AR057992A1 - BENZOILUREA COMPOUND AND USE OF THE SAME - Google Patents
BENZOILUREA COMPOUND AND USE OF THE SAMEInfo
- Publication number
- AR057992A1 AR057992A1 ARP060105381A ARP060105381A AR057992A1 AR 057992 A1 AR057992 A1 AR 057992A1 AR P060105381 A ARP060105381 A AR P060105381A AR P060105381 A ARP060105381 A AR P060105381A AR 057992 A1 AR057992 A1 AR 057992A1
- Authority
- AR
- Argentina
- Prior art keywords
- optionally substituted
- group optionally
- substituents
- group
- halogen atoms
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 125000001424 substituent group Chemical group 0.000 abstract 53
- 125000005843 halogen group Chemical group 0.000 abstract 28
- 125000000217 alkyl group Chemical group 0.000 abstract 15
- 125000003118 aryl group Chemical group 0.000 abstract 9
- 125000003545 alkoxy group Chemical group 0.000 abstract 7
- 125000003342 alkenyl group Chemical group 0.000 abstract 4
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 4
- 125000000304 alkynyl group Chemical group 0.000 abstract 4
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 4
- -1 benzoylurea compound Chemical class 0.000 abstract 4
- 125000000623 heterocyclic group Chemical group 0.000 abstract 4
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 3
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 3
- 125000004414 alkyl thio group Chemical group 0.000 abstract 3
- 125000004429 atom Chemical group 0.000 abstract 3
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 3
- 229910052757 nitrogen Inorganic materials 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- 125000004434 sulfur atom Chemical group 0.000 abstract 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 2
- 125000003277 amino group Chemical group 0.000 abstract 2
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 abstract 2
- 125000005098 aryl alkoxy carbonyl group Chemical group 0.000 abstract 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 2
- 125000003341 7 membered heterocyclic group Chemical group 0.000 abstract 1
- 125000005236 alkanoylamino group Chemical group 0.000 abstract 1
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 1
- 125000005136 alkenylsulfinyl group Chemical group 0.000 abstract 1
- 125000005137 alkenylsulfonyl group Chemical group 0.000 abstract 1
- 125000005108 alkenylthio group Chemical group 0.000 abstract 1
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 1
- 125000005139 alkynylsulfonyl group Chemical group 0.000 abstract 1
- 125000005109 alkynylthio group Chemical group 0.000 abstract 1
- 125000005127 aryl alkoxy alkyl group Chemical group 0.000 abstract 1
- 125000002102 aryl alkyloxo group Chemical group 0.000 abstract 1
- 125000005116 aryl carbamoyl group Chemical group 0.000 abstract 1
- 125000005160 aryl oxy alkyl group Chemical group 0.000 abstract 1
- 125000005161 aryl oxy carbonyl group Chemical group 0.000 abstract 1
- 125000004391 aryl sulfonyl group Chemical group 0.000 abstract 1
- 125000004104 aryloxy group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 239000000470 constituent Substances 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/34—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the groups, e.g. biuret; Thio analogues thereof; Urea-aldehyde condensation products
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/46—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
- C07C275/48—Y being a hydrogen or a carbon atom
- C07C275/54—Y being a carbon atom of a six-membered aromatic ring, e.g. benzoylureas
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D309/10—Oxygen atoms
- C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Reivindicacion 1: Un compuesto benzoilurea caracterizado por que está representado por la formula (1), en donde X e Y cada uno representa independientemente un átomo de oxígeno o un átomo de azufre, R1 representa un átomo de hidrogeno, un grupo formilo, un grupo ciano, un grupo alquilsulfonilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilsulfonilo opcionalmente sustituido con uno o más sustituyentes, un grupo alquilcarboniltio inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alcoxicarboniltio inferior opcionalmente sustituido con uno o más sustituyentes, un grupo ariloxicarboniltio sustituido con uno o más sustituyentes, un grupo mono o di (alquilo inferior) aminosulfonilo opcionalmente sustituido con uno o más sustituyentes, un grupo mono o di(aril)aminosulfonilo opcionalmente. sustituido con uno o más sustituyentes, un grupo alquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquenilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquinilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo cicloalquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilalquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilo opcionalmente sustituido con uno o más sustituyentes, un grupo alcoxilo inferior alquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo ariloxialquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquiltio inferior alquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquilsulfinilo inferior alquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquilsulfonilo inferior alquilo inferior opcionalmente sustituido, con uno o más sustituyentes, un grupo mono o di (alquilo inferior)amino alquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alcanoilo inferior sustituido con uno o más sustituyentes, un grupo alcoxicarbonilo inferior sustituido con uno o más sustituyentes, un grupo ariloxicarbonilo sustituido con uno o más sustituyentes, un grupo arilalcoxicarbonilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo carbamoilo opcionalmente sustituido con uno o más sustituyentes, un grupo tiocarbamoilo opcionalmente sustituido con uno o más sustituyentes, un grupo alcoxioxalquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilalcoxialquilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo ariloxioxalilo opcionalmente sustituido con uno o más sustituyentes, un grupo aminooxalilo opcionalmente sustituido con uno o más sustituyentes, un grupo alcoxilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo ariloxilo opcionalmente sustituido con uno o más sustituyentes, un grupo arilalcoxilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo amino opcionalmente sustituido con uno o más sustituyentes, o un grupo, heterocíclico opcionalmente sustituido con uno o más sustituyentes, R2 representa un grupo alquileno inferior opcionalmente sustituido con uno o más átomos halogenos, A representa, (a) un grupo representado por OR3, (en donde R3 es un grupo alquilo C1-3 sustituido con uno o más substituyentes, representa opcionalmente, un grupo alquenilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquinilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alcanoilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilo opcionalmente sustituido con uno o más sustituyentes, o un grupo arilalquilo inferior opcionalmente sustituido con uno o más sustituyentes), (b) un grupo representado por S(O)nR4, (en donde R4 representa un grupo alquilo C1-3 opcionalmente sustituido con uno o más sustituyentes, un grupo alquenilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquinilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilo opcionalmente sustituido con uno o más sustituyentes, o un grupo arilalquilo inferior opcionalmente sustituido con uno o más sustituyentes, y n representa un entero de 0, 1 o 2), o (c) un grupo representado por NR5R6, (en donde R5 y R6 cada uno representa independientemente un grupo alquilo C1-3 opcionalmente sustituido con uno o más sustituyentes, un grupo alquenilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo alquinilo inferior opcionalmente sustituido con uno o más sustituyentes, un grupo arilo opcionalmente sustituido con uno o más sustituyentes, un grupo arilalquilo inferior opcionalmente sustituido con uno o más sustituyentes, o R5 y R6 pueden enlazarse en los extremos de los mismos para formar junto con el átomo de nitrogeno un anillo heterocíclico de 3 a 7 miembros conteniendo nitrogeno que opcionalmente posee otro átomo de nitrogeno, un átomo de oxígeno o un átomo de azufre como átomo constituyente del anillo), R7 representa un átomo halogeno, un grupo nitro, un grupo ciano, un grupo arilalcoxilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alcanoilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alcoxicarbonilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo arilo opcionalmente sustituido con uno o más átomos halogenos, un grupo arilalcoxicarbonilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo arilcarbamoilo opcionalmente sustituido con uno o más., átomos halogenos, un grupo carbamoilo opcionalmente sustituido con uno o más grupo alquilo inferior, un grupo tiocarbamoilo opcionalmente sustituido con uno o grupos alquilo inferior, un grupo amino opcionalmente sustituido con uno o más grupos alquilo inferior, un grupo alquilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alcoxilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alcoxilo inferior alcoxilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alqueniloxilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquiniloxilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alcanoilamino inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquiltio inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alqueniltio inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquiniltio inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquilsulfinilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquenilsulfinilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquinilsulfinilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquilsulfonilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquenilsulfonilo inferior opcionalmente sustituido con uno o más átomos halogenos, un grupo alquinilsulfonilo inferior opcionalmente sustituido con uno o mas átomos halogenos, un grupo alcoxilo inferior alquiltio inferior opcionalmente sustituido con uno o más átomos halogenos, o un grupo representado por -G-E, donde G representa un átomo de oxígeno, un átomo de azufre, SO, o SO2, y E representa un grupo arilo o un grupo heterocíclico y dicho grupo arilo o grupo heterocíclico puede ser sustituido con uno o más substituyentes seleccionados del grupo que consiste de (a) un átomo de halogeno, (b) un grupo alquilo inferior opcionalmente sustituido con uno o más átomos halogenos, (c) un grupo alcoxilo inferior opcionalmente sustituido con uno o más átomos halogenos, (d) un grupo alquiltio inferior opcionalmente sustituido con uno o más átomos halogenos, (e) un grupo alquilsulfinilo inferior opcionalmente sustituido con uno o más átomos halogenos, (f) un grupo alquilsulfonilo inferior opcionalmente sustituido con uno o más átomos halogenos, (g) un grupo ciano, y (h) un grupo nitro). Q representa un grupo arilo opcionalmente sustituido con uno o más sustituyentes, o un grupo heterocíclico opcionalmente sustituido con uno o más sustituyentes, m representa un entero de valor 1 a 5 (con la condicion que cuando m es un entero de valor 2 a 5, R7 puede ser igual o diferente), o una sal del mismo.Claim 1: A benzoylurea compound characterized in that it is represented by the formula (1), wherein X and Y each independently represents an oxygen atom or a sulfur atom, R1 represents a hydrogen atom, a formyl group, a group cyano, a lower alkylsulfonyl group optionally substituted with one or more substituents, an arylsulfonyl group optionally substituted with one or more substituents, a lower alkylcarbonylthio group optionally substituted with one or more substituents, a lower alkoxycarbonylthio group optionally substituted with one or more substituents, a aryloxycarbonylthio group substituted with one or more substituents, a mono or di (lower alkyl) aminosulfonyl group optionally substituted with one or more substituents, a mono or di (aryl) aminosulfonyl group optionally. substituted with one or more substituents, a lower alkyl group optionally substituted with one or more substituents, a lower alkenyl group optionally substituted with one or more substituents, a lower alkynyl group optionally substituted with one or more substituents, a lower cycloalkyl group optionally substituted with one or more substituents, a lower arylalkyl group optionally substituted with one or more substituents, an aryl group optionally substituted with one or more substituents, a lower alkoxy lower alkyl group optionally substituted with one or more substituents, a lower aryloxyalkyl group optionally substituted with one or more substituents, a lower alkyl lower alkyl group optionally substituted with one or more substituents, a lower alkyl lower alkyl group optionally substituted with one or more substituents, an optionally substituted lower alkyl lower alkylsulfonyl group, c on one or more substituents, a mono or di (lower alkyl) amino lower alkyl group optionally substituted with one or more substituents, a lower alkanoyl group substituted with one or more substituents, a lower alkoxycarbonyl group substituted with one or more substituents, a group aryloxycarbonyl substituted with one or more substituents, a lower arylalkoxycarbonyl group optionally substituted with one or more substituents, a carbamoyl group optionally substituted with one or more substituents, a thiocarbamoyl group optionally substituted with one or more substituents, a lower alkoxyoxalkyl group optionally substituted with one or more substituents, a lower arylalkoxyalkyl group optionally substituted with one or more substituents, an aryloxyoxalyl group optionally substituted with one or more substituents, an aminooxalyl group optionally substituted with one or more substituents, a lower alkoxy group optionally substituted with one or more more substituents, an aryloxy group optionally substituted with one or more substituents, a lower arylalkoxy group optionally substituted with one or more substituents, an amino group optionally substituted with one or more substituents, or a heterocyclic group optionally substituted with one or more substituents, R2 represents a lower alkylene group optionally substituted with one or more halogen atoms, A represents, (a) a group represented by OR3, (where R3 is a C1-3 alkyl group substituted with one or more substituents, optionally represents a group lower alkenyl optionally substituted with one or more substituents, a lower alkynyl group optionally substituted with one or more substituents, a lower alkanoyl group optionally substituted with one or more substituents, an aryl group optionally substituted with one or more substituents, or a lower arylalkyl group optionally substituted with one or more substituents), (b) a group represented by S (O) nR4, (wherein R4 represents a C1-3 alkyl group optionally substituted with one or more substituents, a lower alkenyl group optionally substituted with one or more substituents, a lower alkynyl group optionally substituted with one or more substituents, an aryl group optionally substituted with one or more substituents, or a lower arylalkyl group optionally substituted with one or more substituents, and n represents an integer of 0, 1 or 2), or (c) a group represented by NR5R6, (in wherein R5 and R6 each independently represent a C1-3 alkyl group optionally substituted with one or more substituents, a lower alkenyl group optionally substituted with one or more substituents, a lower alkynyl group optionally substituted with one or more substituents, an aryl group optionally substituted with one or more substituents, a lower arylalkyl group optionally substituted with one or more substituents, or R5 and R6 they can be linked at the ends thereof to form together with the nitrogen atom a 3- to 7-membered heterocyclic ring containing nitrogen that optionally possesses another nitrogen atom, an oxygen atom or a sulfur atom as the constituent atom of the ring), R7 represents a halogen atom, a nitro group, a cyano group, a lower arylalkoxyl group optionally