AR038326A1 - Antibacterianos feniloxazolidinonas sustituidos con heterociclicos biciclicos y composiciones relacionadas y metodos - Google Patents
Antibacterianos feniloxazolidinonas sustituidos con heterociclicos biciclicos y composiciones relacionadas y metodosInfo
- Publication number
- AR038326A1 AR038326A1 ARP030100243A ARP030100243A AR038326A1 AR 038326 A1 AR038326 A1 AR 038326A1 AR P030100243 A ARP030100243 A AR P030100243A AR P030100243 A ARP030100243 A AR P030100243A AR 038326 A1 AR038326 A1 AR 038326A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- carbon atoms
- group
- amino
- straight
- Prior art date
Links
- 229940088710 antibiotic agent Drugs 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 13
- 125000004432 carbon atom Chemical group C* 0.000 abstract 10
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 6
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 5
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 4
- -1 amino, carboxy Chemical group 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 125000003917 carbamoyl group Chemical class [H]N([H])C(*)=O 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- 125000001072 heteroaryl group Chemical group 0.000 abstract 3
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 125000003282 alkyl amino group Chemical group 0.000 abstract 2
- 150000001412 amines Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000001584 benzyloxycarbonyl group Chemical group C(=O)(OCC1=CC=CC=C1)* 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 229920001577 copolymer Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000002757 morpholinyl group Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000004043 oxo group Chemical group O=* 0.000 abstract 1
- UYWQUFXKFGHYNT-UHFFFAOYSA-N phenylmethyl ester of formic acid Natural products O=COCC1=CC=CC=C1 UYWQUFXKFGHYNT-UHFFFAOYSA-N 0.000 abstract 1
- 125000003386 piperidinyl group Chemical group 0.000 abstract 1
- 125000000719 pyrrolidinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000003944 tolyl group Chemical group 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Un compuesto de fórmula (1) en la cual: R se selecciona entre el grupo que consiste en OH, O-Arilo, O-Heteroarilo, N3, OR', OSO2R'', -NR'''R'''', o un compuesto de fórmula (2) en la cual: (i) R' es acilo de cadena recta o ramificada que tiene hasta 6 átomos de carbono de bencilo; (ii) R'' es alquilo de cadena recta o ramificado, que tiene hasta 5 átomos de carbono, fenilo o tolilo; y (iii) R''' y R'''' se seleccionan independientemente entre el grupo que consiste en H, cicloalquilo que tiene de 3 a 6 átomos de carbono, fenilo o terbutoxicarbonilo, fluoreniloxicarbonilo, benciloxicarbonilo, alquilo de cadena recta o ramificado que tiene hasta 6 átomos de carbono que es optativamente sustituido por ciano o alcoxicarbonilo que tiene hasta 4 átomos de carbono, -CO2-R1, -CO-R1, -CS-R1, y -SO2R4, en donde R1 se selecciona entre el grupo que consiste en H, cicloaquilo que tiene de 3 a 6 átomos de carbono, trifluorometilo o fenilo, bencilo o acilo con hasta 5 átomos de carbono, alquilo de cadena recta o ramificado con hasta 6 átomos de carbono, dicho alquilo optativamente sustituido por alcoxicarbonilo de cadena recta o ramificado con hasta 5 átomos de carbono, OH, ciano, hasta 3 átomos de halógeno, y -NR5R6 en donde R5 y R6 son idénticos o diferentes y se seleccionan entre H, fenilo o alquilo, de cadena recta o ramificado con hasta 4 átomos de carbono; R4 se selecciona entre alquilo de cadena recta o ramificado con hasta 4 átomos de carbono o fenilo y; R4a es CN, COR4c, COOR4c, CONHR4c, CO-NR4c, R4d, SO2R4c, ó NO2; R4b es H, alquilo, OR4c, SR4c, amino, NHR4c, NR4c, R4d; R4c y R4d se seleccionan independientemente entre H, alquilo, arilo o en