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BR9407889A - Derivados 2(pyrazol-3-yl)carbapenem - Google Patents

Derivados 2(pyrazol-3-yl)carbapenem

Info

Publication number
BR9407889A
BR9407889A BR9407889A BR9407889A BR9407889A BR 9407889 A BR9407889 A BR 9407889A BR 9407889 A BR9407889 A BR 9407889A BR 9407889 A BR9407889 A BR 9407889A BR 9407889 A BR9407889 A BR 9407889A
Authority
BR
Brazil
Prior art keywords
carbapenem
pyrazol
derivatives
Prior art date
Application number
BR9407889A
Other languages
English (en)
Inventor
Steven Coulton
Jeremy David Hinks
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939322284A external-priority patent/GB9322284D0/en
Priority claimed from GB9410929A external-priority patent/GB9410929D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of BR9407889A publication Critical patent/BR9407889A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D477/00Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/14Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR9407889A 1993-10-29 1994-10-25 Derivados 2(pyrazol-3-yl)carbapenem BR9407889A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939322284A GB9322284D0 (en) 1993-10-29 1993-10-29 Novel compounds
GB9410929A GB9410929D0 (en) 1994-06-01 1994-06-01 Novel compounds
PCT/GB1994/002347 WO1995011905A1 (en) 1993-10-29 1994-10-25 2-(pyrazol-3-yl)carbapenem derivatives

Publications (1)

Publication Number Publication Date
BR9407889A true BR9407889A (pt) 1996-10-29

Family

ID=26303758

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9407889A BR9407889A (pt) 1993-10-29 1994-10-25 Derivados 2(pyrazol-3-yl)carbapenem

Country Status (22)

Country Link
US (1) US5612477A (pt)
EP (1) EP0725783B1 (pt)
JP (1) JP3703146B2 (pt)
KR (1) KR960705827A (pt)
CN (1) CN1167486A (pt)
AP (1) AP9600800A0 (pt)
AT (1) ATE229957T1 (pt)
AU (1) AU697108B2 (pt)
BG (1) BG100551A (pt)
BR (1) BR9407889A (pt)
CA (1) CA2175054C (pt)
CZ (1) CZ122996A3 (pt)
DE (1) DE69431919T2 (pt)
ES (1) ES2188621T3 (pt)
FI (1) FI961817A7 (pt)
HU (1) HUT75519A (pt)
NO (1) NO961654L (pt)
NZ (1) NZ274878A (pt)
OA (1) OA10287A (pt)
PL (1) PL314173A1 (pt)
SK (1) SK53696A3 (pt)
WO (1) WO1995011905A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020147333A1 (en) 1993-10-29 2002-10-10 Smithkline Beecham P.L.C. 2-(pyrazol-3-yl)carbapenem derivatives
WO1996011932A1 (en) * 1994-10-14 1996-04-25 Smithkline Beecham Plc 2-(imidazol-4-yl)carbapeneme derivatives, intermediates thereof and use as antibacterials
IL118092A0 (en) * 1995-05-03 1996-09-12 Smithkline Beecham Plc Antibacterial compounds their preparation and pharmaceutical compositions containing them
JPH11504912A (ja) * 1995-05-03 1999-05-11 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー カルバペネムのエステル
GB0400329D0 (en) * 2004-01-08 2004-02-11 Glaxo Group Ltd Novel processes
GB0400405D0 (en) * 2004-01-09 2004-02-11 Glaxo Group Ltd Novel processes
JP2007039383A (ja) * 2005-08-03 2007-02-15 Dainippon Sumitomo Pharma Co Ltd アリールカルバペネム化合物の製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1593524A (en) * 1976-11-19 1981-07-15 Merck & Co Inc 1-carba-2-penem-3-carboxylic acids
US4260627A (en) * 1978-10-24 1981-04-07 Merck & Co., Inc. 1-, 6- And 2-substituted-1-carba-2-penem-3-carboxylic acids
EP0430037A3 (en) * 1989-11-21 1992-05-27 Banyu Pharmaceutical Co., Ltd. Process for producing 2-carbon-substituted carbapenem derivatives
CA2036960A1 (en) * 1990-02-26 1991-08-27 Thomas A. Rano Novel synthesis of carbapenem intermediates
JP3233434B2 (ja) * 1992-04-01 2001-11-26 塩野義製薬株式会社 カルバペネム誘導体

Also Published As

Publication number Publication date
AP9600800A0 (en) 1996-04-30
DE69431919T2 (de) 2003-11-13
EP0725783A1 (en) 1996-08-14
AU697108B2 (en) 1998-09-24
DE69431919D1 (de) 2003-01-30
NO961654D0 (no) 1996-04-25
CN1167486A (zh) 1997-12-10
ATE229957T1 (de) 2003-01-15
NZ274878A (en) 1998-02-26
HU9601097D0 (en) 1996-07-29
JPH09504285A (ja) 1997-04-28
FI961817A0 (fi) 1996-04-29
SK53696A3 (en) 1996-10-02
CA2175054C (en) 2005-07-12
NO961654L (no) 1996-06-11
ES2188621T3 (es) 2003-07-01
CZ122996A3 (en) 1996-10-16
CA2175054A1 (en) 1995-05-04
PL314173A1 (en) 1996-08-19
FI961817L (fi) 1996-06-28
KR960705827A (ko) 1996-11-08
AU7997594A (en) 1995-05-22
OA10287A (en) 1997-10-07
WO1995011905A1 (en) 1995-05-04
JP3703146B2 (ja) 2005-10-05
HUT75519A (en) 1997-05-28
FI961817A7 (fi) 1996-06-28
BG100551A (bg) 1997-01-31
EP0725783B1 (en) 2002-12-18
US5612477A (en) 1997-03-18

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Legal Events

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