AR031117A1 - Uso de inhibidores de lipasa y secuestrantes de acido biliar para la preparacion de un medicamento, dicho inhibidor de lipasa y secuestrante de acido biliar y combinacion farmaceutica - Google Patents
Uso de inhibidores de lipasa y secuestrantes de acido biliar para la preparacion de un medicamento, dicho inhibidor de lipasa y secuestrante de acido biliar y combinacion farmaceuticaInfo
- Publication number
- AR031117A1 AR031117A1 ARP010103573A ARP010103573A AR031117A1 AR 031117 A1 AR031117 A1 AR 031117A1 AR P010103573 A ARP010103573 A AR P010103573A AR P010103573 A ARP010103573 A AR P010103573A AR 031117 A1 AR031117 A1 AR 031117A1
- Authority
- AR
- Argentina
- Prior art keywords
- biliar
- lipase
- preparation
- pharmaceutical combination
- biliar acid
- Prior art date
Links
- 229940086609 Lipase inhibitor Drugs 0.000 title abstract 3
- 239000002253 acid Substances 0.000 title 2
- 229940127470 Lipase Inhibitors Drugs 0.000 title 1
- 229940126601 medicinal product Drugs 0.000 title 1
- HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 abstract 4
- 229920000080 bile acid sequestrant Polymers 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 1
- AHLBNYSZXLDEJQ-FWEHEUNISA-N orlistat Chemical compound CCCCCCCCCCC[C@H](OC(=O)[C@H](CC(C)C)NC=O)C[C@@H]1OC(=O)[C@H]1CCCCCC AHLBNYSZXLDEJQ-FWEHEUNISA-N 0.000 abstract 1
- 229960001243 orlistat Drugs 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
- A61K31/716—Glucans
- A61K31/718—Starch or degraded starch, e.g. amylose, amylopectin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/74—Synthetic polymeric materials
- A61K31/785—Polymers containing nitrogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
Uso de un inhibidor de lipasa y de un secuestrante de ácido biliar que es para la preparacion de un medicamento para la prevencion y tratamiento de las enfermedades que se asocian con niveles elevados de colesterol plasmático; en especial al uso de un inhibidor de lipasa, por ejemplo, orlistat, y un secuestrante de ácido biliar aceptable para uso farmacéutico para el tratamiento de enfermedades que se relacionan con los niveles elevados de colesterol plasmático; y una combinacion farmacéutica.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00116392 | 2000-07-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR031117A1 true AR031117A1 (es) | 2003-09-10 |
Family
ID=8169383
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP010103573A AR031117A1 (es) | 2000-07-28 | 2001-07-26 | Uso de inhibidores de lipasa y secuestrantes de acido biliar para la preparacion de un medicamento, dicho inhibidor de lipasa y secuestrante de acido biliar y combinacion farmaceutica |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US6562329B2 (es) |
| EP (1) | EP1307263B1 (es) |
| JP (2) | JP4772264B2 (es) |
| KR (1) | KR100556324B1 (es) |
| CN (1) | CN1261094C (es) |
| AR (1) | AR031117A1 (es) |
| AT (1) | ATE293477T1 (es) |
| AU (2) | AU8969601A (es) |
| BR (1) | BR0112800A (es) |
| CA (1) | CA2416900C (es) |
