AU2002237704A1 - Methods for the stereoselective synthesis of substituted piperidines - Google Patents
Methods for the stereoselective synthesis of substituted piperidinesInfo
- Publication number
- AU2002237704A1 AU2002237704A1 AU2002237704A AU3770402A AU2002237704A1 AU 2002237704 A1 AU2002237704 A1 AU 2002237704A1 AU 2002237704 A AU2002237704 A AU 2002237704A AU 3770402 A AU3770402 A AU 3770402A AU 2002237704 A1 AU2002237704 A1 AU 2002237704A1
- Authority
- AU
- Australia
- Prior art keywords
- methods
- stereoselective synthesis
- substituted piperidines
- piperidines
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25120900P | 2000-12-04 | 2000-12-04 | |
| US60/251,209 | 2000-12-04 | ||
| US27560001P | 2001-03-13 | 2001-03-13 | |
| US60/275,600 | 2001-03-13 | ||
| PCT/US2001/047037 WO2002046157A2 (en) | 2000-12-04 | 2001-12-04 | Methods for the stereoselective synthesis of substituted piperidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2002237704A1 true AU2002237704A1 (en) | 2002-06-18 |
Family
ID=26941482
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002237704A Abandoned AU2002237704A1 (en) | 2000-12-04 | 2001-12-04 | Methods for the stereoselective synthesis of substituted piperidines |
Country Status (3)
| Country | Link |
|---|---|
| US (3) | US6703508B2 (en) |
| AU (1) | AU2002237704A1 (en) |
| WO (1) | WO2002046157A2 (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7294637B2 (en) * | 2000-09-11 | 2007-11-13 | Sepracor, Inc. | Method of treating addiction or dependence using a ligand for a monamine receptor or transporter |
| CA2422055A1 (en) * | 2000-09-11 | 2002-03-21 | Sepracor, Inc. | Ligands for monoamine receptors and transporters, and methods of use thereof (neurotransmission) |
| AU2002332659A1 (en) * | 2001-08-21 | 2003-03-03 | Sepracor, Inc. | 2-substituted piperidines that are ligands for monoamine receptors and transporters |
| US7153858B2 (en) | 2003-01-31 | 2006-12-26 | Epix Delaware, Inc. | Arylpiperazinyl compounds |
| JP5424639B2 (en) * | 2005-05-22 | 2014-02-26 | ユー．エス．ボラックス インコーポレイテッド | Symbiotic lethality formulation for polymer materials |
| US7977336B2 (en) | 2006-12-28 | 2011-07-12 | Banyu Pharmaceutical Co. Ltd | Aminopyrimidine derivatives as PLK1 inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3029244A (en) * | 1959-08-31 | 1962-04-10 | Research Corp | Aroylpiperidinols and esters thereof |
| US4012396A (en) | 1973-05-21 | 1977-03-15 | Hoffmann-La Roche Inc. | Processes and intermediates for cis or trans 2-or 3-(1-acyl-3-vinyl-4-piperidine)acetic or propionic acid esters |
| FR2649098A1 (en) | 1989-06-29 | 1991-01-04 | Centre Nat Rech Scient | CHIRAL POLYMERS FOR THE SYNTHESIS OF ENANTIOMERICALLY PURE AMINOACIDES |
| US5332817A (en) | 1990-01-04 | 1994-07-26 | Pfizer Inc. | 3-aminopiperidine derivatives and related nitrogen containing heterocycles |
| US5013842A (en) | 1990-01-22 | 1991-05-07 | Monsanto Company | Synthesis of chiral pyrrolidine and piperidine glycosidase inhibitors |
| US5420283A (en) | 1993-08-02 | 1995-05-30 | Pfizer Inc. | Resolution of (R)-2-benzylsuccinic acid 4-[4-(N-t-butoxycarbonylmethylamino)-piperidine] amide |
| US5972952A (en) | 1995-12-11 | 1999-10-26 | Le Centre National De La Recherche Scientifique | Neuroprotective pharmaceutical composition containing stereoisomers of arylcyclohexylamines |
| US5952506A (en) | 1997-04-24 | 1999-09-14 | American Home Products Corporation | Process for the synthesis of 4- 6- (hexylcarbamoyloxy) hexylcarbamoyloxy!-piperidine-1-carboxylic acid 4-phenoxyphenyl ester |
| US6521561B1 (en) | 1998-05-01 | 2003-02-18 | President And Fellows Of Harvard College | Main-group metal based asymmetric catalysts and applications thereof |
| EP1187810A2 (en) | 1999-05-25 | 2002-03-20 | Sepracor, Inc. | Heterocyclic analgesic compounds and their use |
| US6645980B1 (en) | 2000-05-25 | 2003-11-11 | Sepracor Inc. | Heterocyclic analgesic compounds and methods of use thereof |
| WO2001000207A1 (en) * | 1999-06-30 | 2001-01-04 | Merck & Co., Inc. | Src kinase inhibitor compounds |
-
2001
- 2001-12-04 WO PCT/US2001/047037 patent/WO2002046157A2/en not_active Ceased
- 2001-12-04 AU AU2002237704A patent/AU2002237704A1/en not_active Abandoned
- 2001-12-04 US US10/012,242 patent/US6703508B2/en not_active Expired - Lifetime
-
2004
- 2004-02-27 US US10/789,414 patent/US7005524B2/en not_active Expired - Lifetime
-
2006
- 2006-02-28 US US11/364,506 patent/US7692019B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002046157A3 (en) | 2003-02-27 |
| US7692019B2 (en) | 2010-04-06 |
| US20020177721A1 (en) | 2002-11-28 |
| US6703508B2 (en) | 2004-03-09 |
| US20060211864A1 (en) | 2006-09-21 |
| WO2002046157A2 (en) | 2002-06-13 |
| US7005524B2 (en) | 2006-02-28 |
| US20040235893A1 (en) | 2004-11-25 |
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