AU2001277712A1 - Avermectin derivatives - Google Patents

Avermectin derivatives

Info

Publication number: AU2001277712A1
Authority: AU; Australia
Prior art keywords: avermectin derivatives; avermectin; derivatives
Prior art date: 2000-08-09
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2001277712A

Inventor

Kenichiro Nagai

Satoshi Omura

Toshiaki Sunazuka

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Kitasato Institute

Original Assignee

Kitasato Institute

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-09

Filing date

2001-08-08

Publication date

2002-02-18

2001-08-08 Application filed by Kitasato Institute filed Critical Kitasato Institute

2002-02-18 Publication of AU2001277712A1 publication Critical patent/AU2001277712A1/en

Status Abandoned legal-status Critical Current

Links

RRZXIRBKKLTSOM-XPNPUAGNSA-N avermectin B1a Chemical class C1=C[C@H](C)[C@@H]([C@@H](C)CC)O[C@]11O[C@H](C\C=C(C)\[C@@H](O[C@@H]2O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C2)[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 RRZXIRBKKLTSOM-XPNPUAGNSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Tropical Medicine & Parasitology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

AU2001277712A 2000-08-09 2001-08-08 Avermectin derivatives Abandoned AU2001277712A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2000-240987		2000-08-09
JP2000240987		2000-08-09
PCT/JP2001/006802 WO2002012261A1 (en)	2000-08-09	2001-08-08	Avermectin derivatives

Publications (1)

Publication Number	Publication Date
AU2001277712A1 true AU2001277712A1 (en)	2002-02-18

Family

ID=18732257

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2001277712A Abandoned AU2001277712A1 (en)	2000-08-09	2001-08-08	Avermectin derivatives

Country Status (5)

Country	Link
US (1)	US7144866B2 (en)
JP (2)	JPWO2002012261A1 (en)
AU (1)	AU2001277712A1 (en)
CA (1)	CA2418968C (en)
WO (1)	WO2002012261A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0229804D0 (en) *	2002-12-20	2003-01-29	Syngenta Participations Ag	Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4200581A (en)	1978-08-04	1980-04-29	Merck & Co., Inc.	Alkyl derivatives of C-076 compounds
US4427663A (en) *	1982-03-16	1984-01-24	Merck & Co., Inc.	4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4833168A (en)	1986-10-03	1989-05-23	Merck & Co., Inc.	Avermectin reformatsky adducts
FR2619087B1 (en) *	1987-08-03	1990-03-23	Icp Sa	CORNER STRENGTHENING DEFLECTOR FOR GROUPING PACKAGING
US4895837A (en) *	1988-01-29	1990-01-23	Merck & Co., Inc.	Avermectin derivatives
US4906619A (en)	1988-07-22	1990-03-06	Merck & Co., Inc.	Alkyl avermectin derivatives
US5030622A (en) *	1989-06-02	1991-07-09	Merck & Co., Inc.	Avermectin derivatives
JP2888586B2 (en)	1990-03-05	1999-05-10	社団法人北里研究所	Microorganism for selective production of specific components of avermectin and its selective production method
US5169839A (en) *	1990-05-11	1992-12-08	Merck & Co., Inc.	Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
CA2052860A1 (en)	1990-10-11	1992-04-12	Thomas L. Shih	Avermectin degradation products and derivatives
US5208222A (en) *	1991-03-28	1993-05-04	Merck & Co., Inc.	4"-and 4'-alkylthio avermectin derivatives
US5229415A (en) *	1992-03-24	1993-07-20	Merck & Co., Inc.	Alkylthio alkyl avermectins are active antiparasitic agents
JPH0633273A (en)	1992-07-16	1994-02-08	Asahi Chem Ind Co Ltd	Rust preventive for metal part embedded in alc
GB9312154D0 (en) *	1993-06-12	1993-07-28	Pfizer Ltd	Antiparasitic agents
GB9316129D0 (en) *	1993-08-04	1993-09-22	Pfizer Ltd	Antiprasatic agents
US5437451A (en) *	1993-10-01	1995-08-01	Dd Stud, Inc.	Draw stud poker-type card game
GB9402916D0 (en)	1994-02-16	1994-04-06	Pfizer Ltd	Antiparasitic agents
US5897436A (en) *	1996-06-14	1999-04-27	Ptt, Llc	Modified poker card game
US6416407B1 (en) *	1998-11-16	2002-07-09	Travis Carrico	Multi-draw poker
NZ514026A (en) *	1999-02-09	2001-09-28	Kitasato Inst	A vermectin derivatives

2001
- 2001-08-08 JP JP2002518235A patent/JPWO2002012261A1/en active Pending
- 2001-08-08 US US10/343,980 patent/US7144866B2/en not_active Expired - Fee Related
- 2001-08-08 AU AU2001277712A patent/AU2001277712A1/en not_active Abandoned
- 2001-08-08 WO PCT/JP2001/006802 patent/WO2002012261A1/en not_active Ceased
- 2001-08-08 CA CA002418968A patent/CA2418968C/en not_active Expired - Fee Related
2012
- 2012-05-14 JP JP2012110510A patent/JP2012176971A/en active Pending

Also Published As

Publication number	Publication date
US20040018993A1 (en)	2004-01-29
JP2012176971A (en)	2012-09-13
CA2418968A1 (en)	2003-02-07
WO2002012261A1 (en)	2002-02-14
CA2418968C (en)	2009-11-24
US7144866B2 (en)	2006-12-05
JPWO2002012261A1 (en)	2004-01-15

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