AU2001260110A1 - Novel LHRH-antagonists, Production and Use Thereof as Medicament - Google Patents

Novel LHRH-antagonists, Production and Use Thereof as Medicament

Info

Publication number: AU2001260110A1
Authority: AU; Australia
Prior art keywords: antagonists; medicament; production; novel lhrh; lhrh
Prior art date: 1999-03-17
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001260110A

Other versions

AU2001260110B2 (en

Inventor

Thomas Beckers

Michael Bernd

Eckhard Gunther

Bernhard Kutscher

Thomas Reissmann

Peter Romeis

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Aeterna Zentaris GmbH

Original Assignee

Zentaris AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-03-17

Filing date

2001-03-12

Publication date

2001-12-06

2000-03-11 Priority claimed from PCT/EP2000/002165 external-priority patent/WO2000055190A1/en

2001-03-12 Application filed by Zentaris AG filed Critical Zentaris AG

2001-03-12 Priority claimed from PCT/EP2001/002719 external-priority patent/WO2001068676A2/en

2001-12-06 Publication of AU2001260110A1 publication Critical patent/AU2001260110A1/en

2004-09-30 Assigned to ZENTARIS GMBH reassignment ZENTARIS GMBH Request for Assignment Assignors: ZENTARIS AG

2005-05-05 Application granted granted Critical

2005-05-05 Publication of AU2001260110B2 publication Critical patent/AU2001260110B2/en

2020-03-11 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
DE19911771		1999-03-17
PCT/EP2000/002165 WO2000055190A1 (en)	1999-03-17	2000-03-11	Novel lhrh antagonists with improved solubility characteristics
AU32887/00A AU759442B2 (en)	1999-03-17	2000-03-11	Novel LHRH antagonists with improved solubility characteristics
US09/525,007 US6627609B1 (en)	1999-03-17	2000-03-14	LHRH antagonists having improved solubility properties
US09/525,007		2000-03-14
PCT/EP2001/002719 WO2001068676A2 (en)	2000-03-14	2001-03-12	Lhrh-antagonists, production and use thereof as medicament

Related Parent Applications (1)

Application Number	Title	Priority Date	Filing Date
AU32887/00A Division AU759442B2 (en)	1999-03-17	2000-03-11	Novel LHRH antagonists with improved solubility characteristics

Publications (2)

Publication Number	Publication Date
AU2001260110A1 true AU2001260110A1 (en)	2001-12-06
AU2001260110B2 AU2001260110B2 (en)	2005-05-05

Family

ID=24091545

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU6011001A Pending AU6011001A (en)	2000-03-14	2001-03-12	Novel lhrh-antagonists, production and use thereof as medicament
AU2001260110A Ceased AU2001260110B2 (en)	1999-03-17	2001-03-12	Novel LHRH-antagonists, production and use thereof as medicament

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AU6011001A Pending AU6011001A (en)	2000-03-14	2001-03-12	Novel lhrh-antagonists, production and use thereof as medicament

Country Status (25)

Country	Link
EP (1)	EP1268522B1 (en)
JP (1)	JP3805679B2 (en)
KR (1)	KR100607396B1 (en)
CN (2)	CN100500692C (en)
AT (1)	ATE408619T1 (en)
AU (2)	AU6011001A (en)
BG (1)	BG107121A (en)
BR (1)	BR0109279A (en)
CA (1)	CA2402193C (en)
DE (1)	DE50114335D1 (en)
DK (1)	DK1268522T3 (en)
ES (1)	ES2312435T3 (en)
HR (1)	HRP20020810A2 (en)
HU (1)	HUP0300222A3 (en)
IL (1)	IL151647A0 (en)
MX (1)	MXPA02008870A (en)
NO (1)	NO20024363L (en)
NZ (1)	NZ521273A (en)
PL (1)	PL357999A1 (en)
PT (1)	PT1268522E (en)
RU (1)	RU2248982C9 (en)
SK (1)	SK14332002A3 (en)
UA (1)	UA79070C2 (en)
WO (1)	WO2001068676A2 (en)
ZA (1)	ZA200207248B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN100340572C (en) *	2004-12-01	2007-10-03	中国人民解放军军事医学科学院毒物药物研究所	Novel LHRH antagonist
CN101037472B (en) *	2006-03-14	2013-03-27	中国人民解放军军事医学科学院毒物药物研究所	LHRH antagonist with low-histamine releasing function
ES2633453T3 (en)	2008-01-24	2017-09-21	Esperance Pharmaceuticals	Constructs of fusion of lithic domains and methods of preparation and use thereof
TWI442932B (en) *	2008-02-11	2014-07-01	Ferring Int Ct Sa	Method for treating prostate cancer with GnRH antagonist
CN101597321B (en) *	2008-06-03	2013-04-24	中国人民解放军军事医学科学院毒物药物研究所	LHRH antagonist with long-acting low-histamine release side effect
WO2010142060A1 (en) *	2009-06-11	2010-12-16	中国人民解放军军事医学科学院毒物药物研究所	Lhrh antagonist with long potency and low histamine releasing effect
IL238323B2 (en)	2012-10-30	2023-11-01	Esperance Pharmaceuticals Inc	Antibody/drug conjugates and methods of use
CN104418936B (en) *	2013-08-20	2018-06-05	中国人民解放军军事医学科学院毒物药物研究所	Lhrh antagonist derivative and its medicinal usage
FR3024612B1 (en) *	2014-08-04	2018-03-09	Alstom Transp Tech	POWER SUPPLY MODULE OF A MOTOR BLOCK, TRACTION SYSTEM AND ELECTRIC VEHICLE
RU2585367C1 (en) *	2014-11-05	2016-05-27	Наталья Владимировна Спиридонова	Method of treating infertility in females suffering from uterine myoma

