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NO941726L - Fremgangsmåte for fremstilling av 4-amino-1-hydroxy-butyliden-1,2-bisfosfonsyre - Google Patents

Fremgangsmåte for fremstilling av 4-amino-1-hydroxy-butyliden-1,2-bisfosfonsyre

Info

Publication number
NO941726L
NO941726L NO941726A NO941726A NO941726L NO 941726 L NO941726 L NO 941726L NO 941726 A NO941726 A NO 941726A NO 941726 A NO941726 A NO 941726A NO 941726 L NO941726 L NO 941726L
Authority
NO
Norway
Prior art keywords
amino
preparation
butylidene
hydroxy
bisphosphonic acid
Prior art date
Application number
NO941726A
Other languages
English (en)
Other versions
NO941726D0 (no
NO178228B (no
NO178228C (no
Inventor
Gerald R Kieczykowski
Ronald B Jobson
David G Melillo
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23431886&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO941726(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of NO941726L publication Critical patent/NO941726L/no
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Priority to NO941726A priority Critical patent/NO178228C/no
Publication of NO941726D0 publication Critical patent/NO941726D0/no
Publication of NO178228B publication Critical patent/NO178228B/no
Publication of NO178228C publication Critical patent/NO178228C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Seasonings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO941726A 1989-06-09 1994-05-09 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter NO178228C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO941726A NO178228C (no) 1989-06-09 1994-05-09 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US07/363,820 US4922007A (en) 1989-06-09 1989-06-09 Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof
NO902559A NO177997C (no) 1989-06-09 1990-06-08 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,1-bisfosfonsyre
NO941726A NO178228C (no) 1989-06-09 1994-05-09 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter

Publications (4)

Publication Number Publication Date
NO941726L true NO941726L (no) 1990-12-10
NO941726D0 NO941726D0 (no) 1994-05-09
NO178228B NO178228B (no) 1995-11-06
NO178228C NO178228C (no) 1996-02-14

Family

ID=23431886

Family Applications (2)

Application Number Title Priority Date Filing Date
NO902559A NO177997C (no) 1989-06-09 1990-06-08 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,1-bisfosfonsyre
NO941726A NO178228C (no) 1989-06-09 1994-05-09 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO902559A NO177997C (no) 1989-06-09 1990-06-08 Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,1-bisfosfonsyre

Country Status (23)

Country Link
US (1) US4922007A (no)
EP (1) EP0402152B1 (no)
JP (2) JPH0662651B2 (no)
KR (1) KR0137455B1 (no)
AT (1) ATE129713T1 (no)
AU (1) AU625704C (no)
CA (1) CA2018477C (no)
CH (1) CH0402152H1 (no)
CY (1) CY1894A (no)
DE (1) DE69023280T2 (no)
DK (1) DK0402152T3 (no)
ES (1) ES2080116T3 (no)
FI (1) FI93219C (no)
GR (1) GR3018379T3 (no)
HK (1) HK69596A (no)
HU (1) HU211908A9 (no)
IE (1) IE69564B1 (no)
IL (1) IL94612A (no)
LV (1) LV11472B (no)
NO (2) NO177997C (no)
NZ (1) NZ233972A (no)
PT (1) PT94306B (no)
ZA (1) ZA904446B (no)

Families Citing this family (118)

* Cited by examiner, † Cited by third party
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LV11472B (en) 1996-12-20
AU625704B2 (en) 1992-07-16
FI93219C (fi) 1995-03-10
EP0402152A2 (en) 1990-12-12
PT94306B (pt) 1997-05-28
GR3018379T3 (en) 1996-03-31
ZA904446B (en) 1992-06-24
KR910000768A (ko) 1991-01-30
NO177997C (no) 1996-01-03
ES2080116T3 (es) 1996-02-01
IE902073L (en) 1990-12-09
JPH03101684A (ja) 1991-04-26
IL94612A (en) 1995-03-30
DE69023280D1 (de) 1995-12-07
NO941726D0 (no) 1994-05-09
IL94612A0 (en) 1991-04-15
NO178228B (no) 1995-11-06
PT94306A (pt) 1991-02-08
KR0137455B1 (ko) 1998-05-01
JPH0748391A (ja) 1995-02-21
CH0402152H1 (fr) 2006-02-28
CA2018477C (en) 1995-08-01
JPH0662651B2 (ja) 1994-08-17
DE69023280T2 (de) 1996-06-20
EP0402152B1 (en) 1995-11-02
CA2018477A1 (en) 1990-12-09
AU5701990A (en) 1990-12-13
CY1894A (en) 1990-06-08
EP0402152A3 (en) 1991-07-03
NZ233972A (en) 1992-05-26
AU625704C (en) 2001-07-26
US4922007A (en) 1990-05-01
DK0402152T3 (da) 1995-12-04
NO902559L (no) 1990-12-10
HU211908A9 (en) 1996-01-29
NO178228C (no) 1996-02-14
FI902845A0 (fi) 1990-06-07
IE69564B1 (en) 1996-10-02
HK69596A (en) 1996-04-26
ATE129713T1 (de) 1995-11-15
NO902559D0 (no) 1990-06-08
NO177997B (no) 1995-09-25
LV11472A (lv) 1996-08-20
FI93219B (fi) 1994-11-30

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