el caso de cualquier grupo NR4cR4d, R4c y R4d tomados en conjunto con el átomo de nitrógeno al cual están unidos forman un grupo pirrolidinilo, piperidinilo o morfolinilo insustituido o sustituido; X es 0 a 4 miembros seleccionados independientemente entre el grupo que consiste en halógeno, OH, nitro, alcoxi C1-8, alquil-amino C1-8, di(alquil-C1-8)amino, carboxi, alcoxicarbonilo, alquil C1-8-CO-O-, alquil C1-8-CO-NH-, carboxamida, CN, amina, cicloalquilo C3-6, alquilo C1-8 sustituido optativamente con uno o más miembros seleccionados entre el grupo que consiste en F, Cl, OH; e Y es un radical de las fórmulas (3) ó (4): en donde R5, R6, R7 y R8 son cada uno en forma independiente H, alquilo, CN, nitro, alquilo C1-8, halo-alquilo-C1-8, formilo, carboxi, alcoxicarbonilo, carboxamida o R5 y R6 y/o R7 y R8 juntos forman un grupo oxo; R9 y R10 son individualmente en forma independiente H, halógeno, alquilo, OH, CN, nitro, alquilo C1-8, halo-alquilo-C1-8, alcoxilo C1-8, amino, alquil-C1-8-amino, di(alquil-C1-8)amino, formilo, carboxi, alcoxicarbonilo, alquil-C1-8-CO-O, alquil-C1-8-CO-NH-, carboxamida o amina; Q es un anillo de fenilo fusionado o un anillo heteroaromático de cinco o seis miembros con uno a cuatro miembros seleccionados entre el grupo que consiste en S, O y N; Z es halógeno, alquilo, alquilo sustituido, arilo, arilo sustituido, heteroarilo, heteroarilo sustituido, CN, CHO, COalquilo, amino, alcoxi, HNCO-(alquilo-C1-8), alilo, propargilo, alenilo o N-alquiltiocarbamoílo; y m es 0 ó 1, y sus sales y ésteres farmacéuticamente aceptables.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/058,841 US6608081B2 (en) | 1999-08-12 | 2002-01-28 | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR038326A1 true AR038326A1 (es) | 2005-01-12 |
Family
ID=27658242
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP030100243A AR038326A1 (es) | 2002-01-28 | 2003-01-28 | Antibacterianos feniloxazolidinonas sustituidos con heterociclicos biciclicos y composiciones relacionadas y metodos |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US6608081B2 (es) |
| EP (1) | EP1470123A1 (es) |
| JP (1) | JP2005520815A (es) |
| KR (1) | KR20040085167A (es) |
| CN (1) | CN1642949A (es) |
| AR (1) | AR038326A1 (es) |
| BR (1) | BR0307259A (es) |
| CA (1) | CA2474718A1 (es) |
| MX (1) | MXPA04007240A (es) |
| MY (1) | MY134701A (es) |
| PL (1) | PL371527A1 (es) |
| RU (1) | RU2004123097A (es) |
| TW (1) | TW200307679A (es) |
| WO (1) | WO2003064415A1 (es) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6897230B2 (en) * | 2001-04-17 | 2005-05-24 | Kyorin Pharmaceutical Co., Ltd. | Bicyclo[3/1/0] hexane containing oxazolidinone antibiotics and derivatives thereof |
| WO2005005420A1 (en) * | 2003-07-02 | 2005-01-20 | Merck & Co., Inc. | Cyclopropyl group substituted oyazolidinone antibiotics and derivatives thereof |
| US20070293493A1 (en) * | 2003-07-02 | 2007-12-20 | Milton Hammond | Oxazolidinone antibiotics and derivatives thereof |
| WO2005005398A2 (en) * | 2003-07-02 | 2005-01-20 | Merck & Co., Inc. | Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof |
| EP1656357A1 (en) * | 2003-07-02 | 2006-05-17 | Merck & Co., Inc. | Oxazolidinone antibiotics and derivatives thereof |
| US7687627B2 (en) * | 2003-09-08 | 2010-03-30 | Wockhardt Limited | Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy |
| DOP2006000268A (es) * | 2005-12-22 | 2007-07-31 | Pfizer Prod Inc | Agentes antibacterianos |
| US8124623B2 (en) | 2006-11-10 | 2012-02-28 | Actelion Pharmaceuticals Ltd. | 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
| JP4484965B2 (ja) * | 2006-11-10 | 2010-06-16 | アクテリオン ファーマシューティカルズ リミテッド | ５−ヒドロキシメチル−オキサゾリジン−２−オン誘導体 |
| CN101084901B (zh) * | 2007-06-22 | 2011-12-21 | 复旦大学 | 一种葡萄球菌抑制剂 |
| AU2009318783A1 (en) | 2008-11-20 | 2011-06-23 | Panacea Biotec Ltd. | Novel antimicrobials |
| JP5696142B2 (ja) | 2009-06-26 | 2015-04-08 | パナセア バイオテック リミテッド | 新規アザビシクロヘキサン類 |
| US9487545B2 (en) | 2011-09-30 | 2016-11-08 | Xuanzhu Pharma Co., Ltd. | Fused ring-containing oxazolidinones antibiotics |
| JP6162704B2 (ja) * | 2011-10-11 | 2017-07-12 | カウンシル オブ サイエンティフィク アンド インダストリアル リサーチ | オキサゾリジノン誘導体のシラアナログ及びその合成 |
| US10674982B2 (en) | 2015-08-06 | 2020-06-09 | Covidien Lp | System and method for local three dimensional volume reconstruction using a standard fluoroscope |
| US10716525B2 (en) | 2015-08-06 | 2020-07-21 | Covidien Lp | System and method for navigating to target and performing procedure on target utilizing fluoroscopic-based local three dimensional volume reconstruction |
| US10702226B2 (en) | 2015-08-06 | 2020-07-07 | Covidien Lp | System and method for local three dimensional volume reconstruction using a standard fluoroscope |
| CN106083994B (zh) * | 2016-04-18 | 2019-12-06 | 南京曼杰生物科技有限公司 | 取代的噁唑烷酮水溶性衍生物及其应用 |
| JP6821716B2 (ja) * | 2016-06-29 | 2021-01-27 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | Ｂ型肝炎ウイルス感染の処置および予防のための新規のジヒドロピロロピリミジン |
| US10087171B2 (en) | 2016-12-19 | 2018-10-02 | Actelion Pharmaceuticals Ltd | Crystalline forms of cadazolid |
| US11529190B2 (en) | 2017-01-30 | 2022-12-20 | Covidien Lp | Enhanced ablation and visualization techniques for percutaneous surgical procedures |
| US11793579B2 (en) | 2017-02-22 | 2023-10-24 | Covidien Lp | Integration of multiple data sources for localization and navigation |
| US10699448B2 (en) | 2017-06-29 | 2020-06-30 | Covidien Lp | System and method for identifying, marking and navigating to a target using real time two dimensional fluoroscopic data |
| WO2019075074A1 (en) | 2017-10-10 | 2019-04-18 | Covidien Lp | SYSTEM AND METHOD FOR IDENTIFICATION AND MARKING OF A TARGET IN A THREE-DIMENSIONAL FLUOROSCOPIC RECONSTRUCTION |
| US11364004B2 (en) | 2018-02-08 | 2022-06-21 | Covidien Lp | System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target |
| KR102777328B1 (ko) | 2018-07-25 | 2025-03-10 | 자이두스 라이프사이언시즈 리미티드 | 포유류 감염 치료를 위한 신규 화합물 |
| US11705238B2 (en) | 2018-07-26 | 2023-07-18 | Covidien Lp | Systems and methods for providing assistance during surgery |
| US11877806B2 (en) | 2018-12-06 | 2024-01-23 | Covidien Lp | Deformable registration of computer-generated airway models to airway trees |
| US11801113B2 (en) | 2018-12-13 | 2023-10-31 | Covidien Lp | Thoracic imaging, distance measuring, and notification system and method |
| US11617493B2 (en) | 2018-12-13 | 2023-04-04 | Covidien Lp | Thoracic imaging, distance measuring, surgical awareness, and notification system and method |
| US11357593B2 (en) | 2019-01-10 | 2022-06-14 | Covidien Lp | Endoscopic imaging with augmented parallax |
| US11625825B2 (en) | 2019-01-30 | 2023-04-11 | Covidien Lp | Method for displaying tumor location within endoscopic images |
| US11744643B2 (en) | 2019-02-04 | 2023-09-05 | Covidien Lp | Systems and methods facilitating pre-operative prediction of post-operative tissue function |
| WO2020234636A1 (en) | 2019-05-17 | 2020-11-26 | Cadila Healthcare Limited | Novel compounds for the treatment of mammalian infections |
| US11627924B2 (en) | 2019-09-24 | 2023-04-18 | Covidien Lp | Systems and methods for image-guided navigation of percutaneously-inserted devices |
| US12102298B2 (en) | 2019-12-10 | 2024-10-01 | Covidien Lp | Lymphatic system tracking |
| US12161309B2 (en) | 2020-09-24 | 2024-12-10 | Covidien Lp | Articulating mechanism for the laparoscopic ablation device for blunt dissection |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US3391150A (en) | 1965-12-17 | 1968-07-02 | Merck & Co Inc | Thiadiazole compounds and processes for preparing same |
