NO20024005D0 - Pteridinforbindelser for behandling av psoriasis - Google Patents

Pteridinforbindelser for behandling av psoriasis

Info

Publication number: NO20024005D0
Authority: NO; Norway
Prior art keywords: psoriasis; treatment; pteridine compounds; formula; pteridine
Prior art date: 2000-02-23

Application number

NO20024005A

Other languages

English (en)

Other versions

NO20024005L (no

NO329898B1 (no

Inventor

Roger Victor Bonnert

Stewart Gardiner

Fraser Hunt

Iain Alistair Stewart Walters

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-02-23

Filing date

2002-08-22

Publication date

2002-08-22

2002-08-22 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2002-08-22 Publication of NO20024005D0 publication Critical patent/NO20024005D0/no

2002-10-22 Publication of NO20024005L publication Critical patent/NO20024005L/no

2011-01-24 Publication of NO329898B1 publication Critical patent/NO329898B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Immunology (AREA)
Pulmonology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Dermatology (AREA)
Rheumatology (AREA)
Addiction (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Diabetes (AREA)
Hematology (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Heart & Thoracic Surgery (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO20024005A 2000-02-23 2002-08-22 Pteridin forbindelser, fremgangsmate for fremstilling av slike, mellomprodukter, farmasoytiske sammensetninger og fremstilling omfattende slike, anvendelsen av slike i terapi samt anvendelse for fremstilling av medikamenter for behandling av sykdom NO329898B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0004128A GB2359551A (en)	2000-02-23	2000-02-23	Pharmaceutically active pyrimidine derivatives
PCT/SE2001/000374 WO2001062758A1 (en)	2000-02-23	2001-02-20	Pteridine compounds for the treatment of psoriasis

Publications (3)

Publication Number	Publication Date
NO20024005D0 true NO20024005D0 (no)	2002-08-22
NO20024005L NO20024005L (no)	2002-10-22
NO329898B1 NO329898B1 (no)	2011-01-24

Family

ID=9886153

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20024005A NO329898B1 (no)	2000-02-23	2002-08-22	Pteridin forbindelser, fremgangsmate for fremstilling av slike, mellomprodukter, farmasoytiske sammensetninger og fremstilling omfattende slike, anvendelsen av slike i terapi samt anvendelse for fremstilling av medikamenter for behandling av sykdom

Country Status (32)

Country	Link
US (2)	US6875868B2 (no)
EP (1)	EP1259512B1 (no)
JP (1)	JP2003524012A (no)
KR (1)	KR100795758B1 (no)
CN (1)	CN1190437C (no)
AR (1)	AR029805A1 (no)
AT (1)	ATE250605T1 (no)
AU (1)	AU782509B2 (no)
BG (1)	BG107002A (no)
BR (1)	BR0108600A (no)
CA (1)	CA2400217C (no)
CO (1)	CO5290258A1 (no)
CZ (1)	CZ20022839A3 (no)
DE (1)	DE60100851T2 (no)
DK (1)	DK1259512T3 (no)
EE (1)	EE200200461A (no)
ES (1)	ES2206402T3 (no)
GB (1)	GB2359551A (no)
HU (1)	HUP0204399A3 (no)
IL (2)	IL151132A0 (no)
IS (1)	IS6491A (no)
MX (1)	MXPA02008233A (no)
NO (1)	NO329898B1 (no)
NZ (1)	NZ520355A (no)
PL (1)	PL358004A1 (no)
PT (1)	PT1259512E (no)
RU (1)	RU2002125451A (no)
SK (1)	SK12152002A3 (no)
TR (1)	TR200302214T4 (no)
UA (1)	UA72590C2 (no)
WO (1)	WO2001062758A1 (no)
ZA (1)	ZA200206590B (no)

