OA08647A - Dérivés d'imidazole, procédés pour leur préparation et composition pharmaceutique les contenant. - Google Patents
Dérivés d'imidazole, procédés pour leur préparation et composition pharmaceutique les contenant.Info
- Publication number
- OA08647A OA08647A OA59177A OA59177A OA08647A OA 08647 A OA08647 A OA 08647A OA 59177 A OA59177 A OA 59177A OA 59177 A OA59177 A OA 59177A OA 08647 A OA08647 A OA 08647A
- Authority
- OA
- OAPI
- Prior art keywords
- processes
- preparation
- pharmaceutical composition
- composition containing
- imidazole derivatives
- Prior art date
Links
- 150000002460 imidazoles Chemical class 0.000 title 1
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epoxy Resins (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB868619971A GB8619971D0 (en) | 1986-08-15 | 1986-08-15 | Imidazole compounds |
| GB878715932A GB8715932D0 (en) | 1987-07-07 | 1987-07-07 | Imidazole compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| OA08647A true OA08647A (fr) | 1988-11-30 |
Family
ID=26291182
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| OA59177A OA08647A (fr) | 1986-08-15 | 1987-08-14 | Dérivés d'imidazole, procédés pour leur préparation et composition pharmaceutique les contenant. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4822805A (fr) |
| EP (1) | EP0257897A1 (fr) |
| KR (1) | KR880002840A (fr) |
| CN (1) | CN87105680A (fr) |
| AU (1) | AU7682587A (fr) |
| DK (1) | DK425887A (fr) |
| FI (1) | FI873509A7 (fr) |
| HU (1) | HUT44779A (fr) |
| IL (1) | IL83467A0 (fr) |
| NO (1) | NO873432L (fr) |
| OA (1) | OA08647A (fr) |
| PT (1) | PT85531B (fr) |
Families Citing this family (61)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX9300141A (es) * | 1992-01-13 | 1994-07-29 | Smithkline Beecham Corp | Compuestos de imidazol novedosos, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen. |
| US5916891A (en) * | 1992-01-13 | 1999-06-29 | Smithkline Beecham Corporation | Pyrimidinyl imidazoles |
| US5593991A (en) * | 1993-07-16 | 1997-01-14 | Adams; Jerry L. | Imidazole compounds, use and process of making |
| US5593992A (en) * | 1993-07-16 | 1997-01-14 | Smithkline Beecham Corporation | Compounds |
| US5670527A (en) * | 1993-07-16 | 1997-09-23 | Smithkline Beecham Corporation | Pyridyl imidazole compounds and compositions |
| US6426360B1 (en) | 1994-07-28 | 2002-07-30 | G D Searle & Co. | 4,5-substituted imidazolyl compounds for the treatment of inflammation |
| US5620999A (en) * | 1994-07-28 | 1997-04-15 | Weier; Richard M. | Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation |
| US6613789B2 (en) | 1994-07-28 | 2003-09-02 | G. D. Searle & Co. | Heterocyclo-substituted imidazoles for the treatment of inflammation |
| US5616601A (en) * | 1994-07-28 | 1997-04-01 | Gd Searle & Co | 1,2-aryl and heteroaryl substituted imidazolyl compounds for the treatment of inflammation |
| JP2636819B2 (ja) | 1994-12-20 | 1997-07-30 | 日本たばこ産業株式会社 | オキサゾール系複素環式芳香族化合物 |
| EP0828718A1 (fr) | 1995-06-02 | 1998-03-18 | G.D. SEARLE & CO. | Derives heterocyclo-substitues d'acide hydroxamique utilises comme inhibiteurs de la cyclo-oxygenase-2 et de la 5-lipoxygenase |
| US6515014B2 (en) | 1995-06-02 | 2003-02-04 | G. D. Searle & Co. | Thiophene substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors |
| US6512121B2 (en) | 1998-09-14 | 2003-01-28 | G.D. Searle & Co. | Heterocyclo substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors |
| IL118544A (en) | 1995-06-07 | 2001-08-08 | Smithkline Beecham Corp | History of imidazole, the process for their preparation and the pharmaceutical preparations containing them |
| US5739143A (en) * | 1995-06-07 | 1998-04-14 | Smithkline Beecham Corporation | Imidazole compounds and compositions |
| US6369068B1 (en) | 1995-06-07 | 2002-04-09 | Smithkline Beecham Corporation | Amino substituted pyrimidine containing compounds |
| ZA9610687B (en) * | 1995-12-22 | 1997-09-29 | Smithkline Beecham Corp | Novel synthesis. |