substituted with one or more halogen atoms, a lower alkanoyl group optionally substituted with one or more halogen atoms, a lower alkoxycarbonyl group optionally substituted with one or more halogen atoms, an aryl group optionally substituted with one or more halogen atoms, a lower arylalkoxycarbonyl group optionally substituted with one or more halogen atoms, an arylcarbamoyl group optionally substituted with one or more., halogen atoms, a carbamoyl group optionally substituted with one or more plus lower alkyl group, a thiocarbamoyl group optionally substituted with one or lower alkyl groups, an amino group optionally substituted with one or more lower alkyl groups, a lower alkyl group optionally substituted with one or more halogen atoms, a lower alkoxy group optionally substituted with one or more halogen atoms, a group lower alkoxy lower alkoxy optionally substituted with one or more halogen atoms, a lower alkenyloxy group optionally substituted with one or more halogen atoms, a lower alkynyloxy group optionally substituted with one or more halogen atoms, a lower alkanoylamino group optionally substituted with one or more atoms halogens, a lower alkylthio group optionally substituted with one or more halogen atoms, a lower alkenylthio group optionally substituted with one or more halogen atoms, a lower alkynylthio group optionally substituted with one or more halogen atoms, an optionally substituted lower alkylsulfinyl group with one or more halogen atoms, a lower alkenylsulfinyl group optionally substituted with one or more halogen atoms, a lower alkylsulfinyl group optionally substituted with one or more halogen atoms, a lower alkylsulfonyl group optionally substituted with one or more halogen atoms, a lower alkenyl sulfonyl group optionally substituted with one or more halogen atoms, a lower alkynylsulfonyl group optionally substituted with one or more halogen atoms, a lower alkoxy lower alkylthio group optionally substituted with one or more halogen atoms, or a group represented by -GE, where G represents an atom of oxygen, a sulfur atom, SO, or SO2, and E represents an aryl group or a heterocyclic group and said aryl group or heterocyclic group may be substituted with one or more substituents selected from the group consisting of (a) an atom of halogen, (b) a lower alkyl group optionally substituted with one or more halogen atoms, (c) a lower alkoxy group optionally substituted with one or more halogen atoms, (d) a lower alkylthio group optionally substituted with one or more halogen atoms, (e) a lower alkylsulfinyl group optionally substituted with one or more halogen atoms, (f) a lower alkylsulfonyl group optionally substituted with one or more halogen atoms, (g) a cyano group, and (h) a nitro group). Q represents an aryl group optionally substituted with one or more substituents, or a heterocyclic group optionally substituted with one or more substituents, m represents an integer of value 1 to 5 (with the proviso that when m is an integer of value 2 to 5, R7 may be the same or different), or a salt thereof.
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2005353179 | 2005-12-07 | ||
| JP2006097943 | 2006-03-31 | ||
| JP2006209598 | 2006-08-01 |
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| Publication Number | Publication Date |
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| AR057992A1 true AR057992A1 (en) | 2008-01-09 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060105381A AR057992A1 (en) | 2005-12-07 | 2006-12-06 | BENZOILUREA COMPOUND AND USE OF THE SAME |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR057992A1 (en) |
| TW (1) | TW200804250A (en) |
| WO (1) | WO2007066496A1 (en) |
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| JP5158327B2 (en) * | 2007-07-06 | 2013-03-06 | 住友化学株式会社 | 4- (Trichloromethylthio) aniline and method for producing the same, and method for producing 4- (trifluoromethylthio) aniline |
| CN104430546B (en) * | 2014-12-09 | 2017-04-19 | 陈干忠 | High-yield disease-resistant and mothproof composite preparation for rubber trees as well as preparation method and application thereof |
| DE102016013066A1 (en) | 2016-11-03 | 2018-05-03 | Merck Patent Gmbh | fluorosurfactants |
| CN110526863B (en) * | 2019-08-29 | 2022-05-03 | 贵州大学 | A kind of acylthiourea or acylurea derivatives containing trifluoromethylpyridine and application thereof |
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| HU180240B (en) * | 1978-04-21 | 1983-02-28 | Gyogyszerkutato Intezet | Process for producing new,substituted 1,3-diaryl-2-iminoimidasolidines and 2-imino-hexahydro-pyrimidines |
| US5135953A (en) * | 1984-12-28 | 1992-08-04 | Ciba-Geigy | Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals |
| BR9815401A (en) * | 1997-09-30 | 2000-10-31 | Uniroyal Chem Co Inc | Increase in soybean seed yield by substituted benzoyl urea |
| TWI245761B (en) * | 2001-03-01 | 2005-12-21 | Telik Inc | Antagonists of MCP-1 function and methods of use thereof |
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2006
- 2006-11-13 WO PCT/JP2006/323048 patent/WO2007066496A1/en not_active Ceased
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| Publication number | Publication date |
|---|---|
| TW200804250A (en) | 2008-01-16 |
| WO2007066496A1 (en) | 2007-06-14 |
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