761762A1 (ru) * 1989-11-09 1992-09-15 Ленинградский государственный университет Пара-(4-гидрокси-2,3,5,6-тетрафторбензил)полистирол в качестве активатора дл синтеза пептидов
US5116995A (en) * 1990-05-25 1992-05-26 Taisho Pharmaceutical Co., Ltd. Carbazole compounds
US5266651A (en) * 1991-05-03 1993-11-30 E. I. Du Pont De Nemours And Company Crosslinked poled polymers for nonlinear optic applications and method of making them
SG48166A1 (en) 1993-12-15 1998-04-17 Conbichem Inc Combinatorial libraries and methods for their use
US5792815A (en) * 1995-05-08 1998-08-11 Fmc Corporation Functionalized polymer produced with functionalized initiators by anionic polymerization
US5830539A (en) * 1995-11-17 1998-11-03 The State Of Oregon Acting By And Through The State Board Of Higher Education On Behalf Of The University Of Oregon Methods for functionalizing and coating substrates and devices made according to the methods
WO1998045231A1 (en) 1997-04-09 1998-10-15 Cadus Pharmaceutical Corporation Supports for solid phase synthesis
WO1999025752A1 (en) * 1997-11-18 1999-05-27 Aventis Pharmaceuticals Products Inc. Functionalized resin for the synthesis of amides and peptides

Also Published As

Publication number Publication date
KR100634035B1 (ko) 2006-10-17
EA200100070A1 (ru) 2001-06-25
US6639023B1 (en) 2003-10-28
EP1089988B1 (en) 2009-08-12
PL345116A1 (en) 2001-12-03
AP1347A (en) 2004-12-16
JP2002518555A (ja) 2002-06-25
AU4712899A (en) 2000-01-10
EP1089988A1 (en) 2001-04-11
CA2335760A1 (en) 1999-12-29
AP2000001995A0 (en) 2000-12-31
UA57153C2 (uk) 2003-06-16
NO20006662L (no) 2000-12-27
EA004061B1 (ru) 2003-12-25
CZ20004794A3 (cs) 2001-08-15
IL140001A0 (en) 2002-02-10
DE69941260D1 (de) 2009-09-24
CN1306524A (zh) 2001-08-01
WO1999067228A1 (en) 1999-12-29
OA11575A (en) 2004-07-26
HUP0201967A3 (en) 2010-01-28
BG65208B1 (bg) 2007-07-31
BG105143A (en) 2001-07-31
ATE439351T1 (de) 2009-08-15
IL140001A (en) 2008-11-26
SK20132000A3 (sk) 2001-06-11
AU764153B2 (en) 2003-08-14
KR20010083066A (ko) 2001-08-31
NO20006662D0 (no) 2000-12-27
CN1185259C (zh) 2005-01-19
HUP0201967A2 (en) 2002-09-28
EP1089988A4 (en) 2005-01-19

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements