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AR051778A2 - Derivados del acido dimetilaminocrotonico y procesos para supreparacion - Google Patents

Derivados del acido dimetilaminocrotonico y procesos para supreparacion

Info

Publication number
AR051778A2
AR051778A2 ARP050104937A ARP050104937A AR051778A2 AR 051778 A2 AR051778 A2 AR 051778A2 AR P050104937 A ARP050104937 A AR P050104937A AR P050104937 A ARP050104937 A AR P050104937A AR 051778 A2 AR051778 A2 AR 051778A2
Authority
AR
Argentina
Prior art keywords
supreparation
derivatives
processes
dimethylaminocrotonic acid
dimethylaminocrotonic
Prior art date
Application number
ARP050104937A
Other languages
English (en)
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of AR051778A2 publication Critical patent/AR051778A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4706—4-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/30—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/16—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and unsaturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • External Artificial Organs (AREA)

Abstract

Reivindicacion 1: Un compuesto de formula (1) (CH3)2NCH2=(O)-OH o una sal HCl del mismo. Reivindicacion 2: El compuesto de acuerdo con la reivindicacion 1, donde el compuesto es la sal HCl del mismo.
ARP050104937A 2001-08-07 2005-11-25 Derivados del acido dimetilaminocrotonico y procesos para supreparacion AR051778A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31064601P 2001-08-07 2001-08-07

Publications (1)

Publication Number Publication Date
AR051778A2 true AR051778A2 (es) 2007-02-07

Family

ID=23203475

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP020102977A AR036250A1 (es) 2001-08-07 2002-08-06 Una combinacion antineoplasica, un producto que la comprende y el uso de dicha combinacion para la fabricacion de un medicamento para el tratamiento de un neoplasma en un mamifero
ARP050104937A AR051778A2 (es) 2001-08-07 2005-11-25 Derivados del acido dimetilaminocrotonico y procesos para supreparacion

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP020102977A AR036250A1 (es) 2001-08-07 2002-08-06 Una combinacion antineoplasica, un producto que la comprende y el uso de dicha combinacion para la fabricacion de un medicamento para el tratamiento de un neoplasma en un mamifero

Country Status (26)

Country Link
US (4) US6617333B2 (es)
EP (2) EP1414438B1 (es)
JP (2) JP2005505549A (es)
KR (1) KR20040029406A (es)
CN (3) CN100415753C (es)
AR (2) AR036250A1 (es)
AT (1) ATE314069T1 (es)
AU (2) AU2002330994B2 (es)
BR (1) BR0211769A (es)
CA (1) CA2455126A1 (es)
CY (1) CY1104983T1 (es)
DE (1) DE60208385T2 (es)
DK (1) DK1414438T3 (es)
EA (2) EA006226B1 (es)
ES (1) ES2252512T3 (es)
HU (1) HUP0401089A3 (es)
IL (2) IL159859A0 (es)
MX (1) MXPA04001118A (es)
NO (2) NO325503B1 (es)
NZ (3) NZ530847A (es)
PL (1) PL368303A1 (es)
SG (1) SG170612A1 (es)
TW (2) TWI300351B (es)
UA (1) UA77200C2 (es)
WO (1) WO2003020266A1 (es)
ZA (1) ZA200401801B (es)

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NO20040558L (no) 2004-02-06
AR036250A1 (es) 2004-08-25
CN1326523C (zh) 2007-07-18
DE60208385D1 (de) 2006-02-02
EP1414438A1 (en) 2004-05-06
IL159859A0 (en) 2004-06-20
NO20073801L (no) 2004-02-06
CA2455126A1 (en) 2003-03-13
ZA200401801B (en) 2005-06-06
EA006226B1 (ru) 2005-10-27
NO325503B1 (no) 2008-05-26
CY1104983T1 (el) 2010-03-03
MXPA04001118A (es) 2004-05-20
PL368303A1 (en) 2005-03-21
TWI300351B (en) 2008-09-01
HK1061204A1 (en) 2004-09-10
CN1803806A (zh) 2006-07-19
IL159859A (en) 2009-12-24
JP2010155845A (ja) 2010-07-15
US20030050222A1 (en) 2003-03-13
USRE41084E1 (en) 2010-01-19
CN100415753C (zh) 2008-09-03
HUP0401089A3 (en) 2007-12-28
AU2002330994B2 (en) 2007-10-04
NZ542272A (en) 2007-12-21
USRE41253E1 (en) 2010-04-20
EA200501251A1 (ru) 2008-12-30
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WO2003020266A1 (en) 2003-03-13
BR0211769A (pt) 2004-07-27
SG170612A1 (en) 2011-05-30
TWI305527B (en) 2009-01-21
EA011098B1 (ru) 2008-12-30
JP2005505549A (ja) 2005-02-24
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HUP0401089A2 (hu) 2004-09-28
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EP1414438B1 (en) 2005-12-28
EA200400284A1 (ru) 2004-06-24
DK1414438T3 (da) 2006-03-27
UA77200C2 (en) 2006-11-15
USRE40418E1 (en) 2008-07-01
DE60208385T2 (de) 2006-08-03
US6617333B2 (en) 2003-09-09
KR20040029406A (ko) 2004-04-06
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CN1538842A (zh) 2004-10-20

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