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AU2000246281A1 - Piperidine compounds and process for providing such - Google Patents

Piperidine compounds and process for providing such

Info

Publication number
AU2000246281A1
AU2000246281A1 AU2000246281A AU4628100A AU2000246281A1 AU 2000246281 A1 AU2000246281 A1 AU 2000246281A1 AU 2000246281 A AU2000246281 A AU 2000246281A AU 4628100 A AU4628100 A AU 4628100A AU 2000246281 A1 AU2000246281 A1 AU 2000246281A1
Authority
AU
Australia
Prior art keywords
providing
piperidine compounds
paroxetine
piperidine
synthesis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2000246281A
Inventor
Jacobus Maria Lemmens
Theodorus Hendricus Antonius Peters
Pavel Slanina
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthon BV
Original Assignee
Synthon BV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=19760689&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2000246281(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Synthon BV filed Critical Synthon BV
Publication of AU2000246281A1 publication Critical patent/AU2000246281A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

The tosylate ester of the formula (6) and its salts, are convenient intermediates in the synthesis of paroxetine.
AU2000246281A 2000-05-12 2000-05-12 Piperidine compounds and process for providing such Abandoned AU2000246281A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/NL2000/000321 WO2001085689A1 (en) 2000-05-12 2000-05-12 Piperidine compounds and process for providing such

Publications (1)

Publication Number Publication Date
AU2000246281A1 true AU2000246281A1 (en) 2001-11-20

Family

ID=19760689

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2000246281A Abandoned AU2000246281A1 (en) 2000-05-12 2000-05-12 Piperidine compounds and process for providing such

Country Status (11)

Country Link
US (1) US20020099219A1 (en)
EP (1) EP1286965B1 (en)
AT (1) ATE257823T1 (en)
AU (1) AU2000246281A1 (en)
DE (1) DE60007782T2 (en)
DK (1) DK1286965T3 (en)
ES (1) ES2209876T3 (en)
NL (1) NL1016013C1 (en)
PT (1) PT1286965E (en)
SI (1) SI1286965T1 (en)
WO (1) WO2001085689A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1280775A1 (en) * 2000-05-12 2003-02-05 Synthon B.V. TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0190496A3 (en) * 1984-12-13 1987-05-27 Beecham Group Plc Piperidine derivatives having a gastro-intestinal activity
EP0812827B1 (en) * 1996-06-13 2009-09-02 Sumitomo Chemical Company, Limited Piperidine derivative as intermediates for the preparation of paroxetine and process for their preparation
HU221921B1 (en) * 1996-07-08 2003-02-28 Richter Gedeon Vegyészeti Gyár Rt. N-benzyl-piperidine or tetrahydro-pyridine derivatives and processes for producing them
SK283394B6 (en) * 1997-06-10 2003-07-01 Synthon B. V. 4-phenylpiperidine compounds and its pharmaceutically acceptable salts, process for their preparation, medicament containing them and their use
JP2000095780A (en) * 1998-09-22 2000-04-04 Asahi Glass Co Ltd Method for producing carbamate crystals

Also Published As

Publication number Publication date
PT1286965E (en) 2004-04-30
WO2001085689A1 (en) 2001-11-15
NL1016013C1 (en) 2001-01-30
SI1286965T1 (en) 2004-04-30
EP1286965A1 (en) 2003-03-05
ATE257823T1 (en) 2004-01-15
DE60007782T2 (en) 2004-12-09
US20020099219A1 (en) 2002-07-25
ES2209876T3 (en) 2004-07-01
EP1286965B1 (en) 2004-01-14
DE60007782D1 (en) 2004-02-19
DK1286965T3 (en) 2004-05-03

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