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SE0003828D0 (sv)	2000-10-20	2000-10-20	Astrazeneca Ab	Novel compounds
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JP5111113B2 (ja) *	2004-12-13	2012-12-26	サネシスファーマシューティカルズ，インコーポレイテッド	Ｒａｆキナーゼ阻害剤として有用なピリドピリミジノン、ジヒドロピリミドピリミジノンおよびプテリジノン
AR053347A1 (es)	2005-04-06	2007-05-02	Astrazeneca Ab	Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en)	2005-04-06	2010-05-25	Астразенека Аб	Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
US7439358B2 (en)	2006-02-08	2008-10-21	Boehringer Ingelheim International Gmbh	Specific salt, anhydrous and crystalline form of a dihydropteridione derivative
RU2437889C2 (ru) *	2006-09-29	2011-12-27	Астразенека Аб	НОВЫЕ 5,7-ДИЗАМЕЩЕННЫЕ ПРОИЗВОДНЫЕ [1,3]ТИАЗОЛО[4,5-d]ПИРИМИДИН-2-(3Н)-АМИНА И ИХ ПРИМЕНЕНИЕ В ТЕРАПИИ
TW200820973A (en) *	2006-09-29	2008-05-16	Astrazeneca Ab	Novel compounds 480
EP2185559A1 (en) *	2007-08-03	2010-05-19	Boehringer Ingelheim International GmbH	Crystalline form of a dihydropteridione derivative
RU2011101661A (ru) *	2008-07-16	2012-08-27	Астразенека Аб (Se)	Пиримидилсульфонамидное производное и его применение для лечения хемокин-опосредованных заболеваний
US8546566B2 (en)	2010-10-12	2013-10-01	Boehringer Ingelheim International Gmbh	Process for manufacturing dihydropteridinones and intermediates thereof
US9358233B2 (en)	2010-11-29	2016-06-07	Boehringer Ingelheim International Gmbh	Method for treating acute myeloid leukemia
US9370535B2 (en)	2011-05-17	2016-06-21	Boehringer Ingelheim International Gmbh	Method for treatment of advanced solid tumors
JP6093759B2 (ja)	2011-06-01	2017-03-08	ジャナスバイオセラピューティクス，インク．	新規の免疫系調節剤
CN105722972A (zh)	2013-06-18	2016-06-29	纽约大学	参与金黄色葡萄球菌杀白细胞素的细胞毒性的细胞因素：新型治疗靶点
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2000
- 2000-02-23 GB GB0004128A patent/GB2359551A/en not_active Withdrawn
2001
- 2001-02-20 PT PT01906493T patent/PT1259512E/pt unknown
- 2001-02-20 JP JP2001562540A patent/JP2003524012A/ja active Pending
- 2001-02-20 HU HU0204399A patent/HUP0204399A3/hu unknown
- 2001-02-20 SK SK1215-2002A patent/SK12152002A3/sk unknown
- 2001-02-20 IL IL15113201A patent/IL151132A0/xx unknown
- 2001-02-20 WO PCT/SE2001/000374 patent/WO2001062758A1/en not_active Ceased
- 2001-02-20 EP EP01906493A patent/EP1259512B1/en not_active Expired - Lifetime
- 2001-02-20 DE DE60100851T patent/DE60100851T2/de not_active Expired - Lifetime
- 2001-02-20 US US10/204,814 patent/US6875868B2/en not_active Expired - Fee Related
- 2001-02-20 KR KR1020027011047A patent/KR100795758B1/ko not_active Expired - Fee Related
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- 2001-02-20 CN CNB018054676A patent/CN1190437C/zh not_active Expired - Fee Related
- 2001-02-20 CZ CZ20022839A patent/CZ20022839A3/cs unknown
- 2001-02-20 RU RU2002125451/04A patent/RU2002125451A/ru not_active Application Discontinuation
- 2001-02-20 PL PL01358004A patent/PL358004A1/xx not_active Application Discontinuation
- 2001-02-20 NZ NZ520355A patent/NZ520355A/en not_active IP Right Cessation
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- 2001-02-20 AU AU34316/01A patent/AU782509B2/en not_active Ceased
- 2001-02-20 ES ES01906493T patent/ES2206402T3/es not_active Expired - Lifetime
- 2001-02-20 AT AT01906493T patent/ATE250605T1/de active
- 2001-02-20 EE EEP200200461A patent/EE200200461A/xx unknown
- 2001-02-20 DK DK01906493T patent/DK1259512T3/da active
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- 2001-02-20 MX MXPA02008233A patent/MXPA02008233A/es active IP Right Grant
- 2001-02-20 BR BR0108600-6A patent/BR0108600A/pt not_active Application Discontinuation
- 2001-02-21 CO CO01013781A patent/CO5290258A1/es not_active Application Discontinuation
- 2001-02-21 AR ARP010100773A patent/AR029805A1/es not_active Application Discontinuation
2002
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- 2002-08-07 IS IS6491A patent/IS6491A/is unknown
- 2002-08-14 BG BG107002A patent/BG107002A/bg unknown
- 2002-08-16 ZA ZA200206590A patent/ZA200206590B/en unknown
- 2002-08-22 NO NO20024005A patent/NO329898B1/no not_active IP Right Cessation
2004
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Also Published As

Publication number	Publication date
MXPA02008233A (es)	2004-04-05
CN1404482A (zh)	2003-03-19
JP2003524012A (ja)	2003-08-12
DE60100851T2 (de)	2004-07-15
HK1050899A1 (en)	2003-07-11
CA2400217A1 (en)	2001-08-30
KR20030005207A (ko)	2003-01-17
ATE250605T1 (de)	2003-10-15
HUP0204399A2 (en)	2003-05-28
ZA200206590B (en)	2003-11-17
RU2002125451A (ru)	2004-01-10
DE60100851D1 (de)	2003-10-30
PL358004A1 (en)	2004-08-09
UA72590C2 (uk)	2005-03-15
CO5290258A1 (es)	2003-06-27
PT1259512E (pt)	2004-02-27
WO2001062758A1 (en)	2001-08-30
US20050171345A1 (en)	2005-08-04
DK1259512T3 (da)	2003-12-29
US6875868B2 (en)	2005-04-05
GB0004128D0 (en)	2000-04-12
NZ520355A (en)	2005-01-28
NO20024005L (no)	2002-10-22
TR200302214T4 (tr)	2004-01-21
SK12152002A3 (sk)	2003-03-04
AU3431601A (en)	2001-09-03
NO329898B1 (no)	2011-01-24
BR0108600A (pt)	2002-11-12
HUP0204399A3 (en)	2004-11-29
GB2359551A (en)	2001-08-29
CZ20022839A3 (cs)	2002-11-13
IS6491A (is)	2002-08-07
AR029805A1 (es)	2003-07-16
EP1259512A1 (en)	2002-11-27
EE200200461A (et)	2003-12-15
AU782509B2 (en)	2005-08-04
IL151132A (en)	2010-11-30
US7579342B2 (en)	2009-08-25
EP1259512B1 (en)	2003-09-24
US20030055250A1 (en)	2003-03-20
BG107002A (bg)	2003-04-30
ES2206402T3 (es)	2004-05-16
IL151132A0 (en)	2003-04-10
CA2400217C (en)	2009-02-17
CN1190437C (zh)	2005-02-23
KR100795758B1 (ko)	2008-01-21

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PT1263725E (pt)	2005-02-28	Novos compostos
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ATE365720T1 (de)	2007-07-15	Agonisten von beta-adrenorezeptoren
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BG66080B1 (bg)	2011-03-31	Заместени тиоацетамиди
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MY128924A (en)	2007-02-28	Novel compounds
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SE0302139D0 (sv)	2003-07-28	Novel compounds
SE9902765D0 (sv)	1999-07-21	Novel compounds
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DE60129829D1 (de)	2007-09-20	Zyklisierte benzamid-neurokinin-antagonisten zur verwendung in therapie
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SE0004827D0 (sv)	2000-12-22	Therapeutic compounds

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