| ZA97175B (en) * | 1996-01-11 | 1997-11-04 | Smithkline Beecham Corp | Novel substituted imidazole compounds. |
| US6046208A (en) * | 1996-01-11 | 2000-04-04 | Smithkline Beecham Corporation | Substituted imidazole compounds |
| TR199801361T2 (xx) * | 1996-01-11 | 1998-10-21 | Smithkline Beecham Corporation | Yeni ikameli imidazol bile�imleri. |
| AP9700912A0 (en) | 1996-01-11 | 1997-01-31 | Smithkline Beecham Corp | Novel cycloalkyl substituted imidazoles |
| EP0889888A4 (fr) * | 1996-03-25 | 2003-01-08 | Smithkline Beecham Corp | Nouveau traitement des lesions du systeme nerveux central |
| US6677364B2 (en) * | 1998-04-20 | 2004-01-13 | G.D. Searle & Co. | Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors |
| WO1998007425A1 (fr) | 1996-08-21 | 1998-02-26 | Smithkline Beecham Corporation | Composes d'imidazole, compositions les contenant et leur utilisation |
| US5929076A (en) * | 1997-01-10 | 1999-07-27 | Smithkline Beecham Corporation | Cycloalkyl substituted imidazoles |
| EP1023066A4 (fr) | 1997-06-13 | 2001-05-23 | Smithkline Beecham Corp | Nouveaux composes de pyrazole et de pyrazoline substitues |
| US6610695B1 (en) | 1997-06-19 | 2003-08-26 | Smithkline Beecham Corporation | Aryloxy substituted pyrimidine imidazole compounds |
| US6489325B1 (en) | 1998-07-01 | 2002-12-03 | Smithkline Beecham Corporation | Substituted imidazole compounds |
| AR016294A1 (es) * | 1997-07-02 | 2001-07-04 | Smithkline Beecham Corp | Compuesto de imidazol sustituido, composicion farmaceutica que la contiene, su uso en la fabricacion de un medicamento y procedimiento para supreparacion |
| TW517055B (en) | 1997-07-02 | 2003-01-11 | Smithkline Beecham Corp | Novel substituted imidazole compounds |
| US6562832B1 (en) | 1997-07-02 | 2003-05-13 | Smithkline Beecham Corporation | Substituted imidazole compounds |
| US7301021B2 (en) * | 1997-07-02 | 2007-11-27 | Smithkline Beecham Corporation | Substituted imidazole compounds |
| CA2295762A1 (fr) | 1997-07-02 | 1999-01-14 | Ravi Shanker Garigipati | Nouveaux imidazoles cycloalkyle-substitues |
| IL133731A0 (en) | 1997-07-03 | 2001-04-30 | Neurogen Corp | Certain diarylimidazole derivatives, a new class of npy specific ligands |
| EP1041989A4 (fr) | 1997-10-08 | 2002-11-20 | Smithkline Beecham Corp | Nouveaux composes substitues de cycloalcenyle |
| JP2001526230A (ja) | 1997-12-19 | 2001-12-18 | スミスクライン・ビーチャム・コーポレイション | ヘテロアリール置換イミダゾール化合物、その医薬組成物および使用 |
| WO1999061437A1 (fr) | 1998-05-22 | 1999-12-02 | Smithkline Beecham Corporation | Nouveaux composes d'imidazole a substitution alkyle en position 2 |
| US6858617B2 (en) | 1998-05-26 | 2005-02-22 | Smithkline Beecham Corporation | Substituted imidazole compounds |
| ES2221426T3 (es) * | 1998-08-20 | 2004-12-16 | Smithkline Beecham Corporation | Nuevos compuestos de triazol sustituidos. |
| WO2000025791A1 (fr) * | 1998-11-04 | 2000-05-11 | Smithkline Beecham Corporation | Pyrazines substitues pyridin-4-yle ou pyrimidin-4-yle |
| US6239279B1 (en) | 1998-12-16 | 2001-05-29 | Smithkline Beecham Corporation | Synthesis for 4-aryl-5-pyrimidine imidazole substituted derivatives |
| DE60020595T2 (de) | 1999-11-23 | 2006-03-16 | Smithkline Beecham Corp. | 3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p38-kinase-inhibitoren |
| AU1781601A (en) | 1999-11-23 | 2001-06-04 | Smithkline Beecham Corporation | 3,4-dihydro-(1h)quinazolin-2-one compounds as csbp/p38 kinase inhibitors |
| US6759410B1 (en) * | 1999-11-23 | 2004-07-06 | Smithline Beecham Corporation | 3,4-dihydro-(1H)-quinazolin-2-ones and their use as CSBP/p38 kinase inhibitors |
| AU1782301A (en) | 1999-11-23 | 2001-06-04 | Smithkline Beecham Corporation | 3,4-dihydro-(1h)quinazolin-2-one compounds as csbp/p39 kinase inhibitors |
| SK8452002A3 (en) | 1999-12-16 | 2002-11-06 | Schering Corp | Substituted 4-(phenyl or pyridyl)imidazole derivatives, pharmaceutical composition comprising the same and use thereof |
| US7235551B2 (en) * | 2000-03-02 | 2007-06-26 | Smithkline Beecham Corporation | 1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases |
| KR100850812B1 (ko) * | 2000-10-23 | 2008-08-06 | 스미스클라인 비참 코포레이션 | 신규 화합물 |
| US20030105144A1 (en) | 2001-04-17 | 2003-06-05 | Ping Gao | Stabilized oral pharmaceutical composition |
| US6673818B2 (en) | 2001-04-20 | 2004-01-06 | Pharmacia Corporation | Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation |
| US7329401B2 (en) * | 2002-04-15 | 2008-02-12 | The Regents Of The University Of California | Cyclooxygenase-2 selective agents useful as imaging probes and related methods |
| EP1532118A2 (fr) * | 2002-07-05 | 2005-05-25 | Axxima Pharmaceuticals Aktiengesellschaft | Composes d'imidazole pour le traitement des infections par le virus de l'hepatite c |
| ES2325687T3 (es) | 2002-09-18 | 2009-09-14 | Pfizer Products Inc. | Compuestos de imidazol novedosos como inhibidores del factor de crecimiento transformante (tgf). |
| PA8595001A1 (es) | 2003-03-04 | 2004-09-28 | Pfizer Prod Inc | Nuevos compuestos heteroaromaticos condensados que son inhibidores del factor de crecimiento transforante (tgf) |
| WO2004099130A2 (fr) * | 2003-05-08 | 2004-11-18 | Astellas Pharma Inc. | Inhibiteur de cox |
| AU2006229995A1 (en) * | 2005-03-25 | 2006-10-05 | Glaxo Group Limited | Process for preparing pyrido(2,3-d)pyrimidin-7-one and 3,4-dihydropyrimido(4,5-d)pyrimidin-2(1H)-one derivatives |
| PE20061351A1 (es) | 2005-03-25 | 2007-01-14 | Glaxo Group Ltd | COMPUESTOS 8H-PIRIDO[2,3-d]PIRIMIDIN-7-ONA 2,4,8-TRISUSTITUIDOS COMO INHIBIDORES DE LA QUINASA CSBP/RK/p38 |
| US7728027B2 (en) * | 2007-08-08 | 2010-06-01 | Bristol-Myers Squibb Company | Process for synthesizing compounds useful for treating hepatitis C |
| SG2014014013A (en) | 2008-09-22 | 2014-07-30 | Cayman Chemical Co Inc | Multiheteroaryl compounds as inhibitors of h-pgds and their use for treating prostaglandin d2 mediated diseases |
| US9988366B2 (en) * | 2014-03-28 | 2018-06-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| KR102447094B1 (ko) * | 2014-08-13 | 2022-09-23 | 닛뽕소다 가부시키가이샤 | 디아릴이미다졸 화합물 및 유해 생물 방제제 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3707475A (en) * | 1970-11-16 | 1972-12-26 | Pfizer | Antiinflammatory imidazoles |
| CH561716A5 (fr) * | 1971-05-10 | 1975-05-15 | Ciba Geigy Ag | |
| US3929807A (en) * | 1971-05-10 | 1975-12-30 | Ciba Geigy Corp | 2-Substituted-4(5)-(aryl)-5(4)-(2,3 or -4-pyridyl)-imidazoles |
| SE7601713L (sv) * | 1975-03-03 | 1976-09-06 | Merck & Co Inc | Nya, substituerad imidazoler |
| US4440774A (en) * | 1975-03-03 | 1984-04-03 | Merck & Co., Inc. | 3-Amino-2-hydroxypropoxyaryl imidazole derivatives |
-
1987
- 1987-08-06 IL IL83467A patent/IL83467A0/xx unknown
- 1987-08-07 EP EP87307051A patent/EP0257897A1/fr not_active Withdrawn
- 1987-08-12 AU AU76825/87A patent/AU7682587A/en not_active Abandoned
- 1987-08-13 US US07/084,862 patent/US4822805A/en not_active Expired - Fee Related
- 1987-08-13 PT PT85531A patent/PT85531B/pt unknown
- 1987-08-13 FI FI873509A patent/FI873509A7/fi not_active Application Discontinuation
- 1987-08-14 HU HU873676A patent/HUT44779A/hu unknown
- 1987-08-14 NO NO873432A patent/NO873432L/no unknown
- 1987-08-14 DK DK425887A patent/DK425887A/da not_active Application Discontinuation
- 1987-08-14 CN CN198787105680A patent/CN87105680A/zh active Pending
- 1987-08-14 KR KR1019870008953A patent/KR880002840A/ko not_active Withdrawn
- 1987-08-14 OA OA59177A patent/OA08647A/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK425887A (da) | 1988-02-16 |
| KR880002840A (ko) | 1988-05-11 |
| PT85531B (en) | 1989-12-15 |
| CN87105680A (zh) | 1988-04-27 |
| AU7682587A (en) | 1988-02-18 |
| FI873509L (fi) | 1988-02-16 |
| HUT44779A (en) | 1988-04-28 |
| EP0257897A1 (fr) | 1988-03-02 |
| IL83467A0 (en) | 1988-01-31 |
| FI873509A0 (fi) | 1987-08-13 |
| NO873432D0 (no) | 1987-08-14 |
| PT85531A (en) | 1987-09-01 |
| DK425887D0 (da) | 1987-08-14 |
| NO873432L (no) | 1988-02-16 |
| US4822805A (en) | 1989-04-18 |
| FI873509A7 (fi) | 1988-02-16 |
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