NO323077B1 - Forbindelse, farmasoytisk preparat, nevnte forbindelse eller preparat for medisinsk bruk samt anvendelse av nevnte forbindelse for fremstilling av et medikament for medisinsk behandling. - Google Patents

Forbindelse, farmasoytisk preparat, nevnte forbindelse eller preparat for medisinsk bruk samt anvendelse av nevnte forbindelse for fremstilling av et medikament for medisinsk behandling. Download PDF

Info

Publication number: NO323077B1
Authority: NO; Norway
Prior art keywords: methyl; indole; hydroxy; carboxamide; formula
Prior art date: 1999-11-03

Application number

NO20022105A

Other languages

English (en)

Norwegian (no)

Other versions

NO20022105D0 (no

NO20022105L (no

Inventor

Curley David

James Rosamund

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-11-03

Filing date

2002-05-02

Publication date

2006-12-27

2002-05-02 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2002-05-02 Publication of NO20022105D0 publication Critical patent/NO20022105D0/no

2002-07-02 Publication of NO20022105L publication Critical patent/NO20022105L/no

2006-12-27 Publication of NO323077B1 publication Critical patent/NO323077B1/no

Links

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125000004178 (C1-C4) alkyl group Chemical group 0.000 claims description 2
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PUOAEBLNCXMRLA-UHFFFAOYSA-N 4-hydroxy-N,N-dimethyl-1H-indole-2-carboxamide Chemical compound CN(C(=O)C=1NC2=CC=CC(=C2C1)O)C PUOAEBLNCXMRLA-UHFFFAOYSA-N 0.000 claims description 2
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Classifications

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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C—CHEMISTRY; METALLURGY
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- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
General Chemical & Material Sciences (AREA)
Psychiatry (AREA)
Epidemiology (AREA)
Addiction (AREA)
Psychology (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Indole Compounds (AREA)
Pyridine Compounds (AREA)

NO20022105A 1999-11-03 2002-05-02 Forbindelse, farmasoytisk preparat, nevnte forbindelse eller preparat for medisinsk bruk samt anvendelse av nevnte forbindelse for fremstilling av et medikament for medisinsk behandling. NO323077B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE9903998A SE9903998D0 (sv)	1999-11-03	1999-11-03	New compounds
PCT/SE2000/002147 WO2001032622A1 (en)	1999-11-03	2000-11-01	Positive modulators of nicotinic receptor agonists

Publications (3)

Publication Number	Publication Date
NO20022105D0 NO20022105D0 (no)	2002-05-02
NO20022105L NO20022105L (no)	2002-07-02
NO323077B1 true NO323077B1 (no)	2006-12-27

Family

ID=20417608

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20022105A NO323077B1 (no)	1999-11-03	2002-05-02	Forbindelse, farmasoytisk preparat, nevnte forbindelse eller preparat for medisinsk bruk samt anvendelse av nevnte forbindelse for fremstilling av et medikament for medisinsk behandling.

Country Status (16)

Country	Link
US (2)	US7064143B1 (es)
EP (1)	EP1230218A1 (es)
JP (1)	JP2003513073A (es)
KR (1)	KR20020063175A (es)
CN (1)	CN1216864C (es)
AU (1)	AU783602B2 (es)
BR (1)	BR0015193A (es)
CA (1)	CA2387741A1 (es)
CO (1)	CO5280079A1 (es)
IL (1)	IL149096A0 (es)
MX (1)	MXPA02004240A (es)
NO (1)	NO323077B1 (es)
NZ (1)	NZ518449A (es)
SE (1)	SE9903998D0 (es)
WO (1)	WO2001032622A1 (es)
ZA (1)	ZA200203181B (es)