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA862570B (en) *	1985-04-09	1986-12-30	Univ Tulane	Therapeutic decapeptides
US5140009A (en)	1988-02-10	1992-08-18	Tap Pharmaceuticals, Inc.	Octapeptide LHRH antagonists
US5300492A (en)	1988-02-10	1994-04-05	Tap Pharmaceuticals	LHRH analogs
US5110904A (en) *	1989-08-07	1992-05-05	Abbott Laboratories	Lhrh analogs
IL101074A (en)	1991-03-14	1997-09-30	Salk Inst For Biological Studi	GnRH ANALOGS AND THEIR PREPARATION
ES2052488T3 (en)	1991-04-25	1997-01-01	Romano Deghenghi	ANTAGONIST PEPTIDES OF THE LUTEINIZING HORMONE RELEASE HORMONE.
RU2043362C1 (en) *	1991-08-12	1995-09-10	Синтекс (Ю-Эс-Эй) Инк.	Method of solid-phase peptide synthesis
US5698522A (en)	1992-12-04	1997-12-16	Abbott Laboratories	6-position modified decapeptide LHRH antagonists
CA2136079A1 (en)	1992-12-18	1994-07-07	Fortuna Haviv	Lhrh antagonists having modified aminoacyl residues at positions 5 and 6
IL108509A0 (en)	1993-02-22	1994-05-30	Salk Inst For Biological Studi	GnRH antagonist peptides
DE4320201A1 (en) *	1993-06-18	1995-01-12	Asta Medica Ag	Use of Cetrorelix and other nona and decapeptides for the manufacture of a medicament for combating AIDS and for growth stimulation
DE19544212A1 (en) *	1995-11-28	1997-06-05	Asta Medica Ag	New LH-RH antagonists with improved effects
DE19911771B4 (en)	1999-03-17	2006-03-30	Zentaris Gmbh	LHRH antagonist, process for its preparation and its use

2001
- 2001-03-12 MX MXPA02008870A patent/MXPA02008870A/en active IP Right Grant
- 2001-03-12 DK DK01933682T patent/DK1268522T3/en active
- 2001-03-12 HR HRP20020810 patent/HRP20020810A2/en not_active Application Discontinuation
- 2001-03-12 EP EP01933682A patent/EP1268522B1/en not_active Expired - Lifetime
- 2001-03-12 CN CNB2006100817821A patent/CN100500692C/en not_active Expired - Fee Related
- 2001-03-12 CN CN01807543A patent/CN1443195A/en active Pending
- 2001-03-12 AU AU6011001A patent/AU6011001A/en active Pending
- 2001-03-12 KR KR1020027012059A patent/KR100607396B1/en not_active Expired - Lifetime
- 2001-03-12 PT PT01933682T patent/PT1268522E/en unknown
- 2001-03-12 IL IL15164701A patent/IL151647A0/en unknown
- 2001-03-12 RU RU2002127786/04A patent/RU2248982C9/en active
- 2001-03-12 JP JP2001567766A patent/JP3805679B2/en not_active Expired - Lifetime
- 2001-03-12 CA CA2402193A patent/CA2402193C/en not_active Expired - Lifetime
- 2001-03-12 PL PL01357999A patent/PL357999A1/en unknown
- 2001-03-12 BR BR0109279-0A patent/BR0109279A/en not_active IP Right Cessation
- 2001-03-12 AU AU2001260110A patent/AU2001260110B2/en not_active Ceased
- 2001-03-12 WO PCT/EP2001/002719 patent/WO2001068676A2/en not_active Ceased
- 2001-03-12 DE DE50114335T patent/DE50114335D1/en not_active Expired - Fee Related
- 2001-03-12 HU HU0300222A patent/HUP0300222A3/en unknown
- 2001-03-12 SK SK1433-2002A patent/SK14332002A3/en not_active Application Discontinuation
- 2001-03-12 ES ES01933682T patent/ES2312435T3/en not_active Expired - Lifetime
- 2001-03-12 AT AT01933682T patent/ATE408619T1/en not_active IP Right Cessation
- 2001-03-12 NZ NZ521273A patent/NZ521273A/en unknown
- 2001-12-03 UA UA2002108075A patent/UA79070C2/en unknown
2002
- 2002-09-10 ZA ZA200207248A patent/ZA200207248B/en unknown
- 2002-09-12 NO NO20024363A patent/NO20024363L/en not_active Application Discontinuation
- 2002-09-18 BG BG107121A patent/BG107121A/en unknown

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