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AU2001275115A1 - Methods for coupling benzoyl compounds and amino substituted bicyclic derivatives and enantiomerically pure or enriched compositions made therefrom - Google Patents

Methods for coupling benzoyl compounds and amino substituted bicyclic derivatives and enantiomerically pure or enriched compositions made therefrom

Info

Publication number
AU2001275115A1
AU2001275115A1 AU2001275115A AU7511501A AU2001275115A1 AU 2001275115 A1 AU2001275115 A1 AU 2001275115A1 AU 2001275115 A AU2001275115 A AU 2001275115A AU 7511501 A AU7511501 A AU 7511501A AU 2001275115 A1 AU2001275115 A1 AU 2001275115A1
Authority
AU
Australia
Prior art keywords
coupling
methods
enantiomerically pure
made therefrom
amino substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001275115A
Other languages
English (en)
Inventor
Luc Antoine
Alfio Borghese
Pascal Bouquel
Matthew Fisher
Hugo Gorissen
Joseph A. Jakubowski
Vien V. Khau
Michael Martinelli
Alain Merschaert
Michael Paal
Gerd Ruhter
Carine Rypens
Theo Schotten
Wolfgang Stenzel
Jean-Pierre Van Hoeck
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of AU2001275115A1 publication Critical patent/AU2001275115A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2001275115A 2000-06-02 2001-06-01 Methods for coupling benzoyl compounds and amino substituted bicyclic derivatives and enantiomerically pure or enriched compositions made therefrom Abandoned AU2001275115A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20876200P 2000-06-02 2000-06-02
US60208762 2000-06-02
PCT/US2001/017765 WO2001094333A2 (fr) 2000-06-02 2001-06-01 Procedes de couplage de composes de benzoyle et de derives bicycliques amino substitues, et compositions enantiomeriquement pures ou enrichies en etant faites

Publications (1)

Publication Number Publication Date
AU2001275115A1 true AU2001275115A1 (en) 2001-12-17

Family

ID=22775949

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001275115A Abandoned AU2001275115A1 (en) 2000-06-02 2001-06-01 Methods for coupling benzoyl compounds and amino substituted bicyclic derivatives and enantiomerically pure or enriched compositions made therefrom

Country Status (4)

Country Link
EP (1) EP1286982A2 (fr)
JP (1) JP2003535856A (fr)
AU (1) AU2001275115A1 (fr)
WO (1) WO2001094333A2 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104011012B (zh) * 2012-01-10 2016-01-20 伊莱利利公司 白三烯b4拮抗剂化合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5273982A (en) * 1990-03-09 1993-12-28 Hoffmann-La Roche Inc. Acetic acid derivatives
JPH08511538A (ja) * 1993-06-09 1996-12-03 スミスクライン・ビーチャム・コーポレイション 二環式フィブリノゲン拮抗物質
US5731324A (en) * 1993-07-22 1998-03-24 Eli Lilly And Company Glycoprotein IIb/IIIa antagonists
US6117910A (en) * 1994-12-13 2000-09-12 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists

Also Published As

Publication number Publication date
EP1286982A2 (fr) 2003-03-05
JP2003535856A (ja) 2003-12-02
WO2001094333A3 (fr) 2002-06-06
WO2001094333A2 (fr) 2001-12-13

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