| DE (1) | DE60110232T2 (es) |
| DK (1) | DK1307263T3 (es) |
| ES (1) | ES2240516T3 (es) |
| MX (1) | MXPA03000694A (es) |
| PT (1) | PT1307263E (es) |
| WO (1) | WO2002009814A2 (es) |
| ZA (1) | ZA200300454B (es) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2240516T3 (es) * | 2000-07-28 | 2005-10-16 | F. Hoffmann-La Roche Ag | Nuevo uso de los inhibidores de lipasa. |
| US20030027786A1 (en) | 2001-06-06 | 2003-02-06 | Karsten Maeder | Lipase inhibiting composition |
| JP4353414B2 (ja) * | 2001-07-30 | 2009-10-28 | 田辺三菱製薬株式会社 | 食後過血糖改善剤 |
| US20050276781A1 (en) * | 2004-06-09 | 2005-12-15 | Ross Edward A | Molecularly imprinted phosphate binders for therapeutic use |
| KR101547925B1 (ko) * | 2005-09-15 | 2015-08-27 | 젠자임 코포레이션 | 아민 중합체에 대한 샤셋 제형 |
| US8067402B2 (en) * | 2005-12-12 | 2011-11-29 | Allaccem, Inc. | Methods and systems for coating an oral surface |
| CA2648278C (en) * | 2006-04-03 | 2019-05-28 | Isa Odidi | Drug delivery composition |
| ITRM20060204A1 (it) | 2006-04-10 | 2007-10-11 | Vincenzo Savica | Farmaci e alimentei per diete normoproteiche iperproteiche ipopro teiche tutte ipofosforiche e bevande ipofosforiche |
| EP2478895A3 (en) | 2006-12-22 | 2012-12-19 | Ironwood Pharmaceuticals, Inc. | Compositions for treating esophageal disorders |
| WO2008103847A2 (en) | 2007-02-21 | 2008-08-28 | Allaccem, Incorporated | Bridged polycyclic compound based compositions for the inhibition and amelioration of disease |
| US20090023682A1 (en) * | 2007-07-19 | 2009-01-22 | Joseph Artiss | Composition Comprising Dietary Fat Complexer and Methods of Using Same |
| US8153618B2 (en) * | 2007-08-10 | 2012-04-10 | Allaccem, Inc. | Bridged polycyclic compound based compositions for topical applications for pets |
| US8188068B2 (en) * | 2007-08-10 | 2012-05-29 | Allaccem, Inc. | Bridged polycyclic compound based compositions for coating oral surfaces in pets |
| US8153617B2 (en) * | 2007-08-10 | 2012-04-10 | Allaccem, Inc. | Bridged polycyclic compound based compositions for coating oral surfaces in humans |
| US20090074833A1 (en) * | 2007-08-17 | 2009-03-19 | Whiteford Jeffery A | Bridged polycyclic compound based compositions for controlling bone resorption |
| US8524212B2 (en) * | 2007-10-24 | 2013-09-03 | Mitsubishi Tanabe Pharma Corporation | Prophylactic and/or therapeutic drug for nonalcoholic steatohepatitis |
| US20100004218A1 (en) * | 2008-06-20 | 2010-01-07 | Whiteford Jeffery A | Bridged polycyclic compound based compositions for renal therapy |
| US20100016270A1 (en) * | 2008-06-20 | 2010-01-21 | Whiteford Jeffery A | Bridged polycyclic compound based compositions for controlling cholesterol levels |
| WO2009158625A2 (en) * | 2008-06-26 | 2009-12-30 | Ironwood Pharmaceuticals, Inc. | Compositions and methods for treating or preventing gastrointestinal disorders and gerd-related respiratory disorders |
| US20100008988A1 (en) * | 2008-07-14 | 2010-01-14 | Glenmark Generics, Ltd. | Tablet compositions of amine polymers |
| CN101791296B (zh) * | 2010-01-17 | 2012-08-29 | 山东新时代药业有限公司 | 一种奥利司他片剂及其制备方法 |
| LT2568827T (lt) * | 2010-05-14 | 2018-08-27 | Omega Pharma Innovation & Development Nv | Kompozicija, skirta dietinės mitybos riebalų absorbavimo mažinimui |
| PH12021552553A1 (en) * | 2019-04-16 | 2022-06-20 | Celagenex Res India Pvt Ltd | Synergistic lipid controlling compositions |
| KR102271821B1 (ko) * | 2020-12-18 | 2021-07-01 | 주식회사 엔테로바이옴 | 오를리스타트 및 아커만시아 뮤시니필라 eb-amdk19 균주를 포함하는 조성물 |
| JP2024500188A (ja) * | 2020-12-22 | 2024-01-04 | サイトゼリックス,インク. | 胆道送達方法、その使用のための組成物及びキット |
| CN113057340B (zh) * | 2021-04-29 | 2024-01-19 | 南京邮电大学 | 一种菌菇膳食纤维改性方法 |
| CN116018147A (zh) * | 2021-08-24 | 2023-04-25 | 中美华世通生物医药科技(武汉)股份有限公司 | 用于治疗高尿酸血症的聚合物、组合物和方法 |
| WO2023023938A1 (en) * | 2021-08-24 | 2023-03-02 | Waterstone Pharmaceuticals (Wuhan) Co., Ltd. | Polymers, compositions and methods for treating hyperuricemia |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1247547A (en) | 1983-06-22 | 1988-12-28 | Paul Hadvary | Leucine derivatives |
| CA1270837A (en) | 1984-12-21 | 1990-06-26 | Hoffmann-La Roche Limited | Oxetanones |
| CA1328881C (en) | 1984-12-21 | 1994-04-26 | Pierre Barbier | Process for the manufacture of oxetanones |
| IT1190349B (it) * | 1986-06-16 | 1988-02-16 | Prodotti Formenti Srl | Composizioni farmaceutiche ad attivita' sequestrante degli acidi biliari contenenti colestiramina quale principio attivo,e procedimento per prepararle |
| US5063210A (en) * | 1989-04-20 | 1991-11-05 | Lange Iii Louis G | Use of sulfated polysaccharides to decrease cholesterol and fatty acid absorption |
| CA2035972C (en) | 1990-02-23 | 2006-07-11 | Martin Karpf | Process for the preparation of oxetanones |
| US5298497A (en) * | 1990-05-15 | 1994-03-29 | E. R. Squibb & Sons, Inc. | Method for preventing onset of hypertension employing a cholesterol lowering drug |
| US5274143A (en) | 1991-07-23 | 1993-12-28 | Hoffmann-La Roche Inc. | Process for the preparation of (R)-3-hexyl-5,6-dihydro-4-hydroxy-6-undecyl-2H-pyran-2-one and (R)-5,6-dihydro-6-undecyl-2H-pyran-2,4(3H)-dione |
| US5616570A (en) * | 1991-10-18 | 1997-04-01 | Lange, Iii; Louis G. | Use of non-absorbable synthetic sulfated polysaccharides to decrease cholesterol absorbtion |
| CA2098167C (en) * | 1992-06-24 | 2006-12-19 | Dorothea Isler | Foodstuffs and feedstuffs containing a lipase inhibitor |
| TW381025B (en) * | 1993-08-05 | 2000-02-01 | Hoffmann La Roche | Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor |
| KR19980702533A (ko) * | 1995-12-26 | 1998-07-15 | 도리이 신이찌로 | 프로시아니딘을 유효성분으로 하는 항비만제 |
| US6004996A (en) | 1997-02-05 | 1999-12-21 | Hoffman-La Roche Inc. | Tetrahydrolipstatin containing compositions |
| US6267952B1 (en) | 1998-01-09 | 2001-07-31 | Geltex Pharmaceuticals, Inc. | Lipase inhibiting polymers |
| DE69916288T2 (de) | 1998-08-14 | 2005-03-24 | F. Hoffmann-La Roche Ag | Lipasehemmer und chitosan enthaltende arzneimittel |
| ATE293970T1 (de) * | 1998-08-14 | 2005-05-15 | Hoffmann La Roche | Lipasehemmer enthaltende pharmazeutische zusammensetzungen |
