AR107680A1 - Derivados de heterociclos bicíclicos condensados como pesticidas - Google Patents
Derivados de heterociclos bicíclicos condensados como pesticidasInfo
- Publication number
- AR107680A1 AR107680A1 ARP170100427A ARP170100427A AR107680A1 AR 107680 A1 AR107680 A1 AR 107680A1 AR P170100427 A ARP170100427 A AR P170100427A AR P170100427 A ARP170100427 A AR P170100427A AR 107680 A1 AR107680 A1 AR 107680A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- alkoxy
- cycloalkyl
- alkylsulfinyl
- alkylsulfonyl
- Prior art date
Links
- 239000000575 pesticide Substances 0.000 title 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 55
- -1 C2−6 cyanoalkenyl Chemical group 0.000 abstract 18
- 125000004670 alkyl amino thio carbonyl group Chemical group 0.000 abstract 10
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 9
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 7
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 7
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 6
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 6
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 6
- 125000005089 alkenylaminocarbonyl group Chemical group 0.000 abstract 6
- 229910052736 halogen Inorganic materials 0.000 abstract 6
- 125000001072 heteroaryl group Chemical group 0.000 abstract 6
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 5
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 abstract 5
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 5
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 5
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 abstract 5
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 5
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 5
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 5
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 5
- 150000002367 halogens Chemical class 0.000 abstract 5
- 125000000623 heterocyclic group Chemical group 0.000 abstract 5
- 229910052757 nitrogen Inorganic materials 0.000 abstract 5
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 abstract 4
- 125000004845 (C1-C6) alkylsulfonylamino group Chemical group 0.000 abstract 4
- 125000006642 (C1-C6) cyanoalkyl group Chemical group 0.000 abstract 4
- 125000006577 C1-C6 hydroxyalkyl group Chemical group 0.000 abstract 4
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 4
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 abstract 4
- 125000003118 aryl group Chemical group 0.000 abstract 4
- 125000006310 cycloalkyl amino group Chemical group 0.000 abstract 4
- 125000004844 (C1-C6) alkoxyimino group Chemical group 0.000 abstract 3
- 125000004750 (C1-C6) alkylaminosulfonyl group Chemical group 0.000 abstract 3
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 abstract 3
- 125000005947 C1-C6 alkylsulfonyloxy group Chemical group 0.000 abstract 3
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000005103 alkyl silyl group Chemical group 0.000 abstract 3
- 125000004682 aminothiocarbonyl group Chemical group NC(=S)* 0.000 abstract 3
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 3
- 125000005159 cyanoalkoxy group Chemical group 0.000 abstract 3
- 125000005167 cycloalkylaminocarbonyl group Chemical group 0.000 abstract 3
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 3
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 3
- 125000001424 substituent group Chemical group 0.000 abstract 3
- ZMZDMBWJUHKJPS-UHFFFAOYSA-N thiocyanic acid Chemical compound SC#N ZMZDMBWJUHKJPS-UHFFFAOYSA-N 0.000 abstract 3
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 abstract 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 abstract 2
- 125000004691 alkyl thio carbonyl group Chemical group 0.000 abstract 2
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 125000004122 cyclic group Chemical group 0.000 abstract 2
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000004665 trialkylsilyl group Chemical group 0.000 abstract 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 1
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 1
- 241000607479 Yersinia pestis Species 0.000 abstract 1
- 230000000895 acaricidal effect Effects 0.000 abstract 1
- 239000000642 acaricide Substances 0.000 abstract 1
- 125000004471 alkyl aminosulfonyl group Chemical group 0.000 abstract 1
- 125000006615 aromatic heterocyclic group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000002619 bicyclic group Chemical group 0.000 abstract 1
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
- 239000002917 insecticide Substances 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
- A01N43/52—1,3-Diazoles; Hydrogenated 1,3-diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Su uso como acaricidas y/o insecticidas para el control de plagas animales. Reivindicación 1: Compuestos de la fórmula (1), en donde Aa es nitrógeno o =C(H)-; Ab es nitrógeno o =C(H)-; Ac es nitrógeno o =C(H)-; Ad es nitrógeno o =C(H)-, donde Aa, Ab, Ac y Ad no pueden ser simultáneamente todos nitrógeno; R¹ es C₁₋₆ alquilo, C₁₋₆ haloalquilo, C₁₋₆ cianoalquilo, C₁₋₆ hidroxialquilo, C₁₋₆ alcoxi-C₁₋₆ alquilo, C₁₋₆ haloalcoxi-C₁₋₆ alquilo, C₂₋₆ alquenilo, C₂₋₆ alqueniloxi-C₁₋₆ alquilo, C₂₋₆ haloalqueniloxi-C₁₋₆ alquilo, C₁₋₆ haloalquenilo, C₂₋₆ cianoalquenilo, C₂₋₆ alquinilo, C₂₋₆ alquiniloxi-C₁₋₆ alquilo, C₂₋₆ haloalquiniloxi-C₁₋₆ alquilo, C₂₋₆ haloalquinilo, C₂₋₆ cianoalquinilo, C₃₋₈ cicloalquilo, C₃₋₈ cicloalquilo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo-C₃₋₈ cicloalquilo, halo-C₃₋₈ cicloalquilo, amino, C₁₋₆ alquilamino, di-C₁₋₆ alquilo-amino, C₃₋₈ cicloalquilamino, C₁₋₆ alquilcarbonilo-amino, C₁₋₆ alquiltio-C₁₋₆ alquilo, C₁₋₆ haloalquiltio-C₁₋₆ alquilo, C₁₋₆ alquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ haloalquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ haloalquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquiltio-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ alquilcarbonilo-C₁₋₆ alquilo, C₁₋₆ haloalquilcarbonilo-C₁₋₆ alquilo, C₁₋₆ alcoxicarbonilo-C₁₋₆ alquilo, C₁₋₆ haloalcoxicarbonilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfonilamino, aminosulfonilo-C₁₋₆ alquilo, C₁₋₆ alquilaminosulfonilo-C₁₋₆ alquilo, di-C₁₋₆ alquilo-aminosulfonilo-C₁₋₆ alquilo, o C₁₋₆ alquilo, C₁₋₆ alcoxi, C₂₋₆ alquenilo, C₂₋₆ alquinilo, C₃₋₈ cicloalquilo cada uno opcionalmente mono- o polisustituido de manera idéntica o diferente con arilo, hetarilo o heterociclilo, donde arilo, hetarilo o heterociclilo puede estar cada uno opcionalmente mono- o polisustituido de manera idéntica o diferente con halógeno, ciano, nitro, hidroxi, amino, carboxi, carbamoil, aminosulfonilo, C₁₋₆ alquilo, C₃₋₆ cicloalquilo, C₁₋₆ alcoxi, C₁₋₆ haloalquilo, C₁₋₆ haloalcoxi, C₁₋₆ alquiltio, C₁₋₆ alquilsulfinilo, C₁₋₆ alquilsulfonilo, C₁₋₆ alquilsulfimino, C₁₋₆ alquilsulfimino-C₁₋₆ alquilo, C₁₋₆ alquilsulfimino-C₂₋₆ alquilcarbonilo, C₁₋₆ alquilsulfoximino, C₁₋₆ alquilsulfoximino-C₁₋₆ alquilo, C₁₋₆ alquilsulfoximino-C₂₋₆ alquilcarbonilo, C₁₋₆ alcoxicarbonilo, C₁₋₆ alquilcarbonilo, C₃₋₆ trialquilsililo o bencilo, o R¹ es arilo, hetarilo o heterociclilo, cada uno opcionalmente mono- o polisustituido de manera idéntica o diferente con halógeno, ciano, nitro, hidroxi, amino, carboxi, carbamoil, C₁₋₆ alquilo, C₃₋₈ cicloalquilo, C₁₋₆ alcoxi, C₁₋₆ haloalquilo, C₁₋₆ haloalcoxi, C₁₋₆ alquiltio, C₁₋₆ alquilsulfinilo, C₁₋₆ alquilsulfonilo, C₁₋₆ alquilsulfimino, C₁₋₆ alquilsulfimino-C₁₋₆ alquilo, C₁₋₆ alquilsulfimino-C₂₋₆ alquilcarbonilo, C₁₋₆ alquilsulfoximino, C₁₋₆ alquilsulfoximino-C₁₋₆ alquilo, C₁₋₆ alquilsulfoximino-C₂₋₆ alquilcarbonilo, C₁₋₆ alcoxicarbonilo, C₁₋₆ alquilcarbonilo, C₃₋₆ trialquilsililo, (=O) (en el caso de heterociclilo solamente) o (=O)₂ (en el caso de heterociclilo solamente); R², R³ son en forma independiente hidrógeno, ciano, halógeno, nitro, acetilo, hidroxi, amino, SCN, tri-C₁₋₆ alquilsililo, C₃₋₈ cicloalquilo, C₃₋₈ cicloalquilo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo-C₃₋₈ cicloalquilo, halo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo, C₁₋₆ haloalquilo, C₁₋₆ cianoalquilo, C₁₋₆ hidroxialquilo, hidroxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquilo, C₂₋₆ alquenilo, C₂₋₆ haloalquenilo, C₂₋₆ cianoalquenilo, C₂₋₆ alquinilo, C₂₋₆ haloalquinilo, C₂₋₆ cianoalquinilo, C₁₋₆ alcoxi, C₁₋₆ haloalcoxi, C₁₋₆ cianoalcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxi-C₁₋₆ alcoxi, C₁₋₆ alquilhidroxiimino, C₁₋₆ alcoxiimino, C₁₋₆ alquilo-C₁₋₆ alcoxiimino, C₁₋₆ haloalquilo-C₁₋₆ alcoxiimino, C₁₋₆ alquiltio, C₁₋₆ haloalquiltio, C₁₋₆ alcoxi-C₁₋₆ alquiltio, C₁₋₆ alquiltio-C₁₋₆ alquilo, C₁₋₆ alquilsulfinilo, C₁₋₆ haloalquilsulfinilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfinilo, C₁₋₆ alquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfonilo, C₁₋₆ haloalquilsulfonilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfonilo, C₁₋₆ alquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfoniloxi, C₁₋₆ alquilcarbonilo, C₁₋₆ alquiltiocarbonilo, C₁₋₆ haloalquilcarbonilo, C₁₋₆ alquilcarboniloxi, C₁₋₆ alcoxicarbonilo, C₁₋₆ haloalcoxicarbonilo, aminocarbonilo, C₁₋₆ alquilaminocarbonilo, C₁₋₆ alquilaminotiocarbonilo, di-C₁₋₆ alquilo-aminocarbonilo, di-C₁₋₆ alquilo-aminotiocarbonilo, C₂₋₆ alquenilaminocarbonilo, di-C₂₋₆ alquenilaminocarbonilo, C₃₋₈ cicloalquilaminocarbonilo, C₁₋₆ alquilsulfonilamino, C₁₋₆ alquilamino, di-C₁₋₆ alquilamino, aminosulfonilo, C₁₋₆ alquilaminosulfonilo, di-C₁₋₆ alquilo-aminosulfonilo, C₁₋₆ alquilsulfoximino, aminotiocarbonilo, C₁₋₆ alquilaminotiocarbonilo, di-C₁₋₆ alquilo-aminotiocarbonilo, C₃₋₈ cicloalquilamino, NHCO-C₁₋₆ alquilo (C₁₋₆ alquilcarboniloamino), es arilo, hetarilo o heterociclilo, cada uno opcionalmente mono- o polisustituido de manera idéntica o diferente, donde (en el caso de hetarilo) al menos un grupo carbonilo puede estar presente opcionalmente y/o donde como sustituyentes se pueden considerar en cada caso: ciano, carboxil, halógeno, nitro, acetilo, hidroxi, amino, SCN, tri-C₁₋₆ alquilsililo, C₃₋₈ cicloalquilo, C₃₋₈ cicloalquilo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo-C₃₋₈ cicloalquilo, halo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo, C₁₋₆ haloalquilo, C₁₋₆ cianoalquilo, C₁₋₆ hidroxialquilo, hidroxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquilo, C₂₋₆ alquenilo, C₂₋₆ haloalquenilo, C₂₋₆ cianoalquenilo, C₂₋₆ alquinilo, C₂₋₆ haloalquinilo, C₂₋₆ cianoalquinilo, C₁₋₆ alcoxi, C₁₋₆ haloalcoxi, C₁₋₆ cianoalcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxi-C₁₋₆ alcoxi, C₁₋₆ alquilhidroxiimino, C₁₋₆ alcoxiimino, C₁₋₆ alquilo-C₁₋₆ alcoxiimino, C₁₋₆ haloalquilo-C₁₋₆ alcoxiimino, C₁₋₆ alquiltio, C₁₋₆ haloalquiltio, C₁₋₆ alcoxi-C₁₋₆ alquiltio, C₁₋₆ alquiltio-C₁₋₆ alquilo, C₁₋₆ alquilsulfinilo C₁₋₆ alcoxi-C₁₋₆ alquilsulfinilo, C₁₋₆ alquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfonilo, C₁₋₆ haloalquilsulfonilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfonilo, C₁₋₆ alquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfoniloxi, C₁₋₆ alquilcarbonilo, C₁₋₆ haloalquilcarbonilo, C₁₋₆ alquilcarboniloxi, C₁₋₆ alcoxicarbonilo, C₁₋₆ haloalcoxicarbonilo, aminocarbonilo, C₁₋₆ alquilaminocarbonilo, di-C₁₋₆ alquilo-aminocarbonilo, C₂₋₆ alquenilaminocarbonilo, di-C₂₋₆ alquenilaminocarbonilo, C₃₋₈ cicloalquilaminocarbonilo, C₁₋₆ alquilsulfonilamino, C₁₋₆ alquilamino, di-C₁₋₆ alquilamino, aminosulfonilo, C₁₋₆ alquilaminosulfonilo, di-C₁₋₆ alquilaminosulfonilo, C₁₋₆ alquilsulfoximino, aminotiocarbonilo, C₁₋₆ alquilaminotiocarbonilo, di-C₁₋₆ alquilaminotiocarbonilo, C₃₋₈ cicloalquilamino, C₁₋₆ alquilcarboniloamino; Q es un sistema de anillos bicíclicos o tricíclicos fusionados de 8, 9, 10, 11 ó 12 miembros heterocíclicos o heteroaromáticos saturados o parcialmente saturados, donde al menos un grupo carbonilo puede estar presente opcionalmente y/o donde el sistema de anillos puede estar opcionalmente mono- o polisustituido de manera idéntica o diferente, y donde los sustituyentes pueden seleccionarse de manera independiente entre ciano, halógeno, nitro, acetilo, hidroxi, amino, SCN, tri-C₁₋₆ alquilsililo, C₃₋₈ cicloalquilo, C₃₋₈ cicloalquilo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo-C₃₋₈ cicloalquilo, halo-C₃₋₈ cicloalquilo, C₁₋₆ alquilo, C₁₋₆ haloalquilo, C₁₋₆ cianoalquilo, C₁₋₆ hidroxialquilo, hidroxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alquilo, C₁₋₆ alcoxi-C₁₋₆ alquilo, C₂₋₆ alquenilo, C₂₋₆ haloalquenilo, C₂₋₆ cianoalquenilo, C₂₋₆ alquinilo, C₂₋₆ alquiniloxi-C₁₋₄ alquilo, C₂₋₆ haloalquinilo, C₂₋₆ cianoalquinilo, C₁₋₆ alcoxi, C₁₋₆ haloalcoxi, C₁₋₆ haloalcoxi-C₁₋₆ alquilo, C₂₋₆ alqueniloxi-C₁₋₆ alquilo, C₂₋₆ haloalqueniloxi-C₁₋₆ alquilo, C₁₋₆ cianoalcoxi, C₁₋₆ alcoxicarbonilo-C₁₋₆ alcoxi, C₁₋₆ alcoxi-C₁₋₆ alcoxi, C₁₋₆ alquilhidroxiimino, C₁₋₆ alcoxiimino, C₁₋₆ alquilo-C₁₋₆ alcoxiimino, C₁₋₆ haloalquilo-C₁₋₆ alcoxiimino, C₁₋₆ alquiltio, C₁₋₆ haloalquiltio, C₁₋₆ alcoxi-C₁₋₆ alquiltio, C₁₋₆ alquiltio-C₁₋₆ alquilo, C₁₋₆ alquilsulfinilo, C₁₋₆ haloalquilsulfinilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfinilo, C₁₋₆ alquilsulfinilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfonilo, C₁₋₆ haloalquilsulfonilo, C₁₋₆ alcoxi-C₁₋₆ alquilsulfonilo, C₁₋₆ alquilsulfonilo-C₁₋₆ alquilo, C₁₋₆ alquilsulfoniloxi, C₁₋₆ alquilcarbonilo, C₁₋₆ alquilcarbonilo-C₁₋₆ alquilo, C₁₋₆ alquiltiocarbonilo, C₁₋₆ haloalquilcarbonilo, C₁₋₆ alquilcarboniloxi, C₁₋₆ alcoxicarbonilo, C₁₋₆ haloalcoxicarbonilo, aminocarbonilo, C₁₋₆ alquilaminocarbonilo, C₁₋₆ alquilaminotiocarbonilo, di-C₁₋₆ alquilo-aminocarbonilo, di-C₁₋₆ alquilo-aminotiocarbonilo, C₂₋₆ alquenilaminocarbonilo, di-C₂₋₆ alquenilaminocarbonilo, C₃₋₈ cicloalquilaminocarbonilo, C₁₋₆ alquilsulfonilamino, C₁₋₆ alquilamino, di-C₁₋₆ alquilamino, aminosulfonilo, C₁₋₆ alquilaminosulfonilo, di-C₁₋₆ alquilo-aminosulfonilo, C₁₋₆ alquilsulfoximino, aminotiocarbonilo, C₁₋₆ alquilaminotiocarbonilo, di-C₁₋₆ alquilo-aminotiocarbonilo, C₃₋₈ cicloalquilamino, NHCO-C₁₋₆ alquilo (C₁₋₆ alquilcarboniloamino), o donde los sustituyentes pueden seleccionarse de manera independiente entre fenilo o un anillo heteroaromático de 5 ó 6 miembros, donde fenilo o el anillo puede estar opcionalmente mono- o polisustituido de manera idéntica o diferente con C₁₋₆ alquilo, C₂₋₆ alquenilo, C₂₋₆ alquinilo, C₃₋₆ cicloalquilo, C₁₋₆ haloalquilo, C₂₋₆ haloalquenilo, C₂₋₆ haloalquinilo, C₃₋₆ halocicloalquilo, halógeno, CN, NO₂, C₁₋₄ alcoxi, C₁₋₄ haloalcoxi; n es 0, 1 ó 2; salvo los compuestos de fórmula (2), y (3).
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-
2017
- 2017-02-16 WO PCT/EP2017/053475 patent/WO2017144341A1/de not_active Ceased
- 2017-02-21 AR ARP170100427A patent/AR107680A1/es unknown
- 2017-02-21 TW TW106105673A patent/TW201741310A/zh unknown
- 2017-02-23 UY UY0001037136A patent/UY37136A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| UY37136A (es) | 2017-09-29 |
| WO2017144341A1 (de) | 2017-08-31 |
| TW201741310A (zh) | 2017-12-01 |
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