AU2002235129A1 - Treatment of anti-depression drug-induced sexual dysfunction with apomorphine - Google Patents

Treatment of anti-depression drug-induced sexual dysfunction with apomorphine

Info

Publication number: AU2002235129A1
Authority: AU; Australia
Prior art keywords: hydrochloride; apomoφhine; patient; administered; apomorphine
Prior art date: 2000-11-15
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2002235129A

Other languages

English (en)

Inventor

Renee J. Perdok

Dustin D. Ruff

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Tap Pharmaceuticals Inc

Original Assignee

TAP Holding Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2001-11-14

Publication date

2002-05-27

2001-11-14 Application filed by TAP Holding Inc filed Critical TAP Holding Inc

2002-05-27 Publication of AU2002235129A1 publication Critical patent/AU2002235129A1/en

Status Abandoned legal-status Critical Current

Links

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238000011282 treatment Methods 0.000 title claims description 12
VMWNQDUVQKEIOC-CYBMUJFWSA-N apomorphine Chemical compound C([C@H]1N(C)CC2)C3=CC=C(O)C(O)=C3C3=C1C2=CC=C3 VMWNQDUVQKEIOC-CYBMUJFWSA-N 0.000 title description 28
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Neurosurgery (AREA)
Endocrinology (AREA)
Biomedical Technology (AREA)
Emergency Medicine (AREA)
Neurology (AREA)
Reproductive Health (AREA)
Pain & Pain Management (AREA)
Gynecology & Obstetrics (AREA)
Otolaryngology (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Medicinal Preparation (AREA)

AU2002235129A 2000-11-15 2001-11-14 Treatment of anti-depression drug-induced sexual dysfunction with apomorphine Abandoned AU2002235129A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US24903100P	2000-11-15	2000-11-15
US60/249,031		2000-11-15
PCT/US2001/043933 WO2002039879A2 (fr)	2000-11-15	2001-11-14	Traitement d'un dysfonctionnement sexuel entraine par une medication antidepressive par apomorphine

Publications (1)

Publication Number	Publication Date
AU2002235129A1 true AU2002235129A1 (en)	2002-05-27

Family

ID=22941748

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2002235129A Abandoned AU2002235129A1 (en)	2000-11-15	2001-11-14	Treatment of anti-depression drug-induced sexual dysfunction with apomorphine

Country Status (18)

Country	Link
US (1)	US6528521B2 (fr)
EP (1)	EP1341536A4 (fr)
JP (1)	JP2004513899A (fr)
KR (1)	KR20030077538A (fr)
CN (1)	CN1486183A (fr)
AU (1)	AU2002235129A1 (fr)
BG (1)	BG107874A (fr)
BR (1)	BR0111982A (fr)
CA (1)	CA2429047A1 (fr)
CZ (1)	CZ20031540A3 (fr)
HU (1)	HUP0302436A3 (fr)
IL (1)	IL155667A0 (fr)
MX (1)	MXPA03004288A (fr)
NO (1)	NO20032189L (fr)
PL (1)	PL361875A1 (fr)
SK (1)	SK7422003A3 (fr)
WO (1)	WO2002039879A2 (fr)
ZA (1)	ZA200303471B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6787532B2 (en) *	2000-08-05	2004-09-07	Smithkline Beecham Corporation	Formulation containing anti-inflammatory androstane derivatives
US20060178394A1 (en) *	2003-04-14	2006-08-10	Staniforth John N	Pharmaceutical compositions comprising apomorphine for pulmonary inhalation
US20040204439A1 (en) *	2003-04-14	2004-10-14	Staniforth John Nicholas	Composition, device, and method for treating sexual dysfunction via inhalation
EP1667972B1 (fr)	2003-09-10	2013-06-19	Brentwood Equities Ltd.	Diastereoisomeres de 4-aryloxy-3-hydroxypiperidines
GB0425758D0 (en)	2004-11-23	2004-12-22	Vectura Ltd	Preparation of pharmaceutical compositions
GB0721394D0 (en) *	2007-10-31	2007-12-12	Vectura Group Plc	Compositions for trating parkinson's disease
KR102161392B1 (ko)	2010-12-16	2020-10-05	선오비온 파마슈티컬스 인코포레이티드	설하 필름
CA2893427C (fr)	2012-12-24	2023-01-10	Neurogastrx, Inc.	Methodes de traitement d'affections du tractus digestif
PT3285771T (pt)	2015-04-21	2025-03-31	Sunovion Pharmaceuticals Inc	Métodos de tratamento da doença de parkinson pela administração de apomorfina a uma mucosa oral
WO2017168174A1 (fr)	2016-04-02	2017-10-05	N4 Pharma Uk Limited	Nouvelles formes pharmaceutiques du sildénafil
AU2019208396B2 (en)	2018-01-18	2024-11-14	Leukos Biotech, S. L.	Apomorphine·palmitic acid cocrystal solid particle crystalline form
US11717495B2 (en) *	2020-03-16	2023-08-08	Vella Bioscience, Inc.	Use of cannabinoids in treating anti-depressant-induced female sexual dysfunction
US10836757B1 (en)	2020-04-02	2020-11-17	Neurogastrx, Inc.	Polymorphic forms of metopimazine
CN115671106B (zh) *	2021-07-21	2024-03-19	广州新济药业科技有限公司	吗啡的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4521421A (en) *	1983-09-26	1985-06-04	Eli Lilly And Company	Treatment of sexual dysfunction
DK0689438T3 (da) *	1993-03-26	2003-09-29	Franciscus Wilhelmus He Merkus	Farmaceutiske præparater til intranasal administration af apomorfin
ES2143049T3 (es)	1994-04-22	2000-05-01	Pentech Pharmaceuticals Inc	Formas sublinguales de dosificacion que contienen apomorfina y su uso para el tratamiento de la disfuncion erectil.
US5562917A (en)	1994-12-23	1996-10-08	Pentech Pharmaceuticals, Inc.	Transdermal administration of apomorphine
US5888534A (en) *	1995-06-13	1999-03-30	Pentech Pharmaceuticals, Inc.	Controlled release of drugs delivered by sublingual or buccal administration
DK0914097T3 (da)	1996-03-12	2002-04-29	Alza Corp	Sammensætning og doseringsform omfattende opioid antagonist
US5897864A (en)	1996-05-23	1999-04-27	Cohen; Alan J.	Method for treating sexual dysfunction disorders with compositions containing ginkgo biloba
JP2001504851A (ja) *	1996-12-02	2001-04-10	メルクシヤープエンドドームリミテツド	性的機能不全の治療のためのｎｋ−１受容体拮抗薬の使用
US5945117A (en)	1998-01-30	1999-08-31	Pentech Pharmaceuticals, Inc.	Treatment of female sexual dysfunction
US6399826B1 (en) *	1999-08-11	2002-06-04	Sepracor Inc.	Salts of sibutramine metabolites, methods of making sibutramine metabolites and intermediates useful in the same, and methods of treating pain

