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BR0311749A - Processo para produzir um composto, e, composto - Google Patents

Processo para produzir um composto, e, composto

Info

Publication number
BR0311749A
BR0311749A BR0311749-9A BR0311749A BR0311749A BR 0311749 A BR0311749 A BR 0311749A BR 0311749 A BR0311749 A BR 0311749A BR 0311749 A BR0311749 A BR 0311749A
Authority
BR
Brazil
Prior art keywords
compound
producing
protecting group
arila
alkylene
Prior art date
Application number
BR0311749-9A
Other languages
English (en)
Inventor
Hiroshi Tomori
Keijiro Kobayashi
Fumihiko Toriyama
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of BR0311749A publication Critical patent/BR0311749A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/52Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"PROCESSO PARA PRODUZIR UM COMPOSTO, E, COMPOSTO". Um processo para produzir um tioéter cíclico e um intermediário sintético do mesmo. Particularmente, um composto de fórmula geral (5): em que G^ 1^ representa um alquileno, R^ 1^ representa um grupo de proteção para tiol, R^ 2^ representa hidrogênio ou um grupo de proteção para amino, e Ar representa uma arila, etc.
BR0311749-9A 2002-06-11 2003-06-09 Processo para produzir um composto, e, composto BR0311749A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002169967 2002-06-11
PCT/JP2003/007291 WO2003104240A1 (ja) 2002-06-11 2003-06-09 環状チオエーテル類の製造法及びその合成中間体

Publications (1)

Publication Number Publication Date
BR0311749A true BR0311749A (pt) 2005-03-08

Family

ID=29727753

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0311749-9A BR0311749A (pt) 2002-06-11 2003-06-09 Processo para produzir um composto, e, composto

Country Status (9)

Country Link
EP (1) EP1533314A4 (pt)
KR (1) KR20050008813A (pt)
CN (1) CN100334092C (pt)
AU (1) AU2003242092A1 (pt)
BR (1) BR0311749A (pt)
CA (1) CA2489255A1 (pt)
IL (1) IL165512A0 (pt)
TW (1) TW200403203A (pt)
WO (1) WO2003104240A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2812526A1 (en) 2010-05-06 2011-11-10 Vertex Pharmaceuticals Incorporated Heterocyclic chromene-spirocyclic piperidine amides as modulators of ion channels
DK2670752T3 (en) 2011-02-02 2016-07-04 Vertex Pharma PYRROLOPYRAZINE SPIROCYCLIC PIPERIDINAMIDE AS ION CHANNEL MODULATORS
WO2012112743A1 (en) 2011-02-18 2012-08-23 Vertex Pharmaceuticals Incorporated Chroman - spirocyclic piperidine amides as modulators of ion channels
EP2686325B1 (en) 2011-03-14 2016-12-14 Vertex Pharmaceuticals Incorporated Morpholine-spirocyclic piperidine amides as modulators of ion channels

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2135494C1 (ru) * 1995-12-01 1999-08-27 Санкио Компани Лимитед Гетероциклические соединения и композиция на их основе, проявляющая антагонистическое действие в отношении рецепторов тахикинина
PT1048658E (pt) * 1997-12-04 2005-10-31 Sankyo Co Derivados heterociclicos acilados aliciclicos
AU6621600A (en) * 1999-08-04 2001-03-05 Millennium Pharmaceuticals, Inc. Melanocortin-4 receptor binding compounds and methods of use thereof
WO2001029027A1 (en) * 1999-10-22 2001-04-26 Sankyo Company, Limited 2-alkoxybenzene derivatives
EP1363890A4 (en) * 2001-02-07 2009-06-10 Ore Pharmaceuticals Inc MELANOCORTIN-4-RECEPTOR BINDING COMPOUNDS AND METHOD FOR THEIR APPLICATION

Also Published As

Publication number Publication date
AU2003242092A1 (en) 2003-12-22
CA2489255A1 (en) 2003-12-18
IL165512A0 (en) 2006-01-15
KR20050008813A (ko) 2005-01-21
CN100334092C (zh) 2007-08-29
TW200403203A (en) 2004-03-01
EP1533314A4 (en) 2006-08-02
CN1675221A (zh) 2005-09-28
WO2003104240A1 (ja) 2003-12-18
EP1533314A1 (en) 2005-05-25

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A E 8A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2116 DE 26/07/2011.