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US7226942B2 (en)	2004-11-15	2007-06-05	Bristol-Myers Squibb Company	2-amino-4-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
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FR2888847B1 (fr)	2005-07-22	2007-08-31	Sanofi Aventis Sa	Derives de n-(heteriaryl)-1-heteorarylalkyl-1h-indole-2- carboxamides, leur preparation et application en therapeutique
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KR101026570B1 (ko)	2005-11-30	2011-03-31	에프. 호프만-라 로슈 아게	3-아미노-1-아릴프로필 아자인돌 및 이의 용도
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US8383657B2 (en)	2007-12-21	2013-02-26	Abbott Laboratories	Thiazolylidine urea and amide derivatives and methods of use thereof
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1999
- 1999-11-03 SE SE9903998A patent/SE9903998D0/xx unknown
2000
- 2000-11-01 MX MXPA02004240A patent/MXPA02004240A/es not_active Application Discontinuation
- 2000-11-01 EP EP00976499A patent/EP1230218A1/en not_active Withdrawn
- 2000-11-01 CN CN008154406A patent/CN1216864C/zh not_active Expired - Fee Related
- 2000-11-01 IL IL14909600A patent/IL149096A0/xx unknown
- 2000-11-01 AU AU14263/01A patent/AU783602B2/en not_active Ceased
- 2000-11-01 KR KR1020027005705A patent/KR20020063175A/ko not_active Ceased
- 2000-11-01 WO PCT/SE2000/002147 patent/WO2001032622A1/en not_active Ceased
- 2000-11-01 NZ NZ518449A patent/NZ518449A/en unknown
- 2000-11-01 US US10/111,029 patent/US7064143B1/en not_active Expired - Fee Related
- 2000-11-01 BR BR0015193-9A patent/BR0015193A/pt not_active IP Right Cessation
- 2000-11-01 JP JP2001534774A patent/JP2003513073A/ja not_active Abandoned
- 2000-11-01 CO CO00083137A patent/CO5280079A1/es not_active Application Discontinuation
- 2000-11-01 CA CA002387741A patent/CA2387741A1/en not_active Abandoned
2002
- 2002-04-22 ZA ZA200203181A patent/ZA200203181B/xx unknown
- 2002-05-02 NO NO20022105A patent/NO323077B1/no unknown
2005
- 2005-07-11 US US11/178,668 patent/US7402604B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU1426301A (en)	2001-05-14
NO20022105D0 (no)	2002-05-02
BR0015193A (pt)	2002-06-18
IL149096A0 (en)	2002-11-10
MXPA02004240A (es)	2002-10-17
CN1387513A (zh)	2002-12-25
WO2001032622A1 (en)	2001-05-10
US20050245595A1 (en)	2005-11-03
US7064143B1 (en)	2006-06-20
EP1230218A1 (en)	2002-08-14
SE9903998D0 (sv)	1999-11-03
CN1216864C (zh)	2005-08-31
US7402604B2 (en)	2008-07-22
ZA200203181B (en)	2003-07-22
NZ518449A (en)	2004-07-30
CA2387741A1 (en)	2001-05-10
CO5280079A1 (es)	2003-05-30
NO20022105L (no)	2002-07-02
JP2003513073A (ja)	2003-04-08
KR20020063175A (ko)	2002-08-01
AU783602B2 (en)	2005-11-10

Publication	Publication Date	Title
NO323077B1 (no)	2006-12-27	Forbindelse, farmasoytisk preparat, nevnte forbindelse eller preparat for medisinsk bruk samt anvendelse av nevnte forbindelse for fremstilling av et medikament for medisinsk behandling.
AU783507B2 (en)	2005-11-03	Positive modulators of nicotinic receptor agonists
EP0593559A1 (en)	1994-04-27	Aromatic compounds, pharmaceutical compositions containing them and their use in therapy
AU2595095A (en)	1996-01-04	Tachykinin (nk1) receptor antagonists
HRP20000847A2 (en)	2001-12-31	4,5,6 i 7 - INDOLE AND INDOLINE DERIVATIVES, THEIR PREPARATION AND USE
ZA200508860B (en)	2007-03-28	Positive modulators of nicotinic acetylcholine receptors
US20080081833A1 (en)	2008-04-03	Novel Pyrazole Derivatives And Their Use As Modulators Of Nicotinic Acetylcholine Receptors
JP2022547079A (ja)	2022-11-10	てんかんを治療する方法を使用しててんかんを治療する方法
JP2014514259A (ja)	2014-06-19	疼痛および他の障害の処置のための化合物および方法
KR20080007046A (ko)	2008-01-17	멜라노코틴 수용체의 항진제
JP2011509285A (ja)	2011-03-24	疼痛治療のためのカンナビノイド受容体のリガンドとしてのプロリン類似体
EP1230217B1 (en)	2005-10-05	Positive modulators of nicotinic receptor agonists
KR20160077153A (ko)	2016-07-01	Nmda 수용체 조절인자 및 이들의 전구약물, 염, 그리고 용도
ES2461520T3 (es)	2014-05-20	Modulador de receptores de andrógenos y sus usos
RU2637928C2 (ru)	2017-12-08	Производные арилциклоалкиламинов, нейропротектор (варианты), вещество, обладающее сочетанным нейропротекторным, анальгетическим и антидепрессивным действием, фармацевтические композиции на его основе
TW202045477A (zh)	2020-12-16	用於治療腦機能障礙的氮呯-吲哚及其他雜環
NO162763B (no)	1989-11-06	Analogifremgangsmaate for fremstilling av terapeutisk aktive indol-derivater.
DK165976B (da)	1993-02-22	5-aminosulfonyl-methyl-indolderivater og farmaceutiske praeparater med indhold deraf