| WO1989005643A1 (en) | 1987-12-18 | 1989-06-29 | Pfizer Inc. | Heterocyclic-substituted quinoline-carboxylic acids |
| DE4121214A1 (de) | 1991-06-27 | 1993-01-14 | Bayer Ag | 7-azaisoindolinyl-chinolon- und -naphthyridoncarbonsaeure-derivate |
| AU659501B2 (en) | 1991-10-23 | 1995-05-18 | Biota Scientific Management Pty Ltd | Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of alpha-D-neuraminic acid |
| KR100257418B1 (ko) | 1991-11-01 | 2000-05-15 | 로렌스 티. 마이젠헬더 | 치환된 아릴-및 헤테로아릴-페닐옥사졸리디논 |
| US5289157A (en) | 1991-12-23 | 1994-02-22 | Vitafit International, Inc. | Medicine reminder and storage device |
| MY115155A (en) | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
| EP0788498B1 (en) | 1994-10-26 | 2001-08-16 | PHARMACIA & UPJOHN COMPANY | Phenyloxazolidinone antimicrobials |
| US5952324A (en) | 1994-11-15 | 1999-09-14 | Pharmacia & Upjohn Company | Bicyclic oxazine and thiazine oxazolidinone antibacterials |
| BR9607017A (pt) | 1995-02-03 | 1997-10-28 | Upjohn Co | Composto e uso do mesmo |
| US6124334A (en) | 1995-02-03 | 2000-09-26 | Pharmacia & Upjohn Company | Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials |
| CA2218088A1 (en) | 1995-05-11 | 1996-11-14 | Pharmacia & Upjohn Company | Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
| MX9703040A (es) | 1995-09-12 | 1997-07-31 | Upjohn Co | Antimicrobianos de feniloxazolidinona. |
| DE19601264A1 (de) | 1996-01-16 | 1997-07-17 | Bayer Ag | Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone |
| DE19604223A1 (de) | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
| CZ298060B6 (cs) | 1996-04-11 | 2007-06-06 | Pharmacia & Upjohn Company | Zpusob prípravy oxazolidinonu |
| CN1138765C (zh) | 1997-05-30 | 2004-02-18 | 法玛西雅厄普约翰美国公司 | 带有硫代羰基功能基的噁唑烷酮抗菌剂 |
| GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
| JPH11322729A (ja) | 1998-03-09 | 1999-11-24 | Hokuriku Seiyaku Co Ltd | ジチオカルバミド酸誘導体 |
| GB9812019D0 (en) | 1998-06-05 | 1998-07-29 | Zeneca Ltd | Chemical compounds |
| US6413981B1 (en) * | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
-
2002
- 2002-01-28 US US10/058,841 patent/US6608081B2/en not_active Expired - Lifetime
-
2003
- 2003-01-21 EP EP03705830A patent/EP1470123A1/en not_active Withdrawn
- 2003-01-21 BR BR0307259-2A patent/BR0307259A/pt not_active IP Right Cessation
- 2003-01-21 MX MXPA04007240A patent/MXPA04007240A/es active IP Right Grant
- 2003-01-21 PL PL03371527A patent/PL371527A1/xx not_active Application Discontinuation
- 2003-01-21 CA CA002474718A patent/CA2474718A1/en not_active Abandoned
- 2003-01-21 CN CNA038067897A patent/CN1642949A/zh active Pending
- 2003-01-21 RU RU2004123097/04A patent/RU2004123097A/ru not_active Application Discontinuation
- 2003-01-21 WO PCT/US2003/001673 patent/WO2003064415A1/en not_active Ceased
- 2003-01-21 JP JP2003564038A patent/JP2005520815A/ja active Pending
- 2003-01-21 KR KR10-2004-7011552A patent/KR20040085167A/ko not_active Ceased
- 2003-01-28 MY MYPI20030273A patent/MY134701A/en unknown
- 2003-01-28 AR ARP030100243A patent/AR038326A1/es unknown
- 2003-01-28 TW TW092101784A patent/TW200307679A/zh unknown
- 2003-06-09 US US10/457,271 patent/US6770664B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003064415A1 (en) | 2003-08-07 |
| US6608081B2 (en) | 2003-08-19 |
| US20040067994A1 (en) | 2004-04-08 |
| MY134701A (en) | 2007-12-31 |
| CA2474718A1 (en) | 2003-08-07 |
| JP2005520815A (ja) | 2005-07-14 |
| EP1470123A1 (en) | 2004-10-27 |
| US6770664B2 (en) | 2004-08-03 |
| MXPA04007240A (es) | 2005-03-31 |
| TW200307679A (en) | 2003-12-16 |
| CN1642949A (zh) | 2005-07-20 |
| RU2004123097A (ru) | 2006-01-20 |
| BR0307259A (pt) | 2004-12-07 |
| US20020161029A1 (en) | 2002-10-31 |
| KR20040085167A (ko) | 2004-10-07 |
| PL371527A1 (en) | 2005-06-27 |
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