| GB9900416D0 (en) | 1999-01-08 | 1999-02-24 | Alizyme Therapeutics Ltd | Inhibitors |
| AU2001289699B2 (en) * | 2000-07-28 | 2006-06-01 | Cheplapharm Arzneimittel Gmbh | New pharmaceutical composition |
| ES2240516T3 (es) * | 2000-07-28 | 2005-10-16 | F. Hoffmann-La Roche Ag | Nuevo uso de los inhibidores de lipasa. |
-
2001
- 2001-07-19 ES ES01969436T patent/ES2240516T3/es not_active Expired - Lifetime
- 2001-07-19 AU AU8969601A patent/AU8969601A/xx active Pending
- 2001-07-19 MX MXPA03000694A patent/MXPA03000694A/es active IP Right Grant
- 2001-07-19 AT AT01969436T patent/ATE293477T1/de active
- 2001-07-19 JP JP2002515365A patent/JP4772264B2/ja not_active Expired - Fee Related
- 2001-07-19 KR KR1020037001188A patent/KR100556324B1/ko not_active Expired - Fee Related
- 2001-07-19 CN CNB018135218A patent/CN1261094C/zh not_active Expired - Lifetime
- 2001-07-19 DE DE60110232T patent/DE60110232T2/de not_active Expired - Lifetime
- 2001-07-19 WO PCT/EP2001/008353 patent/WO2002009814A2/en not_active Ceased
- 2001-07-19 DK DK01969436T patent/DK1307263T3/da active
- 2001-07-19 BR BR0112800-0A patent/BR0112800A/pt not_active Application Discontinuation
- 2001-07-19 EP EP01969436A patent/EP1307263B1/en not_active Expired - Lifetime
- 2001-07-19 CA CA002416900A patent/CA2416900C/en not_active Expired - Lifetime
- 2001-07-19 PT PT01969436T patent/PT1307263E/pt unknown
- 2001-07-19 AU AU2001289696A patent/AU2001289696B2/en not_active Expired
- 2001-07-25 US US09/912,956 patent/US6562329B2/en not_active Expired - Lifetime
- 2001-07-26 AR ARP010103573A patent/AR031117A1/es unknown
-
2002
- 2002-12-06 US US10/313,409 patent/US20030138396A1/en not_active Abandoned
-
2003
- 2003-01-16 ZA ZA200300454A patent/ZA200300454B/en unknown
-
2006
- 2006-04-20 US US11/408,232 patent/US20060189574A1/en not_active Abandoned
-
2008
- 2008-10-29 JP JP2008278382A patent/JP2009108062A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP4772264B2 (ja) | 2011-09-14 |
| EP1307263B1 (en) | 2005-04-20 |
| CN1444496A (zh) | 2003-09-24 |
| DE60110232D1 (de) | 2005-05-25 |
| JP2004505066A (ja) | 2004-02-19 |
| AU8969601A (en) | 2002-02-13 |
| BR0112800A (pt) | 2003-07-01 |
| DK1307263T3 (da) | 2005-08-22 |
| KR20030069978A (ko) | 2003-08-27 |
| ES2240516T3 (es) | 2005-10-16 |
| US20060189574A1 (en) | 2006-08-24 |
| WO2002009814A2 (en) | 2002-02-07 |
| US20020042395A1 (en) | 2002-04-11 |
| US20030138396A1 (en) | 2003-07-24 |
| AU2001289696B2 (en) | 2006-07-06 |
| CN1261094C (zh) | 2006-06-28 |
| MXPA03000694A (es) | 2003-06-04 |
| US6562329B2 (en) | 2003-05-13 |
| ATE293477T1 (de) | 2005-05-15 |
| DE60110232T2 (de) | 2006-01-19 |
| CA2416900A1 (en) | 2002-02-07 |
| EP1307263A2 (en) | 2003-05-07 |
| ZA200300454B (en) | 2004-04-16 |
| KR100556324B1 (ko) | 2006-03-03 |
| WO2002009814A3 (en) | 2002-04-18 |
| JP2009108062A (ja) | 2009-05-21 |
| PT1307263E (pt) | 2005-08-31 |
| CA2416900C (en) | 2007-07-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |