AU2016403208B2 - An improved process for the preparation of Linezolid - Google Patents
An improved process for the preparation of Linezolid Download PDFInfo
- Publication number
- AU2016403208B2 AU2016403208B2 AU2016403208A AU2016403208A AU2016403208B2 AU 2016403208 B2 AU2016403208 B2 AU 2016403208B2 AU 2016403208 A AU2016403208 A AU 2016403208A AU 2016403208 A AU2016403208 A AU 2016403208A AU 2016403208 B2 AU2016403208 B2 AU 2016403208B2
- Authority
- AU
- Australia
- Prior art keywords
- fluoro
- formula
- compound
- phenyl
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- FKZUTWSVQLXKQE-OAHLLOKOSA-N O=C(c1c2cccc1)N(C[C@@H](CN1c(cc3F)ccc3N3CCOCC3)OC1=O)C2=O Chemical compound O=C(c1c2cccc1)N(C[C@@H](CN1c(cc3F)ccc3N3CCOCC3)OC1=O)C2=O FKZUTWSVQLXKQE-OAHLLOKOSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201641013830 | 2016-04-21 | ||
| IN201641013830 | 2016-04-21 | ||
| PCT/IB2016/053003 WO2017182853A1 (fr) | 2016-04-21 | 2016-05-23 | Procédé perfectionné pour la préparation de linézolide |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2016403208A1 AU2016403208A1 (en) | 2018-05-10 |
| AU2016403208B2 true AU2016403208B2 (en) | 2018-10-25 |
Family
ID=60115753
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2016403208A Active AU2016403208B2 (en) | 2016-04-21 | 2016-05-23 | An improved process for the preparation of Linezolid |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP3250568A4 (fr) |
| KR (1) | KR101832115B1 (fr) |
| AU (1) | AU2016403208B2 (fr) |
| NZ (1) | NZ741891A (fr) |
| RU (1) | RU2766082C9 (fr) |
| WO (1) | WO2017182853A1 (fr) |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN2013CH05865A (fr) * | 2013-12-16 | 2015-06-19 | Optimus Drugs P Ltd |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0004388A3 (en) | 1997-11-07 | 2001-10-29 | Upjohn Co | Process for the preparation of oxazolidinones, intermediates and preparation thereof |
| PL1768967T3 (pl) * | 2004-07-20 | 2009-09-30 | Symed Labs Ltd | Nowe związki pośrednie do wytwarzania linezolidu oraz związki pokrewne |
| WO2011114210A2 (fr) * | 2010-03-15 | 2011-09-22 | Jubilant Life Sciences Limited | Procédés de préparation de linézolide |
| US9206141B2 (en) * | 2010-04-30 | 2015-12-08 | Indiana University Research And Technology Corporation | Processes for preparing linezolid |
| SI2595968T1 (sl) * | 2011-02-24 | 2016-01-29 | Lee Pharma Limited | Novi postopek za pripravo linezolida in njegovih novih intermediatov |
| CN103420933B (zh) * | 2012-05-26 | 2016-03-02 | 鲁南制药集团股份有限公司 | 一种利奈唑胺的制备方法 |
| US9593104B2 (en) | 2013-03-14 | 2017-03-14 | Benova Labs Pvt. Limited | Process for the preparation of oxazolidinone derivatives |
| IN2014CH00444A (fr) | 2014-01-31 | 2015-08-07 | Optimus Drugs P Ltd |
-
2016
- 2016-05-23 EP EP16876979.2A patent/EP3250568A4/fr not_active Withdrawn
- 2016-05-23 KR KR1020177029421A patent/KR101832115B1/ko active Active
- 2016-05-23 AU AU2016403208A patent/AU2016403208B2/en active Active
- 2016-05-23 NZ NZ741891A patent/NZ741891A/en unknown
- 2016-05-23 RU RU2018109135A patent/RU2766082C9/ru active
- 2016-05-23 WO PCT/IB2016/053003 patent/WO2017182853A1/fr not_active Ceased
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN2013CH05865A (fr) * | 2013-12-16 | 2015-06-19 | Optimus Drugs P Ltd |
Also Published As
| Publication number | Publication date |
|---|---|
| KR101832115B1 (ko) | 2018-02-23 |
| RU2766082C1 (ru) | 2022-02-07 |
| EP3250568A4 (fr) | 2018-08-01 |
| KR20170128485A (ko) | 2017-11-22 |
| NZ741891A (en) | 2020-05-29 |
| AU2016403208A1 (en) | 2018-05-10 |
| EP3250568A1 (fr) | 2017-12-06 |
| WO2017182853A1 (fr) | 2017-10-26 |
| RU2766082C9 (ru) | 2022-02-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FGA | Letters patent sealed or granted (standard patent) |