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AU2001260406A1 - Antidiarrheal cannabinoid cb-1 receptor antagonist - Google Patents

Antidiarrheal cannabinoid cb-1 receptor antagonist

Info

Publication number
AU2001260406A1
AU2001260406A1 AU2001260406A AU6040601A AU2001260406A1 AU 2001260406 A1 AU2001260406 A1 AU 2001260406A1 AU 2001260406 A AU2001260406 A AU 2001260406A AU 6040601 A AU6040601 A AU 6040601A AU 2001260406 A1 AU2001260406 A1 AU 2001260406A1
Authority
AU
Australia
Prior art keywords
antidiarrheal
cannabinoid
receptor antagonist
antagonist
receptor
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001260406A
Other languages
English (en)
Inventor
Tiziano Croci
Luciano Manara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo SA filed Critical Sanofi Synthelabo SA
Publication of AU2001260406A1 publication Critical patent/AU2001260406A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2001260406A 2000-05-12 2001-05-11 Antidiarrheal cannabinoid cb-1 receptor antagonist Abandoned AU2001260406A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR00/06178 2000-05-12
FR0006178A FR2809621B1 (fr) 2000-05-12 2000-05-12 Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles comme antidiarrheiques
PCT/FR2001/001432 WO2001085092A2 (fr) 2000-05-12 2001-05-11 Antagoniste des recepteurs aux cannabinoides cb-1 antidiarrheique

Publications (1)

Publication Number Publication Date
AU2001260406A1 true AU2001260406A1 (en) 2001-11-20

Family

ID=8850242

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001260406A Abandoned AU2001260406A1 (en) 2000-05-12 2001-05-11 Antidiarrheal cannabinoid cb-1 receptor antagonist

Country Status (3)

Country Link
AU (1) AU2001260406A1 (fr)
FR (1) FR2809621B1 (fr)
WO (1) WO2001085092A2 (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ534757A (en) 2002-03-12 2006-07-28 Merck & Co Inc Substituted amides
CA2479618A1 (fr) 2002-03-26 2003-10-09 William K. Hagmann Amides spirocycliques en tant que modulateurs du recepteur cannabinoide
US7271266B2 (en) 2002-03-28 2007-09-18 Merck & Co., Inc. Substituted 2,3-diphenyl pyridines
WO2003086288A2 (fr) 2002-04-12 2003-10-23 Merck & Co., Inc. Amides bicycliques
US7129239B2 (en) 2002-10-28 2006-10-31 Pfizer Inc. Purine compounds and uses thereof
US7247628B2 (en) 2002-12-12 2007-07-24 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
KR100704097B1 (ko) * 2003-01-02 2007-04-06 에프. 호프만-라 로슈 아게 신규 cb 1 수용체 역작용제
US7329658B2 (en) 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7176210B2 (en) 2003-02-10 2007-02-13 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7141669B2 (en) 2003-04-23 2006-11-28 Pfizer Inc. Cannabiniod receptor ligands and uses thereof
US7268133B2 (en) 2003-04-23 2007-09-11 Pfizer, Inc. Patent Department Cannabinoid receptor ligands and uses thereof
US7145012B2 (en) 2003-04-23 2006-12-05 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7232823B2 (en) 2003-06-09 2007-06-19 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
EP1574211A1 (fr) 2004-03-09 2005-09-14 Inserm Utilisation d'antagonistes des récepteurs CB1 pour la fabrication d'un médicament destiné au traitement des maladies hépatiques
CA2586011C (fr) 2004-07-12 2011-07-19 Cadila Healthcare Limited Derives tricycliques de la pyrazole en tant que modulateurs de recepteurs cannabinoides
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
WO2007039797A1 (fr) * 2005-10-03 2007-04-12 Pfizer Products Inc. Utilisation d'antagonistes du recepteur cannabinoide de type 1 pour traiter les inflammations et l'arthrite

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2789079B3 (fr) * 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant

Also Published As

Publication number Publication date
FR2809621A1 (fr) 2001-12-07
WO2001085092A3 (fr) 2002-08-29
FR2809621B1 (fr) 2002-09-06
WO2001085092A2 (fr) 2001-11-15

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