2001
- 2001-11-14 PL PL01361875A patent/PL361875A1/xx not_active Application Discontinuation
- 2001-11-14 BR BR0111982-6A patent/BR0111982A/pt not_active IP Right Cessation
- 2001-11-14 CA CA002429047A patent/CA2429047A1/fr not_active Abandoned
- 2001-11-14 SK SK742-2003A patent/SK7422003A3/sk not_active Application Discontinuation
- 2001-11-14 IL IL15566701A patent/IL155667A0/xx unknown
- 2001-11-14 AU AU2002235129A patent/AU2002235129A1/en not_active Abandoned
- 2001-11-14 JP JP2002542257A patent/JP2004513899A/ja active Pending
- 2001-11-14 CZ CZ20031540A patent/CZ20031540A3/cs unknown
- 2001-11-14 HU HU0302436A patent/HUP0302436A3/hu unknown
- 2001-11-14 US US09/993,782 patent/US6528521B2/en not_active Expired - Fee Related
- 2001-11-14 KR KR10-2003-7006518A patent/KR20030077538A/ko not_active Withdrawn
- 2001-11-14 MX MXPA03004288A patent/MXPA03004288A/es unknown
- 2001-11-14 WO PCT/US2001/043933 patent/WO2002039879A2/fr not_active Ceased
- 2001-11-14 EP EP01985480A patent/EP1341536A4/fr not_active Withdrawn
- 2001-11-14 CN CNA018220282A patent/CN1486183A/zh active Pending
2003
- 2003-05-06 ZA ZA200303471A patent/ZA200303471B/en unknown
- 2003-05-14 NO NO20032189A patent/NO20032189L/no unknown
- 2003-06-04 BG BG107874A patent/BG107874A/bg unknown

Also Published As

Publication number	Publication date
HUP0302436A2 (hu)	2003-11-28
JP2004513899A (ja)	2004-05-13
WO2002039879A3 (fr)	2002-07-25
PL361875A1 (en)	2004-10-04
CN1486183A (zh)	2004-03-31
CZ20031540A3 (cs)	2004-05-12
WO2002039879A2 (fr)	2002-05-23
BR0111982A (pt)	2003-10-28
US6528521B2 (en)	2003-03-04
IL155667A0 (en)	2003-11-23
CA2429047A1 (fr)	2002-05-23
US20020115683A1 (en)	2002-08-22
KR20030077538A (ko)	2003-10-01
BG107874A (bg)	2004-01-30
NO20032189L (no)	2003-07-08
EP1341536A4 (fr)	2007-08-01
NO20032189D0 (no)	2003-05-14
SK7422003A3 (en)	2004-01-08
MXPA03004288A (es)	2004-09-10
HUP0302436A3 (en)	2004-10-28
ZA200303471B (en)	2004-08-06
EP1341536A2 (fr)	2003-09-10

Publication	Publication Date	Title
US6506765B2 (en)	2003-01-14	Apomorphine derivatives and methods for their use
US6528521B2 (en)	2003-03-04	Treatment of anti-depression drug-induced sexual dysfunction with apomorphine
KR100719977B1 (ko)	2007-05-21	성기능 장애 치료를 위하여 효과 발현이 신속한 선택적 세로토닌 재흡수 억제제를 사용하는 방법
EP0767660A1 (fr)	1997-04-16	Procede et formulations servant a moduler la reaction sexuelle chez l'homme ou la femme
EP1397126B1 (fr)	2006-05-24	Utilisation du tramadol pour retarder l'ejaculation
US20020006933A1 (en)	2002-01-17	Method for treating sexual dysfunction with apomorphine at specified plasma concentration levels
AU749703B2 (en)	2002-07-04	Combination therapy for modulating the human sexual response
AU2002252361A1 (en)	2003-03-27	Method of delaying ejaculation
US20020086876A1 (en)	2002-07-04	Treatment of anti-depression drug-induced sexual dysfunction with apomorphine

Legal Events

Date	Code	Title	Description
2007-06-28	MK4	Application lapsed section 142(2)(d) - no continuation fee paid for the application